KR850003399A - 치환된 5-아실아미노-1-페닐피라졸의 제조방법 - Google Patents

치환된 5-아실아미노-1-페닐피라졸의 제조방법 Download PDF

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KR850003399A
KR850003399A KR1019840006345A KR840006345A KR850003399A KR 850003399 A KR850003399 A KR 850003399A KR 1019840006345 A KR1019840006345 A KR 1019840006345A KR 840006345 A KR840006345 A KR 840006345A KR 850003399 A KR850003399 A KR 850003399A
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South Korea
Prior art keywords
cyano
phenylpyrazole
acylamino
halogenoalkyl
alkoxycarbonyl
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KR1019840006345A
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English (en)
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KR900007179B1 (ko
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게링 라인홀트 (외 5)
Original Assignee
귄터 피터스,하인쯔-게르트 믈러
바이엘 아크티엔 게젤샤프트
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Publication of KR850003399A publication Critical patent/KR850003399A/ko
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Publication of KR900007179B1 publication Critical patent/KR900007179B1/ko

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C243/00—Compounds containing chains of nitrogen atoms singly-bound to each other, e.g. hydrazines, triazanes
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • C07D231/40—Acylated on said nitrogen atom

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Lubricants (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

내용 없음

Description

치환된 5-아실아미노-1-페닐피라졸의 제조방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (2)

  1. 다음 일반식(II)의 5-아미노피라졸을 다음 일반식(III)의 아실화제와, 필요시 희석제 존재하 및 필요시 산 결합제 존재하에 반응시킴을 특징으로 하여, 다음 일반식(I)의 치환된 5-아실아미노-1-페닐피라졸을 제조하는 방법.
    상기식에서, R1은 시아노, 알콕시카보닐, 알케닐옥시카보닐, 알킬옥시카보닐, 알킬아미노카보닐, 알케닐아미노카보닐 또는 알키닐아미노카보닐이고, R2는 수소, 알킬, 알케닐, 알키닐, 임의 치환된 시클로알킬, 알콕시알킬, 알킬티오알킬, 할로게노알킬 또는 임의 치환된 아릴이고, R3, R4, R5, R6및 R7은 같거나 다르며, 수소, 할로겐, 시아노, 니트로, 알킬, 알콕시, 알킬설포닐, 알콕시카보닐 또는 라디칼-(X)n-R8(여기에서 X는 산소, 황, 설피닐 또는 설포닐이고, n은 0 또는 1이고 R8은 할로게노알킬이다)이고, A는 활성화 이탈 그룹이고, 단, 라디칼, R3, R4, R5, R6또는 R7중 적어도 하나가 -(X)N-R8이나, R5가 트리플루오로메틸일 경우 R1은 시아노가 아니다.
  2. 제1항에 있어서, 5-프로피오닐아미노-4-시아노-1-(2, 6-디클로로-4-트리플루오로메틸티오-페닐)-페라졸의 제조방법.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019840006345A 1983-10-15 1984-10-13 치환된 5-아실아미노-1-페닐피라졸의 제조방법 KR900007179B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
DE3337543 1983-10-15
DEP3337543.7 1983-10-15
DE3337543.7 1983-10-15
DE3420985.9 1984-06-06
DE19843420985 DE3420985A1 (de) 1983-10-15 1984-06-06 Substituierte 5-acylamino-1-phenylpyrazole

Publications (2)

Publication Number Publication Date
KR850003399A true KR850003399A (ko) 1985-06-17
KR900007179B1 KR900007179B1 (ko) 1990-09-29

Family

ID=25814889

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019840006345A KR900007179B1 (ko) 1983-10-15 1984-10-13 치환된 5-아실아미노-1-페닐피라졸의 제조방법

Country Status (16)

