KR840000544A - 항균성 나프탈리딘 또는 퀴놀린 화합물의 염을 제조하는 방법 - Google Patents

항균성 나프탈리딘 또는 퀴놀린 화합물의 염을 제조하는 방법 Download PDF

Info

Publication number
KR840000544A
KR840000544A KR1019820002588A KR820002588A KR840000544A KR 840000544 A KR840000544 A KR 840000544A KR 1019820002588 A KR1019820002588 A KR 1019820002588A KR 820002588 A KR820002588 A KR 820002588A KR 840000544 A KR840000544 A KR 840000544A
Authority
KR
South Korea
Prior art keywords
antimicrobial
naphthalidine
quinoline compounds
preparing salts
acid
Prior art date
Application number
KR1019820002588A
Other languages
English (en)
Other versions
KR880002087B1 (ko
Inventor
프레드릭 미치 토마스
Original Assignee
토마스 디 몰리테르노
워너-람버트 홈파니
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 토마스 디 몰리테르노, 워너-람버트 홈파니 filed Critical 토마스 디 몰리테르노
Publication of KR840000544A publication Critical patent/KR840000544A/ko
Application granted granted Critical
Publication of KR880002087B1 publication Critical patent/KR880002087B1/ko

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Saccharide Compounds (AREA)

Abstract

내용 없음

Description

항균성 나트탈리딘 및 퀴놀린 화합물의 염을 제조하는 방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (1)

  1. 아래의 일반식을 가진 화합물과 Z로 나타낸 산을 반응시키는 것으로 구성된 일반적 C의 화합물을 제조하는 방법.
    식중,
    X는 N 또는 CH
    Z는 갈락튜론산, 아스파라긴산, 글루콘산 또는 글루마민산
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR8202588A 1981-06-11 1982-06-10 항균성 나프티리딘 또는 퀴놀린 화합물의 염 및 그의 제조방법 KR880002087B1 (ko)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US27260181A 1981-06-11 1981-06-11
US272,601 1981-06-11
US272601 1981-06-11
US33418281A 1981-12-24 1981-12-24
US334182 1981-12-24
US334,182 1981-12-24

Publications (2)

Publication Number Publication Date
KR840000544A true KR840000544A (ko) 1984-02-25
KR880002087B1 KR880002087B1 (ko) 1988-10-15

Family

ID=26955624

Family Applications (1)

Application Number Title Priority Date Filing Date
KR8202588A KR880002087B1 (ko) 1981-06-11 1982-06-10 항균성 나프티리딘 또는 퀴놀린 화합물의 염 및 그의 제조방법

Country Status (17)

Country Link
EP (1) EP0067666B1 (ko)
KR (1) KR880002087B1 (ko)
AU (1) AU551596B2 (ko)
CA (1) CA1191842A (ko)
DD (1) DD202561A5 (ko)
DE (1) DE3267135D1 (ko)
DK (1) DK155998C (ko)
ES (1) ES8304117A1 (ko)
FI (1) FI78292C (ko)
GR (1) GR77194B (ko)
HU (1) HU188181B (ko)
IE (1) IE53259B1 (ko)
IL (1) IL66027A (ko)
NO (1) NO157739C (ko)
NZ (1) NZ200908A (ko)
PH (1) PH19091A (ko)
SU (1) SU1192624A3 (ko)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3318145A1 (de) * 1983-05-18 1984-11-22 Bayer Ag, 5090 Leverkusen 7-amino-1-cyclopropyl-6,8-difluor-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
DE3333719A1 (de) * 1983-09-17 1985-04-04 Bayer Ag Loesungen milchsaurer salze von piperazinylchinolon- und piperazinyl-azachinoloncarbonsaeuren
IT1196051B (it) * 1984-03-16 1988-11-10 Schiena Ricerche Composti ad attivita' antibatterica
DE3517709A1 (de) * 1985-01-05 1986-07-10 Bayer Ag Basische zubereitungen von chinoloncarbonsaeuren
US4657913A (en) * 1985-04-18 1987-04-14 Warner-Lambert Company Trifluoro- quinoline -3- carboxylic acids and their use as anti-bacterial agents
HUT40429A (en) * 1985-04-29 1986-12-28 Chinoin Gyogyszer Es Vegyeszet Process for production of salts of derivatives of kynolin carbonic acid
DE3525335A1 (de) * 1985-07-16 1987-01-22 Bayer Ag Embonate von chinoloncarbonsaeuren und ihren derivaten
DE3537761A1 (de) * 1985-10-24 1987-04-30 Bayer Ag Infusionsloesungen der 1-cyclopropyl-6-fluor-1,4-dihydro-4-oxo-7- (1-piperazinyl)-chinolin-3-carbonsaeure
IT1196429B (it) * 1986-07-01 1988-11-16 Mediolanum Farmaceutici Srl Processo per la preparazione di pirido benzotiazine ad attivita' antibatterica e loro sali con acidi solfonici
IL80459A (en) * 1986-10-30 1991-04-15 Abic Ltd Water-soluble adduct of norfloxacin and nicotinic acid
US5188833A (en) * 1987-12-28 1993-02-23 Kyorin Seiyaku Kabushiki Kaisha Freeze-dried pharmaceutical preparations for parenteral use
JPH01175935A (ja) * 1987-12-28 1989-07-12 Kyorin Pharmaceut Co Ltd 凍結乾燥注射剤
US4948894A (en) * 1989-02-21 1990-08-14 American Cyanamid Company 8-fluoro and 7, 8, 10-trifluoro-9-(substituted)-6-oxo-6H-benzo-(C)quinolizine-5-carboxylic acids
KR0159540B1 (ko) * 1992-01-21 1998-12-01 김정순 퀴놀론-카복실산의 염 및 그 함유조성물
ES2127036B1 (es) * 1994-03-21 1999-11-16 Ind Quimica Agropecuaria S A Aducto de norfloxacina soluble en agua.
ES2088742B1 (es) * 1994-06-29 1997-03-16 Salvat Lab Sa Composicion antibiotica de aplicacion otica.
DE19500784A1 (de) * 1995-01-13 1996-07-18 Bayer Ag Enrofloxacin-Injektions- oder Infusionslösungen
MA24500A1 (fr) 1997-03-21 1998-10-01 Lg Life Sciences Ltd Derive du sel d'acide carboxylique de naphthyridine .
DK2134712T3 (da) 2007-04-13 2013-11-18 Dong Wha Pharm Co Ltd Aspartat af 1-cyclopropyl-6-fluoro-7-(8-methoxyimino-2,6-diaza-spiro(3, 4)oct-6-yl)-4-oxo-1,4-dihydro-(1,8) naphthyridin-3-karboxylsyre, fremgangsmåde til fremstilling af samme og antimikrobielt farmaceutisk sammensætning omfattende samme

