KR20140138824A - 부인과 질환을 치료하기 위한 방법 - Google Patents
부인과 질환을 치료하기 위한 방법 Download PDFInfo
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- KR20140138824A KR20140138824A KR1020147027575A KR20147027575A KR20140138824A KR 20140138824 A KR20140138824 A KR 20140138824A KR 1020147027575 A KR1020147027575 A KR 1020147027575A KR 20147027575 A KR20147027575 A KR 20147027575A KR 20140138824 A KR20140138824 A KR 20140138824A
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- South Korea
- Prior art keywords
- pharmaceutical composition
- vaginal
- progesterone receptor
- administration
- receptor modulator
- Prior art date
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- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
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Landscapes
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261614785P | 2012-03-23 | 2012-03-23 | |
| US61/614,785 | 2012-03-23 | ||
| EP12160956.4 | 2012-03-23 | ||
| EP12160956.4A EP2641602A1 (en) | 2012-03-23 | 2012-03-23 | Method for treating gynecological diseases |
| PCT/IB2013/052274 WO2013140372A1 (en) | 2012-03-23 | 2013-03-22 | Method for treating gynecological diseases |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20140138824A true KR20140138824A (ko) | 2014-12-04 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020147027575A Ceased KR20140138824A (ko) | 2012-03-23 | 2013-03-22 | 부인과 질환을 치료하기 위한 방법 |
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| Country | Link |
|---|---|
| US (1) | US10441534B2 (enExample) |
| EP (3) | EP2641602A1 (enExample) |
| JP (2) | JP2015514700A (enExample) |
| KR (1) | KR20140138824A (enExample) |
| CN (1) | CN104203246A (enExample) |
| AU (1) | AU2013236960B2 (enExample) |
| CA (1) | CA2864073A1 (enExample) |
| CO (1) | CO7111317A2 (enExample) |
| EA (1) | EA031488B1 (enExample) |
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|---|---|---|---|---|
| WO2017112909A1 (en) | 2015-12-23 | 2017-06-29 | Oric Pharmaceuticals, Inc. | Inhibitors of glucocorticoid receptor |
| WO2017112904A1 (en) | 2015-12-23 | 2017-06-29 | Oric Pharmaceuticals, Inc. | Inhibitors of glucocorticoid receptor |
| JP6906525B2 (ja) | 2015-12-23 | 2021-07-21 | オリック ファーマシューティカルズ,インク. | グルココルチコイド受容体の阻害剤 |
| WO2017165707A1 (en) * | 2016-03-24 | 2017-09-28 | Juniper Pharmaceuticals, Inc. | Vaginal administration of agents for treating and preventing pain associated with gynecological medical procedures |
| CN110099915A (zh) | 2016-10-07 | 2019-08-06 | 欧瑞克制药公司 | 糖皮质激素受体抑制剂 |
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| US3545439A (en) | 1968-01-04 | 1970-12-08 | Upjohn Co | Medicated devices and methods |
| US3920805A (en) | 1971-12-09 | 1975-11-18 | Upjohn Co | Pharmaceutical devices and method |
| IL48277A (en) | 1974-10-18 | 1978-03-10 | Schering Ag | Vaginal ring |
| US4155991A (en) | 1974-10-18 | 1979-05-22 | Schering Aktiengesellschaft | Vaginal ring |
| US3991760A (en) | 1975-12-02 | 1976-11-16 | The Procter & Gamble Company | Vaginal medicament dispensing means |
| US3995634A (en) | 1975-12-02 | 1976-12-07 | The Procter & Gamble Company | Vaginal cavity dispensing means and method |
| US3995633A (en) | 1975-12-02 | 1976-12-07 | The Procter & Gamble Company | Vaginal Medicament dispensing device |
| US4286587A (en) | 1978-10-11 | 1981-09-01 | Alza Corporation | Vaginal drug delivery system made from polymer |
| US4292965A (en) | 1978-12-29 | 1981-10-06 | The Population Council, Inc. | Intravaginal ring |
| US4250611A (en) | 1979-04-19 | 1981-02-17 | Alza Corporation | Process for making drug delivery device with reservoir |
| US4596576A (en) | 1984-10-12 | 1986-06-24 | Akzo N.V. | Release system for two or more active substances |
| NL8500470A (nl) | 1985-02-19 | 1986-09-16 | Achel Homesteel Pvba | Intravaginaal orgaan. |
