KR830001295A - 세파로스포린 유도체의 제조법 - Google Patents
세파로스포린 유도체의 제조법 Download PDFInfo
- Publication number
- KR830001295A KR830001295A KR1019790004155A KR790004155A KR830001295A KR 830001295 A KR830001295 A KR 830001295A KR 1019790004155 A KR1019790004155 A KR 1019790004155A KR 790004155 A KR790004155 A KR 790004155A KR 830001295 A KR830001295 A KR 830001295A
- Authority
- KR
- South Korea
- Prior art keywords
- preparation
- sepharosporin
- derivatives
- aminothiazol
- tetrazol
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
- A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/36—Methylene radicals, substituted by sulfur atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cephalosporin Compounds (AREA)
Abstract
내용 없음
Description
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음
제1도는 실시예 1에서 얻은 분말 X선회석도(CuKa. 40KV. 45mA)를, 제2도는 실시예 1에서 얻은 목적물의 적외선 흡수스펙틀(KBr)을 나타냄.
Claims (1)
- 7β-[2-(2-아미노티아졸-4-일)-(Z)-2-메톡시이미노아세타미드]-3-[(1-메틸-1H-테트라졸-5-일)티오메틸]세프]-3-엠-4-카르본산과 HCl 또는 HBr과를 반응시키는 것을 특징으로 하는 7β-[2-(2-아미노티아졸-4-일)-(Z)-2-메톡시이미노아세타미드]-3-[(1-메틸-1H-테트라졸-5-일티오메틸]세프-3-엠-4-카르본산 1분자와 HCl 또는 HBr2분의 1분자와의 결정성염의 제조법.※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR7904155A KR880000181B1 (ko) | 1979-11-27 | 1979-11-27 | 세팔로스포린 유도체의 결정성염의 제조방법 |
| KR1019850002935A KR890000787B1 (ko) | 1979-11-27 | 1985-04-30 | 세팔로스포린 유도체 성분의 주사용 또는 외용제의 제조방법 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR7904155A KR880000181B1 (ko) | 1979-11-27 | 1979-11-27 | 세팔로스포린 유도체의 결정성염의 제조방법 |
Related Child Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1019850002935A Division KR890000787B1 (ko) | 1979-11-27 | 1985-04-30 | 세팔로스포린 유도체 성분의 주사용 또는 외용제의 제조방법 |
| KR1019850002934A Division KR850007927A (ko) | 1985-04-30 | 1985-04-30 | 세팔로스포린 유도체 결정성염의 제조방법 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| KR830001295A true KR830001295A (ko) | 1983-04-30 |
| KR880000181B1 KR880000181B1 (ko) | 1988-03-12 |
Family
ID=19213669
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR7904155A KR880000181B1 (ko) | 1979-11-27 | 1979-11-27 | 세팔로스포린 유도체의 결정성염의 제조방법 |
| KR1019850002935A KR890000787B1 (ko) | 1979-11-27 | 1985-04-30 | 세팔로스포린 유도체 성분의 주사용 또는 외용제의 제조방법 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1019850002935A KR890000787B1 (ko) | 1979-11-27 | 1985-04-30 | 세팔로스포린 유도체 성분의 주사용 또는 외용제의 제조방법 |
Country Status (1)
| Country | Link |
|---|---|
| KR (2) | KR880000181B1 (ko) |
-
1979
- 1979-11-27 KR KR7904155A patent/KR880000181B1/ko active
-
1985
- 1985-04-30 KR KR1019850002935A patent/KR890000787B1/ko not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| KR850007928A (ko) | 1985-12-11 |
| KR890000787B1 (ko) | 1989-04-07 |
| KR880000181B1 (ko) | 1988-03-12 |
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