KR20130023381A - Ppar 활성 화합물 - Google Patents

Ppar 활성 화합물 Download PDF

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Publication number
KR20130023381A
KR20130023381A KR1020137002335A KR20137002335A KR20130023381A KR 20130023381 A KR20130023381 A KR 20130023381A KR 1020137002335 A KR1020137002335 A KR 1020137002335A KR 20137002335 A KR20137002335 A KR 20137002335A KR 20130023381 A KR20130023381 A KR 20130023381A
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South Korea
Prior art keywords
optionally substituted
propionic acid
indol
methoxy
binding
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KR1020137002335A
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English (en)
Korean (ko)
Inventor
제임스 아놀드
딘 알. 아티스
클라렌스 알. 허트
프라브하 엔. 이브라힘
하이케 크루프카
잭 린
마이클 브이. 밀번
웨이루 왕
차오 장
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플렉시콘, 인코퍼레이티드
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Publication of KR20130023381A publication Critical patent/KR20130023381A/ko

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    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
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    • C07D209/04Indoles; Hydrogenated indoles
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    • C07D209/32Oxygen atoms
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    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
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    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
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    • C04B35/626Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B
    • C04B35/63Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B using additives specially adapted for forming the products, e.g.. binder binders
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KR1020137002335A 2003-07-17 2004-07-16 Ppar 활성 화합물 KR20130023381A (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US48852303P 2003-07-17 2003-07-17
US60/488,523 2003-07-17
US55299404P 2004-03-12 2004-03-12
US60/552,994 2004-03-12
PCT/US2004/023234 WO2005009958A1 (en) 2003-07-17 2004-07-16 Ppar active compounds

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KR1020067001015A Division KR101415503B1 (ko) 2003-07-17 2004-07-16 Ppar 활성 화합물

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KR1020137002335A KR20130023381A (ko) 2003-07-17 2004-07-16 Ppar 활성 화합물
KR1020067001015A KR101415503B1 (ko) 2003-07-17 2004-07-16 Ppar 활성 화합물

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AU (1) AU2004259738B2 (US07476746-20090113-C00115.png)
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US7348338B2 (en) 2003-07-17 2008-03-25 Plexxikon, Inc. PPAR active compounds
JP4845730B2 (ja) 2003-07-17 2011-12-28 プレキシコン,インコーポレーテッド Ppar活性化合物
US7574340B2 (en) * 2003-09-08 2009-08-11 The United States Of America As Represented By The Secretary Of The Army Small molecules and a pharmacophore model for inhibition of botulinum toxin and methods of making and using thereof
PE20060303A1 (es) 2004-06-23 2006-05-19 Wyeth Corp Metabolitos de indolilalquilamina como ligandos de 5-hidroxitriptamina-6
US7531568B2 (en) * 2004-11-30 2009-05-12 Plexxikon, Inc. PPAR active compounds
AU2005311826A1 (en) * 2004-11-30 2006-06-08 Plexxikon, Inc. Indole derivatives for use as PPAR active compounds
EP1911759A4 (en) * 2005-07-22 2010-07-21 Shionogi & Co AZAINDOL DERIVATIVE ANTAGONISTIC EFFECT ON PGD2 RECEPTOR
FR2890071B1 (fr) * 2005-08-30 2007-11-09 Fournier Sa Sa Lab Nouveaux composes de l'indole
FR2890072A1 (fr) 2005-09-01 2007-03-02 Fournier S A Sa Lab Nouveaux composesde pyrrolopyridine
TW200800872A (en) * 2005-09-07 2008-01-01 Plexxikon Inc PPAR active compounds
US20080234349A1 (en) * 2005-09-07 2008-09-25 Jack Lin PPAR active compounds
US20070072904A1 (en) * 2005-09-07 2007-03-29 Jack Lin PPAR active compounds
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