KR20220078604A - 헤테로시클리덴아세트아미드 유도체 함유 의약 - Google Patents

헤테로시클리덴아세트아미드 유도체 함유 의약 Download PDF

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Publication number
KR20220078604A
KR20220078604A KR1020227012080A KR20227012080A KR20220078604A KR 20220078604 A KR20220078604 A KR 20220078604A KR 1020227012080 A KR1020227012080 A KR 1020227012080A KR 20227012080 A KR20227012080 A KR 20227012080A KR 20220078604 A KR20220078604 A KR 20220078604A
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KR
South Korea
Prior art keywords
eye
dry eye
item
composition
ylidene
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Pending
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KR1020227012080A
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English (en)
Korean (ko)
Inventor
다케시 다루이
신야 고바야시
Original Assignee
센주 세이야꾸 가부시키가이샤
모찌다 세이야쿠 가부시끼가이샤
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Application filed by 센주 세이야꾸 가부시키가이샤, 모찌다 세이야쿠 가부시끼가이샤 filed Critical 센주 세이야꾸 가부시키가이샤
Publication of KR20220078604A publication Critical patent/KR20220078604A/ko
Pending legal-status Critical Current

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0048—Eye, e.g. artificial tears
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/04—Artificial tears; Irrigation solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Ophthalmology & Optometry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Molecular Biology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Inorganic Chemistry (AREA)
  • Biochemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
KR1020227012080A 2019-10-04 2020-10-02 헤테로시클리덴아세트아미드 유도체 함유 의약 Pending KR20220078604A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2019184053 2019-10-04
JPJP-P-2019-184053 2019-10-04
PCT/JP2020/037548 WO2021066144A1 (ja) 2019-10-04 2020-10-02 ヘテロシクリデンアセトアミド誘導体含有医薬

Publications (1)

Publication Number Publication Date
KR20220078604A true KR20220078604A (ko) 2022-06-10

Family

ID=75338162

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020227012080A Pending KR20220078604A (ko) 2019-10-04 2020-10-02 헤테로시클리덴아세트아미드 유도체 함유 의약

Country Status (17)

Country Link
US (2) US12533337B2 (https=)
EP (2) EP4545095A3 (https=)
JP (4) JP7025094B2 (https=)
KR (1) KR20220078604A (https=)
CN (1) CN114585357A (https=)
AU (1) AU2026202464A1 (https=)
BR (1) BR112022005992A2 (https=)
CA (1) CA3156484A1 (https=)
DK (1) DK4043014T3 (https=)
ES (1) ES3031607T3 (https=)
HU (1) HUE072085T2 (https=)
MX (2) MX2022004027A (https=)
MY (1) MY207759A (https=)
PH (1) PH12022550805A1 (https=)
PL (1) PL4043014T3 (https=)
PT (1) PT4043014T (https=)
WO (1) WO2021066144A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3156484A1 (en) 2019-10-04 2021-04-08 Senju Pharmaceutical Co., Ltd. PHARMACEUTICAL MEDICINAL PRODUCT CONTAINING A HETEROCYCLIDENE ACETAMIDE DERIVATIVE
CN117120048A (zh) 2021-03-30 2023-11-24 千寿制药株式会社 含杂环亚基乙酰胺衍生物的悬浮液
KR20250065723A (ko) 2022-09-29 2025-05-13 센주 세이야꾸 가부시키가이샤 멸균 처리한 헤테로시클리덴아세트아미드 유도체 함유 현탁액
JP7589394B2 (ja) * 2022-09-29 2024-11-25 千寿製薬株式会社 ヘテロシクリデンアセトアミド誘導体を含む配合剤

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5621566A (en) 1979-08-01 1981-02-28 Alpha- Shokuhin Kk Preparation of bifun from homegrown rice and apparatus used for it
CN101228131B (zh) * 2005-07-22 2013-01-09 持田制药株式会社 新的杂环亚基乙酰胺衍生物
JP4754566B2 (ja) 2005-07-22 2011-08-24 持田製薬株式会社 新規なヘテロシクリデンアセトアミド誘導体
RU2451014C2 (ru) 2005-07-22 2012-05-20 Мотида Фармасьютикал Ко., Лтд. Новое производное гетероциклиден ацетамида
TW200927192A (en) 2007-11-19 2009-07-01 Alcon Res Ltd Use of TRPV1 receptor antagonists for treating dry eye and ocular pain
US20100210682A1 (en) * 2009-02-19 2010-08-19 Abbott Laboratories Repeated Dosing of TRPV1 Antagonists
EP2377850A1 (en) 2010-03-30 2011-10-19 Pharmeste S.r.l. TRPV1 vanilloid receptor antagonists with a bicyclic portion
WO2012045729A1 (en) * 2010-10-05 2012-04-12 Glaxo Group Limited Imidazo [1, 2 -a] pyridine and pyrazolo [1, 5 -a] pyridine derivatives as trpv1 antagonists
GB201215857D0 (en) * 2012-09-05 2012-10-24 Sylentis Sau siRNA and their use in methods and compositions for the treatment and/or prevention of eye conditions
JP6230743B1 (ja) * 2017-05-31 2017-11-15 持田製薬株式会社 ヘテロシクリデンアセトアミド誘導体の結晶
JP7373909B2 (ja) 2018-04-06 2023-11-06 株式会社シマノ 変速制御装置および変速システム
CA3156484A1 (en) 2019-10-04 2021-04-08 Senju Pharmaceutical Co., Ltd. PHARMACEUTICAL MEDICINAL PRODUCT CONTAINING A HETEROCYCLIDENE ACETAMIDE DERIVATIVE

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
파마시아 Vol.50 No.3 2014:201 내지 206

Also Published As

Publication number Publication date
JP2022065024A (ja) 2022-04-26
EP4043014A4 (en) 2023-10-11
MY207759A (en) 2025-03-17
WO2021066144A1 (ja) 2021-04-08
CA3156484A1 (en) 2021-04-08
EP4545095A2 (en) 2025-04-30
US12502375B2 (en) 2025-12-23
PH12022550805A1 (en) 2023-10-02
JPWO2021066144A1 (ja) 2021-12-02
DK4043014T3 (da) 2025-06-23
HUE072085T2 (hu) 2025-10-28
JP7248836B2 (ja) 2023-03-29
MX2025005474A (es) 2025-06-02
US20220370404A1 (en) 2022-11-24
EP4043014B1 (en) 2025-03-19
US20250134854A1 (en) 2025-05-01
AU2020361093A1 (en) 2022-05-19
MX2022004027A (es) 2022-07-19
JP2023011735A (ja) 2023-01-24
JP7801201B2 (ja) 2026-01-16
PT4043014T (pt) 2025-06-09
AU2026202464A1 (en) 2026-04-16
PL4043014T3 (pl) 2025-08-11
CN114585357A (zh) 2022-06-03
US12533337B2 (en) 2026-01-27
ES3031607T3 (en) 2025-07-09
EP4545095A3 (en) 2025-07-02
BR112022005992A2 (pt) 2022-06-21
JP2026042857A (ja) 2026-03-11
EP4043014A1 (en) 2022-08-17
JP7025094B2 (ja) 2022-02-24

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