KR20090092288A - 뉴로키닌 길항제를 포함하는 제약 제형 - Google Patents
뉴로키닌 길항제를 포함하는 제약 제형Info
- Publication number
- KR20090092288A KR20090092288A KR1020097012819A KR20097012819A KR20090092288A KR 20090092288 A KR20090092288 A KR 20090092288A KR 1020097012819 A KR1020097012819 A KR 1020097012819A KR 20097012819 A KR20097012819 A KR 20097012819A KR 20090092288 A KR20090092288 A KR 20090092288A
- Authority
- KR
- South Korea
- Prior art keywords
- solid dispersion
- carrier
- pharmaceutical composition
- methyl
- suspension
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
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- 235000019812 sodium carboxymethyl cellulose Nutrition 0.000 description 1
- 229920001027 sodium carboxymethylcellulose Polymers 0.000 description 1
- NRHMKIHPTBHXPF-TUJRSCDTSA-M sodium cholate Chemical compound [Na+].C([C@H]1C[C@H]2O)[C@H](O)CC[C@]1(C)[C@@H]1[C@@H]2[C@@H]2CC[C@H]([C@@H](CCC([O-])=O)C)[C@@]2(C)[C@@H](O)C1 NRHMKIHPTBHXPF-TUJRSCDTSA-M 0.000 description 1
- DVQHRBFGRZHMSR-UHFFFAOYSA-N sodium methyl 2,2-dimethyl-4,6-dioxo-5-(N-prop-2-enoxy-C-propylcarbonimidoyl)cyclohexane-1-carboxylate Chemical compound [Na+].C=CCON=C(CCC)[C-]1C(=O)CC(C)(C)C(C(=O)OC)C1=O DVQHRBFGRZHMSR-UHFFFAOYSA-N 0.000 description 1
- 229940045902 sodium stearyl fumarate Drugs 0.000 description 1
- 239000008279 sol Substances 0.000 description 1
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- 229960002920 sorbitol Drugs 0.000 description 1
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- 239000003381 stabilizer Substances 0.000 description 1
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- 125000004079 stearyl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])[H] 0.000 description 1
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- ODLHGICHYURWBS-LKONHMLTSA-N trappsol cyclo Chemical compound CC(O)COC[C@H]([C@H]([C@@H]([C@H]1O)O)O[C@H]2O[C@@H]([C@@H](O[C@H]3O[C@H](COCC(C)O)[C@H]([C@@H]([C@H]3O)O)O[C@H]3O[C@H](COCC(C)O)[C@H]([C@@H]([C@H]3O)O)O[C@H]3O[C@H](COCC(C)O)[C@H]([C@@H]([C@H]3O)O)O[C@H]3O[C@H](COCC(C)O)[C@H]([C@@H]([C@H]3O)O)O3)[C@H](O)[C@H]2O)COCC(O)C)O[C@@H]1O[C@H]1[C@H](O)[C@@H](O)[C@@H]3O[C@@H]1COCC(C)O ODLHGICHYURWBS-LKONHMLTSA-N 0.000 description 1
- QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical compound [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
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Classifications
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Inorganic Chemistry (AREA)
- Pulmonology (AREA)
- Dispersion Chemistry (AREA)
- Urology & Nephrology (AREA)
- Nutrition Science (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP06126964A EP1938804A1 (en) | 2006-12-22 | 2006-12-22 | Pharmaceutical formulation comprising neurokinin antagonist |
| EP06126964.3 | 2006-12-22 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20090092288A true KR20090092288A (ko) | 2009-08-31 |
Family
ID=37762542
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020097012819A Withdrawn KR20090092288A (ko) | 2006-12-22 | 2007-12-20 | 뉴로키닌 길항제를 포함하는 제약 제형 |
Country Status (25)
| Country | Link |
|---|---|
| US (1) | US20100015225A1 (https=) |
| EP (2) | EP1938804A1 (https=) |
| JP (1) | JP2010513356A (https=) |
| KR (1) | KR20090092288A (https=) |
| CN (1) | CN101541309A (https=) |
| AR (1) | AR064622A1 (https=) |