Country Link
US (4) US4668280A (ko)
EP (1) EP0138149B1 (ko)
KR (1) KR900007179B1 (ko)
AT (1) ATE40120T1 (ko)
AU (1) AU569916B2 (ko)
BR (1) BR8405151A (ko)
CA (1) CA1233473A (ko)
DD (1) DD228157A5 (ko)
DE (2) DE3420985A1 (ko)
DK (1) DK491384A (ko)
ES (1) ES8506638A1 (ko)
GR (1) GR80631B (ko)
HU (1) HU196030B (ko)
IL (3) IL83364A (ko)
NZ (1) NZ209874A (ko)
TR (1) TR23212A (ko)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3423582A1 (de) * 1984-06-27 1986-01-09 Bayer Ag, 5090 Leverkusen Substituierte 5-acylamino-1-phenylpyrazole
DE3426424A1 (de) * 1984-07-18 1986-01-23 Bayer Ag, 5090 Leverkusen Substituierte 5-amino-1-phenylpyrazole
DE3447211A1 (de) * 1984-12-22 1986-06-26 Bayer Ag, 5090 Leverkusen Verfahren zur herstellung von substituierten phenylhydrazinen
US4752326A (en) * 1985-05-15 1988-06-21 Hokko Chemical Industry Co., Ltd. 1-arylpyrazoles, composition containing them, and herbicidal method of using them
DE3520331A1 (de) * 1985-06-07 1986-12-11 Bayer Ag, 5090 Leverkusen 1-aryl-5-alkoximinoalkylamino-pyrazole
DE3539844A1 (de) 1985-11-09 1987-05-14 Bayer Ag Substituierte 5-amino-1-aryl-pyrazole
DE3603291A1 (de) * 1986-02-04 1987-08-06 Bayer Ag 5-amino-1-phenyl-pyrazole
DE3631003A1 (de) * 1986-09-12 1988-03-24 Bayer Ag Verfahren zur herstellung von 4-substituierten 1-aryl-5-amino-pyrazolen
US5167691A (en) * 1991-10-03 1992-12-01 Fmc Corporation Herbicidal 5-amino-1-phenyl pyrazole compounds
US5198014A (en) * 1991-11-20 1993-03-30 Fmc Corporation Herbicidal beta-pyrazolylacrylic acid compound
US5556873A (en) * 1993-02-24 1996-09-17 Rhone-Poulenc Inc. Pesticidal 1-aryl-5-(substituted alkyl (thio) amido)pyrazoles
ID21775A (id) * 1996-10-25 1999-07-22 Yoshitomi Pharmaceutical Senyawa-senyawa 1-fenilpirazol dan penggunaan farmasinya
EP0977756A1 (en) * 1997-04-25 2000-02-09 Pfizer Limited PYRAZOLOPYRIMIDINONES WHICH INHIBIT TYPE 5 CYCLIC GUANOSINE 3',5'-MONOPHOSPHATE PHOSPHODIESTERASE (cGMP PDE5) FOR THE TREATMENT OF SEXUAL DYSFUNCTION
US5998424A (en) 1997-06-19 1999-12-07 Dupont Pharmaceuticals Company Inhibitors of factor Xa with a neutral P1 specificity group
JP2002507968A (ja) * 1997-06-19 2002-03-12 デュポン ファーマシューティカルズ カンパニー 中性のＰ１特異性基を有するＸａ因子阻害剤
AU4308300A (en) * 1999-05-03 2000-11-17 Dr. Reddy's Research Foundation Pyrazoles having antiinflammatory activity
DE10219435A1 (de) * 2002-05-02 2003-11-13 Bayer Cropscience Ag Substituierte Pyrazolo-pyrimidin-4-one
EP2423188B1 (en) * 2003-08-29 2021-03-10 Mitsui Chemicals Agro, Inc. Intermediates in the preparation of agricultural/horticultural insecticides and method for using the same

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4496390A (en) * 1980-02-26 1985-01-29 May & Baker Limited N-Phenylpyrazole derivatives
CS223840B2 (en) * 1980-02-26 1983-11-25 May & Baker Ltd Herbicide means and method of making the active substances
DE3160972D1 (en) * 1980-12-05 1983-10-27 Basf Ag 2'-phenyl-hydrazino-2-cyanacrylic-acid esters and herbicides containing them
DE3045903A1 (de) * 1980-12-05 1982-07-08 Basf Ag, 6700 Ludwigshafen 5-amino-1-phenylpyrazol-4-carbonsaeureester, verfahren zu ihrer herstellung, diese enthaltende herbizide und ihre anwendung als herbizide
MA19539A1 (fr) * 1981-07-17 1983-04-01 May & Baker Ltd N Acylaminophenylpyrazoles
MA19540A1 (fr) * 1981-07-17 1983-04-01 May & Baker Ltd Derives du n-phenylpyrazole
DE3129429A1 (de) * 1981-07-25 1983-02-10 Basf Ag, 6700 Ludwigshafen 5-amino-1-phenyl-pyrazol-4-carbonsaeurederivate, verfahren zu ihrer herstellung und ihre verwendung zur bekaempfung unerwuenschten pflanzenwuchses
MA19840A1 (fr) * 1982-07-15 1984-04-01 May & Baker Ltd Alcoylamino n-phenyl pyrazole et n-phenyl pyrazole lactames herbicides .
DE3603291A1 (de) * 1986-02-04 1987-08-06 Bayer Ag 5-amino-1-phenyl-pyrazole

Also Published As

Publication number Publication date
US4668280A (en) 1987-05-26
NZ209874A (en) 1986-12-05
EP0138149A2 (de) 1985-04-24
GR80631B (en) 1985-02-12
CA1233473A (en) 1988-03-01
US4770693A (en) 1988-09-13
HUT36347A (en) 1985-09-30
TR23212A (tr) 1989-06-21
DK491384A (da) 1985-04-16
EP0138149A3 (ko) 1985-05-29
ATE40120T1 (de) 1989-02-15
EP0138149B1 (de) 1989-01-18
IL83364A0 (en) 1987-12-31
US4882437A (en) 1989-11-21
DK491384D0 (da) 1984-10-12
IL73221A0 (en) 1985-01-31
BR8405151A (pt) 1985-08-27
ES536768A0 (es) 1985-07-16
IL83364A (en) 1988-11-30
AU569916B2 (en) 1988-02-25
US4791212A (en) 1988-12-13
DD228157A5 (de) 1985-10-09
IL73221A (en) 1988-11-30
ES8506638A1 (es) 1985-07-16
HU196030B (en) 1988-09-28
DE3420985A1 (de) 1985-04-25
KR900007179B1 (ko) 1990-09-29
DE3476199D1 (de) 1989-02-23
AU3410684A (en) 1985-04-18

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