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR223983A1 (es) * 1978-08-25 1981-10-15 Dainippon Pharmaceutical Co Un procedimiento para-preparar derivados de acido 6-halogeno-4-oxo-7-(1-piperazinil)-1,8-naftiridin-3-carboxilico
ZA811304B (en) * 1980-03-11 1982-06-30 Warner Lambert Co Pharmaceutical salts of 4'-(9-acridinylamino)methanesulfon-m-anisidide

Also Published As

Publication number Publication date
NO157739C (no) 1988-05-11
DK261582A (da) 1982-12-12
KR880002087B1 (ko) 1988-10-15
AU551596B2 (en) 1986-05-08
IL66027A0 (en) 1982-09-30
DE3267135D1 (en) 1985-12-05
PH19091A (en) 1985-12-19
IL66027A (en) 1986-02-28
DK155998B (da) 1989-06-12
EP0067666A1 (en) 1982-12-22
HU188181B (en) 1986-03-28
FI78292B (fi) 1989-03-31
ES512969A0 (es) 1983-02-16
FI822066A0 (fi) 1982-06-10
AU8475782A (en) 1982-12-16
DD202561A5 (de) 1983-09-21
CA1191842A (en) 1985-08-13
IE53259B1 (en) 1988-09-28
NO821931L (no) 1982-12-13
NO157739B (no) 1988-02-01
ES8304117A1 (es) 1983-02-16
DK155998C (da) 1989-11-06
FI78292C (fi) 1989-07-10
SU1192624A3 (ru) 1985-11-15
GR77194B (ko) 1984-09-11
NZ200908A (en) 1984-09-28
IE821390L (en) 1982-12-11
EP0067666B1 (en) 1985-10-30

Similar Documents

Publication Publication Date Title
KR840000544A (ko) 항균성 나프탈리딘 또는 퀴놀린 화합물의 염을 제조하는 방법
KR870008879A (ko) 티아제핀류의 제조 방법
KR850000406A (ko) 4-클로로-2-페닐이미다졸-5-아세트산유도체의 제조방법
KR840003245A (ko) 티아졸리딘 유도체의 제법
KR830007486A (ko) 신규 2-아릴에텔에테르 유도체 및 티오에테르 유도체 제법 및 살충, 살응애제
KR860001110A (ko) 항균제 ⅱ의 제법
KR830000214A (ko) 펩타이드 유도체의 제법
KR850006415A (ko) 항균제의 제조방법
KR830006255A (ko) 피페라진 유도체의 제조방법
KR840003610A (ko) 요소 유도체의 제조방법
KR840005101A (ko) 2-퀴놀린유도체의 제조방법
KR930700435A (ko) 디티오카르밤산의 염류, 그 제조방법 및 그 디티오카르밤산의 염류를 사용하는 이소티오시아네이트류의 제조방법
UA8032A1 (uk) Спосіб одержання 2-(4-метоксіфенілпропіоніл)аміно-6-н-пропіламіно-4,5,6,7-тетрагідробензотіазола у вигляді рацемата або (-)-енантіомера або його кислотно-аддітивної солі
KR830006185A (ko) p-이소부틸-페닐-프로피온산의 아미드유도체의 제조방법
KR880006177A (ko) 구아니디노 메틸벤조산 유도체
KR830009074A (ko) 염기-치환된 안트라닐 산의 제조방법
KR840000504A (ko) N- 페닐피라졸 유도체의 제조방법
KR830003451A (ko) 식물 생장 조절제로 유용한 2-옥소-3-벤조티아졸린 아세트산으로부터 유래된 이미드아미드
KR930700433A (ko) 신규 디술피드 화합물
ATE17851T1 (de) Imidazolylkarbonsaeure, deren derivate und herstellung.
KR830009130A (ko) 인산 아닐리드 유도체의 제조방법
KR840007718A (ko) 3-(메틸술포닐)-2-플로로프로판니트릴 화합물의 제법 및 그 조성물
KR830001203A (ko) N-(1-메틸-2-필로리디닐-메틸)-2,3-디메톡시-5-메틸설파모일 벤즈아미드의 제조방법
KR830009131A (ko) 인산아닐리드 유도체의 제조방법
KR840008335A (ko) 살충제의 제조방법