| AU (1) | AU2007338359B2 (https=) |
| BR (1) | BRPI0720937A2 (https=) |
| CA (1) | CA2672402A1 (https=) |
| CL (1) | CL2007003767A1 (https=) |
| CO (1) | CO6180497A2 (https=) |
| EA (1) | EA200900827A1 (https=) |
| EC (1) | ECSP099450A (https=) |
| GT (1) | GT200900173A (https=) |
| IL (1) | IL198780A0 (https=) |
| MA (1) | MA31004B1 (https=) |
| MX (1) | MX2009006747A (https=) |
| MY (1) | MY145919A (https=) |
| NO (1) | NO20092722L (https=) |
| NZ (1) | NZ576987A (https=) |
| PE (1) | PE20081848A1 (https=) |
| TN (1) | TN2009000253A1 (https=) |
| TW (1) | TW200848056A (https=) |
| WO (1) | WO2008077591A2 (https=) |
| ZA (1) | ZA200903271B (https=) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW201309635A (zh) * | 2006-02-10 | 2013-03-01 | Dow Agrosciences Llc | 殺蟲性之ｎ-取代（６-鹵烷基吡啶-３-基）烷基磺醯亞胺（二） |
| JPWO2010092925A1 (ja) * | 2009-02-12 | 2012-08-16 | あすか製薬株式会社 | 固体分散体とその医薬組成物、並びにそれらの製造方法 |
| US20120077803A1 (en) * | 2009-02-24 | 2012-03-29 | Novartis Ag | Uses Of NK Receptor Antagonists |
| US8263119B2 (en) * | 2010-12-01 | 2012-09-11 | Shire Llc | Capsule formulations containing lanthanum compounds |
| US9487495B2 (en) | 2012-01-06 | 2016-11-08 | The Scripts Research Institute | Carbamate compounds and of making and using same |
| MX2017011469A (es) * | 2015-03-10 | 2018-01-23 | Shionogi Inc | Dispersiones sólidas. |
| SG10202012002TA (en) | 2015-05-11 | 2021-01-28 | Lundbeck La Jolla Research Center Inc | Methods of treating inflammation or neuropathic pain |
| ES3063790T3 (en) | 2015-06-09 | 2026-04-20 | Lonza Sales Ag | Formulations to achieve rapid dissolution of drug from spray-dried dispersions in capsules |
| KR20190085046A (ko) * | 2016-11-16 | 2019-07-17 | 어바이드 테라퓨틱스, 인크. | 약학 제제 |
| DK3541807T3 (da) | 2016-11-16 | 2021-12-06 | H Lundbeck As | Krystallinsk form af en magl-inhibitor |
| IL297470A (en) | 2020-04-21 | 2022-12-01 | H Lundbeck As | Synthesis of a monoacylglycerol lipase inhibitor |
| CN111904960A (zh) * | 2020-05-19 | 2020-11-10 | 合肥合源药业有限公司 | 一种固体分散体及药用组合物 |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3622677A (en) * | 1969-07-07 | 1971-11-23 | Staley Mfg Co A E | Compressed tablets containing compacted starch as binder-disintegrant ingredient |
| JPH054919A (ja) * | 1990-07-25 | 1993-01-14 | Sankyo Co Ltd | チアゾリジン誘導体の固体分散体 |
| MY132550A (en) * | 1996-08-22 | 2007-10-31 | Novartis Ag | Acylaminoalkenylene-amide derivatives as nk1 and nk2 antogonists |
| KR20010023729A (ko) * | 1997-11-03 | 2001-03-26 | 디르크 반테 | 지질 저하제 조성물 |
| ME00189B (me) * | 1998-03-26 | 2011-02-10 | Astellas Pharma Inc | Preparati sa neprekidnim oslobađanjem |
| US20010053791A1 (en) * | 2000-03-16 | 2001-12-20 | Babcock Walter C. | Glycogen phosphorylase inhibitor |
| JP2004131393A (ja) * | 2002-10-08 | 2004-04-30 | Kowa Co | 易溶出性製剤 |
| GB2394417A (en) * | 2002-10-24 | 2004-04-28 | Novartis Ag | Solid dispersion comprising a piperidine substance P antagonist and a carrier |
| EP1686985A2 (en) * | 2003-10-27 | 2006-08-09 | Novartis AG | Use of neurokinin antagonists in the treatment of urinary incontinence |
| GB0402679D0 (en) * | 2004-02-06 | 2004-03-10 | Novartis Ag | Organic compounds |
| KR100627687B1 (ko) * | 2005-04-20 | 2006-09-25 | 주식회사 씨티씨바이오 | 시부트라민 유리염기 함유 조성물 및 이의 제조방법 |
| WO2006112649A1 (en) * | 2005-04-20 | 2006-10-26 | Ctc Bio, Inc. | Pharmaceutical composition containing sibutramine free base and manufacturing method thereof |
