KR20120017421A - 인지 장애의 치료를 위한 ５-ｈｔ₄ 수용체 아고니스트 화합물 - Google Patents
인지 장애의 치료를 위한 ５-ｈｔ₄ 수용체 아고니스트 화합물 Download PDFInfo
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- KR20120017421A KR20120017421A KR1020117026729A KR20117026729A KR20120017421A KR 20120017421 A KR20120017421 A KR 20120017421A KR 1020117026729 A KR1020117026729 A KR 1020117026729A KR 20117026729 A KR20117026729 A KR 20117026729A KR 20120017421 A KR20120017421 A KR 20120017421A
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- compound
- amino
- methyl
- carboxylic acid
- isopropyl
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Landscapes
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| DE10164139A1 (de) | 2001-12-27 | 2003-07-10 | Bayer Ag | 2-Heteroarylcarbonsäureamide |
| LT2889033T (lt) | 2008-11-19 | 2018-07-10 | Forum Pharmaceuticals Inc. | Šizofrenijos negatyvių simptomų gydymas (r)-7-chlor-n-(chinuklidin-3-il)benzo[b]tiofen-2-karboksamidu ir jo farmaciniu požiūriu priimtinomis druskomis |
| JP5808319B2 (ja) * | 2009-05-11 | 2015-11-10 | フォルム ファーマシューティカルズ、インコーポレイテッド | アセチルコリンエステラーゼ阻害剤と組み合わせた特定のα７ニコチン酸受容体を用いた認知障害の治療 |
| PE20170923A1 (es) | 2010-05-17 | 2017-07-12 | Forum Pharmaceuticals Inc | Una forma cristalina de clorhidrato de (r)-7-cloro-n-(quinuclidin-3-il)benzo[b]tiofeno-2-carboxamida monohidratado |
| EP3461481A1 (en) | 2012-05-08 | 2019-04-03 | Forum Pharmaceuticals Inc. | Methods of maintaining, treating or improving cognitive function |
| US10874701B2 (en) | 2012-08-16 | 2020-12-29 | University-Industry Cooperation Group Of Kyung Hee University | Lactic acid bacteria capable of preventing and/or treating senescence and dementia |
| JP6009080B2 (ja) | 2012-08-16 | 2016-10-19 | ユニバーシティ−インダストリー コオペレーション グループ オブ キョン ヒ ユニバーシティＵｎｉｖｅｒｓｉｔｙ−Ｉｎｄｕｓｔｒｙ Ｃｏｏｐｅｒａｔｉｏｎ Ｇｒｏｕｐ Ｏｆ Ｋｙｕｎｇ Ｈｅｅ Ｕｎｉｖｅｒｓｉｔｙ | 老化及び認知症の予防及び／または治療活性を有する乳酸菌 |
| BR112019001145A2 (pt) | 2017-05-24 | 2019-04-30 | H. Lundbeck A/S | combinação de um antagonista do receptor 5-ht6 e de um inibidor de acetilcolinesterase para uso no tratamento da doença de alzheimer em uma subpopulação de pacientes portadores de alelos de apoe4 |
| KR20200010211A (ko) | 2017-06-01 | 2020-01-30 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | Pde9 저해제를 포함하는 약제학적 조성물 |
| KR20190137936A (ko) | 2017-06-02 | 2019-12-11 | 후지필름 도야마 케미컬 가부시키가이샤 | 뇌 위축 예방 또는 치료제 |
| BR112020000482A2 (pt) | 2017-07-31 | 2020-07-21 | Theravance Biopharma R&D Ip, Llc | métodos de tratamento de sintomas de gastroparesia usando velusetrag |
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| EP2133078A1 (en) * | 2000-03-03 | 2009-12-16 | Eisai R&D Management Co., Ltd. | Use of a cholinesterase inhibitor for the treatment of dementia and cognitive impairments |
| TWI351282B (en) * | 2004-04-07 | 2011-11-01 | Theravance Inc | Quinolinone-carboxamide compounds as 5-ht4 recepto |
| US7598265B2 (en) * | 2004-09-30 | 2009-10-06 | Epix Delaware, Inc. | Compositions and methods for treating CNS disorders |
| TWI377206B (en) * | 2005-04-06 | 2012-11-21 | Theravance Inc | Crystalline form of a quinolinone-carboxamide compound |
| MY147756A (en) * | 2005-05-25 | 2013-01-15 | Theravance Inc | Benzimidazole-carboxamide compounds as 5-ht4 receptor agonists |
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- 2010-04-12 SM SM20180036T patent/SMT201800036T1/it unknown
- 2010-04-12 PT PT107137903T patent/PT2419104T/pt unknown
- 2010-04-12 CN CN201610257689.5A patent/CN105832735A/zh active Pending
- 2010-04-12 EP EP10713790.3A patent/EP2419104B1/en active Active
- 2010-04-12 KR KR1020117026729A patent/KR20120017421A/ko not_active Ceased
- 2010-04-12 SI SI201031632T patent/SI2419104T1/en unknown
- 2010-04-12 AU AU2010236734A patent/AU2010236734B2/en not_active Ceased
- 2010-04-12 HU HUE10713790A patent/HUE038141T2/hu unknown
- 2010-04-12 LT LTEP10713790.3T patent/LT2419104T/lt unknown
- 2010-04-12 ES ES10713790.3T patent/ES2654930T3/es active Active
- 2010-04-12 HR HRP20180018TT patent/HRP20180018T1/hr unknown
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- 2010-04-12 JP JP2012504924A patent/JP2012523437A/ja active Pending
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2011
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2013
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Also Published As
| Publication number | Publication date |
|---|---|
| PT2419104T (pt) | 2018-01-31 |
| RU2011146032A (ru) | 2013-05-20 |
| EP2419104B1 (en) | 2017-11-08 |
| IL215660A0 (en) | 2012-01-31 |
| WO2010120695A3 (en) | 2010-12-02 |
| JP2012523437A (ja) | 2012-10-04 |
| US20140057939A1 (en) | 2014-02-27 |
| DK2419104T3 (en) | 2018-02-05 |
| BRPI1013777A8 (pt) | 2017-09-19 |
| US20100261752A1 (en) | 2010-10-14 |
| CA2758321A1 (en) | 2010-10-21 |
| SI2419104T1 (en) | 2018-03-30 |
| AU2010236734A8 (en) | 2012-02-16 |
| NO2419104T3 (https=) | 2018-04-07 |
| CN105832735A (zh) | 2016-08-10 |
| US8404711B2 (en) | 2013-03-26 |
| CN102395371A (zh) | 2012-03-28 |
| MX2011010782A (es) | 2012-01-20 |
| ES2654930T3 (es) | 2018-02-15 |
| LT2419104T (lt) | 2018-02-12 |
| WO2010120695A2 (en) | 2010-10-21 |
| ZA201107490B (en) | 2012-06-27 |
| HRP20180018T1 (hr) | 2018-02-09 |
| RU2569056C2 (ru) | 2015-11-20 |
| SMT201800036T1 (it) | 2018-03-08 |
| BRPI1013777A2 (pt) | 2016-04-05 |
| AU2010236734B2 (en) | 2015-06-11 |
| AU2010236734A1 (en) | 2011-11-03 |
| PL2419104T3 (pl) | 2018-04-30 |
| EP2419104A2 (en) | 2012-02-22 |
| HUE038141T2 (hu) | 2018-10-29 |
| CY1119800T1 (el) | 2018-06-27 |
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