KR930007263B1 - 세프-3-엠-4-카르복실산 유도체의 제조방법 - Google Patents

세프-3-엠-4-카르복실산 유도체의 제조방법 Download PDF

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Publication number
KR930007263B1
KR930007263B1 KR1019860005723A KR860005723A KR930007263B1 KR 930007263 B1 KR930007263 B1 KR 930007263B1 KR 1019860005723 A KR1019860005723 A KR 1019860005723A KR 860005723 A KR860005723 A KR 860005723A KR 930007263 B1 KR930007263 B1 KR 930007263B1
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KR
South Korea
Prior art keywords
chloro
carboxylic acid
methyl
thiomethyl
acetamido
Prior art date
Application number
KR1019860005723A
Other languages
English (en)
Korean (ko)
Other versions
KR870001219A (ko
Inventor
엘렉 산도르
마로시 카탈린
미호크 미클로스
미호크 일디코
얀크소 산도르
코바크스 이스트반
코냐 마리아
키스 일로나
렘페르트 카롤리
돌레스칼 가보르
페테르 조세프
호르냑 귤라
니트라이 조세프
시미그 귤라
자우에르 카롤리
콤보스 스잔나
Original Assignee
비오갈 교기쎄르 기아르
이스트반 체르누스, 바르나코크사르
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 비오갈 교기쎄르 기아르, 이스트반 체르누스, 바르나코크사르 filed Critical 비오갈 교기쎄르 기아르
Publication of KR870001219A publication Critical patent/KR870001219A/ko
Application granted granted Critical
Publication of KR930007263B1 publication Critical patent/KR930007263B1/ko

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36—Methylene radicals, substituted by sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04—Five-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1019860005723A 1985-07-16 1986-07-15 세프-3-엠-4-카르복실산 유도체의 제조방법 KR930007263B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
HU2725 1985-07-16
HU2251/2725 1985-07-16
HU852725A HU203243B (en) 1985-07-16 1985-07-16 Process for producing cefalosporin derivative

Publications (2)

Publication Number Publication Date
KR870001219A KR870001219A (ko) 1987-03-12
KR930007263B1 true KR930007263B1 (ko) 1993-08-04

Family

ID=10960853

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019860005723A KR930007263B1 (ko) 1985-07-16 1986-07-15 세프-3-엠-4-카르복실산 유도체의 제조방법

Country Status (14)

Country Link
JP (1) JPS6222787A (it)
KR (1) KR930007263B1 (it)
CN (1) CN1012614B (it)
AT (1) AT389877B (it)
BE (1) BE905113A (it)
DE (1) DE3623900A1 (it)
FI (1) FI83877C (it)
FR (1) FR2591598B1 (it)
GB (1) GB2177696B (it)
GR (1) GR861855B (it)
HU (1) HU203243B (it)
IL (1) IL79410A0 (it)
IT (1) IT1196494B (it)
NL (1) NL8601842A (it)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2012729C (en) 1989-04-07 1997-05-20 Takashi Kuroda Dulled stretched molding and process for producing the same
JP2893286B2 (ja) * 1990-05-17 1999-05-17 グンゼ株式会社 熱収縮性発泡複合フィルム及びその製法
JP2515295Y2 (ja) * 1993-06-30 1996-10-30 株式会社川崎製作所 管継手
KR100408343B1 (ko) * 2001-11-01 2003-12-06 주식회사 이앤티 자돈의 항상성(Homeostasis)을 유지시킬 수 있는 사료 및그 제조방법

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7402778A (it) * 1973-03-02 1974-09-04
JPS539787A (en) * 1976-07-16 1978-01-28 Yamanouchi Pharmaceut Co Ltd Novel cephalosporin derivatives and their preparation

Also Published As

Publication number Publication date
FI83877B (fi) 1991-05-31
HUT48890A (en) 1989-07-28
DE3623900A1 (de) 1987-01-29
BE905113A (fr) 1986-11-03
CN86104805A (zh) 1987-02-18
FI862965A (fi) 1987-01-17
GB8617181D0 (en) 1986-08-20
GR861855B (en) 1986-11-18
IT8621135A0 (it) 1986-07-15
IL79410A0 (en) 1986-10-31
NL8601842A (nl) 1987-02-16
GB2177696A (en) 1987-01-28
IT1196494B (it) 1988-11-16
KR870001219A (ko) 1987-03-12
ATA192686A (de) 1989-07-15
AT389877B (de) 1990-02-12
FI83877C (fi) 1991-09-10
FR2591598A1 (fr) 1987-06-19
JPS6222787A (ja) 1987-01-30
CN1012614B (zh) 1991-05-15
GB2177696B (en) 1989-01-05
FR2591598B1 (fr) 1990-01-26
HU203243B (en) 1991-06-28
FI862965A0 (fi) 1986-07-16

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