| US4954490A (en) | 1988-06-23 | 1990-09-04 | Research Triangle Institute | 11 β-substituted progesterone analogs |
| FI95768C (fi) | 1993-06-17 | 1996-03-25 | Leiras Oy | Emättimensisäinen antosysteemi |
| US5929262A (en) | 1995-03-30 | 1999-07-27 | The United States Of America As Represented By The Department Of Health And Human Services | Method for preparing 17α-acetoxy-11β-(4-N, N-dimethylaminophyl)-19-Norpregna-4,9-diene-3, 20-dione, intermediates useful in the method, and methods for the preparation of such intermediates |
| US5972372A (en) | 1996-07-31 | 1999-10-26 | The Population Council, Inc. | Intravaginal rings with insertable drug-containing core |
| ES2212912B1 (es) | 2003-01-22 | 2005-10-01 | Crystal Pharma, S.A. | Procedimiento para la obtencion de 17alfa-acetoxi-11beta-(4-n,n-dimetilaminofenil)-19-norpregna-4,9-dien-3,20-diona. |
| US20060111577A1 (en) | 2003-02-28 | 2006-05-25 | Kim Hyun K | Method for preparing 17 alpha-acetoxy-11beta-(4-n,n-dimethylaminophenyl)-19-norpregna-4,9-diene-3,20-dione, intermediates thereof, and methods for the preparation of such intermediates |
| KR101229701B1 (ko) | 2004-07-09 | 2013-02-05 | 라보라토이레 에이치알에이 파르마 | 프로게스테론 수용체 조절제를 함유하는 서방형 조성물 |
| US8569274B2 (en) * | 2007-04-20 | 2013-10-29 | Preglem S.A. | Progesterone antagonist and selective progesterone modulator in the treatment of excessive uterine bleeding |
| US8299050B2 (en) * | 2008-01-29 | 2012-10-30 | Laboratoire Hra-Pharma | Method for treating uterine fibroids |
| LT2249757T (lt) * | 2008-02-04 | 2017-09-25 | Ferring B.V. | Vientisi intravaginaliniai žiedai, apimantys progesteroną, ir jų gamybos bei panaudojimo būdai |
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2012
- 2012-03-23 EP EP12160956.4A patent/EP2641602A1/en not_active Withdrawn
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2013
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- 2013-03-22 AU AU2013236960A patent/AU2013236960B2/en not_active Ceased
- 2013-03-22 HK HK15100309.9A patent/HK1199827A1/xx unknown
- 2013-03-22 US US14/386,726 patent/US10441534B2/en not_active Expired - Fee Related
- 2013-03-22 CA CA2864073A patent/CA2864073A1/en not_active Abandoned
- 2013-03-22 GE GEAP201313608A patent/GEP201706696B/en unknown
- 2013-03-22 EA EA201491614A patent/EA031488B1/ru not_active IP Right Cessation
- 2013-03-22 TW TW107104368A patent/TW201832767A/zh unknown
- 2013-03-22 EP EP13721095.1A patent/EP2827873A1/en not_active Ceased
- 2013-03-22 WO PCT/IB2013/052274 patent/WO2013140372A1/en not_active Ceased
- 2013-03-22 CN CN201380014168.1A patent/CN104203246A/zh active Pending
- 2013-03-22 SG SG11201404921QA patent/SG11201404921QA/en unknown
- 2013-03-22 MY MYPI2014002228A patent/MY172530A/en unknown
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2014
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2018
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Also Published As
| Publication number | Publication date |
|---|---|
| CA2864073A1 (en) | 2013-09-26 |
| CN104203246A (zh) | 2014-12-10 |
| AU2013236960B2 (en) | 2017-11-23 |
| TW201832767A (zh) | 2018-09-16 |
| GEP201706696B (en) | 2017-07-10 |
| JP2015514700A (ja) | 2015-05-21 |
| HK1199827A1 (en) | 2015-07-24 |
| MX2014011487A (es) | 2015-01-12 |
| MX369520B (es) | 2019-11-11 |
| TW201400121A (zh) | 2014-01-01 |
| US10441534B2 (en) | 2019-10-15 |
| JP2018109025A (ja) | 2018-07-12 |
| EP2641602A1 (en) | 2013-09-25 |
| CO7111317A2 (es) | 2014-11-10 |
| ZA201407575B (en) | 2015-12-23 |
| NZ630011A (en) | 2016-12-23 |
| US20150038476A1 (en) | 2015-02-05 |
| WO2013140372A1 (en) | 2013-09-26 |
| MY172530A (en) | 2019-11-29 |
| EP2827873A1 (en) | 2015-01-28 |
| EA031488B1 (ru) | 2019-01-31 |
| AU2013236960A1 (en) | 2014-09-25 |
| SG11201404921QA (en) | 2014-10-30 |
| EA201491614A1 (ru) | 2015-01-30 |
| EP3363500A1 (en) | 2018-08-22 |
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