-
2006
- 2006-12-22 EP EP06126964A patent/EP1938804A1/en not_active Ceased
-
2007
- 2007-12-20 US US12/520,312 patent/US20100015225A1/en not_active Abandoned
- 2007-12-20 NZ NZ576987A patent/NZ576987A/en not_active IP Right Cessation
- 2007-12-20 AR ARP070105788A patent/AR064622A1/es not_active Application Discontinuation
- 2007-12-20 MX MX2009006747A patent/MX2009006747A/es not_active Application Discontinuation
- 2007-12-20 MY MYPI20092111A patent/MY145919A/en unknown
- 2007-12-20 JP JP2009541897A patent/JP2010513356A/ja active Pending
- 2007-12-20 CA CA002672402A patent/CA2672402A1/en not_active Abandoned
- 2007-12-20 WO PCT/EP2007/011293 patent/WO2008077591A2/en not_active Ceased
- 2007-12-20 AU AU2007338359A patent/AU2007338359B2/en not_active Ceased
- 2007-12-20 EA EA200900827A patent/EA200900827A1/ru unknown
- 2007-12-20 CN CNA2007800435054A patent/CN101541309A/zh active Pending
- 2007-12-20 KR KR1020097012819A patent/KR20090092288A/ko not_active Withdrawn
- 2007-12-20 BR BRPI0720937-1A patent/BRPI0720937A2/pt not_active IP Right Cessation
- 2007-12-20 EP EP07857016A patent/EP2117511A2/en not_active Withdrawn
- 2007-12-21 TW TW096149580A patent/TW200848056A/zh unknown
- 2007-12-21 CL CL200703767A patent/CL2007003767A1/es unknown
-
2008
- 2008-01-02 PE PE2008000080A patent/PE20081848A1/es not_active Application Discontinuation
-
2009
- 2009-05-12 ZA ZA200903271A patent/ZA200903271B/xx unknown
- 2009-05-14 IL IL198780A patent/IL198780A0/en unknown
- 2009-06-17 MA MA32008A patent/MA31004B1/fr unknown
- 2009-06-17 CO CO09062883A patent/CO6180497A2/es not_active Application Discontinuation
- 2009-06-19 TN TNP2009000253A patent/TN2009000253A1/fr unknown
- 2009-06-19 GT GT200900173A patent/GT200900173A/es unknown
- 2009-06-22 EC EC2009009450A patent/ECSP099450A/es unknown
- 2009-07-17 NO NO20092722A patent/NO20092722L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| EP1938804A1 (en) | 2008-07-02 |
| MY145919A (en) | 2012-05-15 |
| TW200848056A (en) | 2008-12-16 |
| US20100015225A1 (en) | 2010-01-21 |
| NO20092722L (no) | 2009-07-21 |
| BRPI0720937A2 (pt) | 2014-03-11 |
| MA31004B1 (fr) | 2009-12-01 |
| CA2672402A1 (en) | 2008-07-03 |
| ECSP099450A (es) | 2009-07-31 |
| ZA200903271B (en) | 2010-04-28 |
| WO2008077591A3 (en) | 2009-04-09 |
| CO6180497A2 (es) | 2010-07-19 |
| GT200900173A (es) | 2010-06-24 |
| IL198780A0 (en) | 2010-02-17 |
| AR064622A1 (es) | 2009-04-15 |
| WO2008077591A2 (en) | 2008-07-03 |
| TN2009000253A1 (en) | 2010-10-18 |
| AU2007338359B2 (en) | 2011-04-28 |
| AU2007338359A1 (en) | 2008-07-03 |
| PE20081848A1 (es) | 2009-01-19 |
| JP2010513356A (ja) | 2010-04-30 |
| CN101541309A (zh) | 2009-09-23 |
| EA200900827A1 (ru) | 2009-12-30 |
| CL2007003767A1 (es) | 2008-07-18 |
| EP2117511A2 (en) | 2009-11-18 |
| NZ576987A (en) | 2011-10-28 |
| MX2009006747A (es) | 2009-06-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PA0105 | International application |
Patent event date: 20090619 Patent event code: PA01051R01D Comment text: International Patent Application |
|
| PG1501 | Laying open of application | ||
| PC1203 | Withdrawal of no request for examination | ||
| WITN | Application deemed withdrawn, e.g. because no request for examination was filed or no examination fee was paid |