KR880002013B1 - 1-[3-(6-플루오로-1,2-벤즈이속사졸-3-일)프로필]-4-(치환된)-피페라진 및 이의 제조방법 - Google Patents

1-[3-(6-플루오로-1,2-벤즈이속사졸-3-일)프로필]-4-(치환된)-피페라진 및 이의 제조방법 Download PDF

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Publication number
KR880002013B1
KR880002013B1 KR8204814A KR820004814A KR880002013B1 KR 880002013 B1 KR880002013 B1 KR 880002013B1 KR 8204814 A KR8204814 A KR 8204814A KR 820004814 A KR820004814 A KR 820004814A KR 880002013 B1 KR880002013 B1 KR 880002013B1
Authority
KR
South Korea
Prior art keywords
compound
fluoro
propyl
benzisoxazol
piperazine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
KR8204814A
Other languages
English (en)
Korean (ko)
Other versions
KR840001974A (ko
Inventor
데이비스 래리
토마스 클레인 죠셉
Original Assignee
마크 에드워드 로가트
훽스트-러셀 파마슈티칼 인코포레이티드
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/366,248 external-priority patent/US4536578A/en
Priority claimed from US06/366,244 external-priority patent/US4390544A/en
Application filed by 마크 에드워드 로가트, 훽스트-러셀 파마슈티칼 인코포레이티드 filed Critical 마크 에드워드 로가트
Publication of KR840001974A publication Critical patent/KR840001974A/ko
Priority to KR1019880010742A priority Critical patent/KR880002511B1/ko
Application granted granted Critical
Publication of KR880002013B1 publication Critical patent/KR880002013B1/ko
Expired legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
KR8204814A 1982-04-09 1982-10-26 1-[3-(6-플루오로-1,2-벤즈이속사졸-3-일)프로필]-4-(치환된)-피페라진 및 이의 제조방법 Expired KR880002013B1 (ko)

Priority Applications (1)

Application Number Priority Date Filing Date Title
KR1019880010742A KR880002511B1 (ko) 1982-04-09 1988-08-24 1-[3-(6-플루오로-1,2-벤즈이속사졸-3-일)프로필]-4-(치환된)-피페리딘 및 이의 제조방법

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US06/366,248 US4536578A (en) 1982-04-09 1982-04-09 1-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines
US06/366,244 US4390544A (en) 1982-04-09 1982-04-09 {1-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(2-oxo-1-benzimidazolinyl}p
US366,248 1982-04-09
US366,244 1982-04-09

Related Child Applications (1)

Application Number Title Priority Date Filing Date
KR1019880010742A Division KR880002511B1 (ko) 1982-04-09 1988-08-24 1-[3-(6-플루오로-1,2-벤즈이속사졸-3-일)프로필]-4-(치환된)-피페리딘 및 이의 제조방법

Publications (2)

Publication Number Publication Date
KR840001974A KR840001974A (ko) 1984-06-07
KR880002013B1 true KR880002013B1 (ko) 1988-10-12

Family

ID=27003274

Family Applications (1)

Application Number Title Priority Date Filing Date
KR8204814A Expired KR880002013B1 (ko) 1982-04-09 1982-10-26 1-[3-(6-플루오로-1,2-벤즈이속사졸-3-일)프로필]-4-(치환된)-피페라진 및 이의 제조방법

Country Status (16)

Country Link
EP (1) EP0091511B1 (enExample)
KR (1) KR880002013B1 (enExample)
AT (1) ATE34170T1 (enExample)
CA (1) CA1209146A (enExample)
DE (1) DE3278471D1 (enExample)
DK (1) DK474382A (enExample)
ES (1) ES516830A0 (enExample)
FI (1) FI823433A7 (enExample)
GR (1) GR77706B (enExample)
HU (1) HU191075B (enExample)
IE (1) IE54065B1 (enExample)
IL (1) IL66866A (enExample)
NO (1) NO823556L (enExample)
NZ (1) NZ202044A (enExample)
PH (1) PH18252A (enExample)
PT (1) PT75726A (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2807577B2 (ja) * 1990-06-15 1998-10-08 エーザイ株式会社 環状アミド誘導体
US5055476A (en) * 1990-08-13 1991-10-08 Hoechst-Roussel Pharmaceuticals Incorporated 3-(1,2-benzisoxazol-3-yl)-4-pyridinamines and derivatives
US5114936A (en) * 1990-08-23 1992-05-19 Hoechst-Roussel Pharmaceuticals Incorporated 6,7-dihydro-3-phenyl-1,2-benzisoxazol-4(5h)-ones and -ols, compositions and pharmaceutical use
ES2188584T3 (es) * 1991-03-28 2003-07-01 Eisai Co Ltd Derivados heterociclicos de amina.
US5750542A (en) 1993-09-28 1998-05-12 Pfizer Benzisoxazole and benzisothizole derivatives as cholinesterase inhibitors
US5225412A (en) * 1991-04-29 1993-07-06 Hoechst-Roussel Pharmaceuticals Incorporated Benzoisothiazole-and benzisoxazole-3-carboxamides
US5143923B1 (en) * 1991-04-29 1993-11-02 Hoechst-Roussel Pharmaceuticals Incorporated Benzoisothiazole-and benzisoxazole-3-carboxamides
MX377708B (es) * 2012-12-19 2025-03-11 Henkel Ag & Co Kgaa Método para la amortiguación de sonido y/o aislamiento de sonido de componentes.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI60390C (fi) * 1975-03-05 1982-01-11 Sumitomo Chemical Co Foerfarande foer framstaellning av neuroleptiska butyrofenoner
JPS6043064B2 (ja) * 1979-11-28 1985-09-26 ウェルファイド株式会社 新規イソオキサゾ−ル誘導体

Also Published As

Publication number Publication date
CA1209146A (en) 1986-08-05
IE822558L (en) 1983-10-09
FI823433L (fi) 1983-10-10
IE54065B1 (en) 1989-06-07
ES8400431A1 (es) 1983-10-16
IL66866A0 (en) 1982-12-31
FI823433A0 (fi) 1982-10-08
KR840001974A (ko) 1984-06-07
ES516830A0 (es) 1983-10-16
DE3278471D1 (en) 1988-06-16
EP0091511A3 (en) 1984-12-12
HU191075B (en) 1987-01-28
IL66866A (en) 1987-08-31
EP0091511A2 (en) 1983-10-19
PH18252A (en) 1985-05-13
NZ202044A (en) 1987-04-30
PT75726A (en) 1982-11-01
FI823433A7 (fi) 1983-10-10
EP0091511B1 (en) 1988-05-11
GR77706B (enExample) 1984-09-25
NO823556L (no) 1983-10-10
ATE34170T1 (de) 1988-05-15
DK474382A (da) 1983-10-10

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