RS77904A - Oral administration form for difficulty soluble basic active ingredients which are applied orally - Google Patents

Oral administration form for difficulty soluble basic active ingredients which are applied orally

Info

Publication number
RS77904A
RS77904A YU77904A YUP77904A RS77904A RS 77904 A RS77904 A RS 77904A YU 77904 A YU77904 A YU 77904A YU P77904 A YUP77904 A YU P77904A RS 77904 A RS77904 A RS 77904A
Authority
RS
Serbia
Prior art keywords
oral administration
active ingredients
administration form
soluble basic
applied orally
Prior art date
Application number
YU77904A
Other languages
English (en)
Inventor
Ulrich Brauns
Stefan-Rolf Brickl
Original Assignee
Boehringer Ingelheim Pharma Gmbh. & Co.Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma Gmbh. & Co.Kg filed Critical Boehringer Ingelheim Pharma Gmbh. & Co.Kg
Priority to MEP-435/08A priority Critical patent/MEP43508A/xx
Publication of RS77904A publication Critical patent/RS77904A/sr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
    • A61K9/1676—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface having a drug-free core with discrete complete coating layer containing drug
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Hematology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Pronalazak se odnosi na nov oblik za oralnu primenu, delotvorne supstance, čija je rastvorljivost zavisna od pH-vrednosti, i njenih farmakološki podnošljivih soli, koji poboljšava bio-dostupnost delotvorne supstance.
YU77904A 2002-03-07 2003-03-04 Oral administration form for difficulty soluble basic active ingredients which are applied orally RS77904A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
MEP-435/08A MEP43508A (en) 2002-03-07 2003-03-04 Oral administration form for difficulty soluble basic active ingredients which are applied orally

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10209982A DE10209982A1 (de) 2002-03-07 2002-03-07 Oral zu applizierende Darreichungsform für schwerlösliche basische Wirkstoffe
PCT/EP2003/002184 WO2003074032A1 (de) 2002-03-07 2003-03-04 Oral zu applizierende darreichungsform für schwerlösliche basische wirkstoffe

Publications (1)

Publication Number Publication Date
RS77904A true RS77904A (en) 2006-10-27

Family

ID=27771069

Family Applications (1)

Application Number Title Priority Date Filing Date
YU77904A RS77904A (en) 2002-03-07 2003-03-04 Oral administration form for difficulty soluble basic active ingredients which are applied orally

Country Status (10)

Country Link
US (1) US20050095293A1 (sr)
EP (2) EP1499298A1 (sr)
JP (1) JP2005526738A (sr)
AU (1) AU2003229555A1 (sr)
BR (1) BR0308188A (sr)
DE (1) DE10209982A1 (sr)
ME (1) MEP43508A (sr)
NO (1) NO20043998L (sr)
RS (1) RS77904A (sr)
WO (1) WO2003074032A1 (sr)

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US20040048877A1 (en) * 2002-05-22 2004-03-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Pharmaceutical compositions containing flibanserin
DE10339862A1 (de) * 2003-08-29 2005-03-24 Boehringer Ingelheim Pharma Gmbh & Co. Kg 3-[(2-{[4-(Hexyloxycarbonylamino-imino-methyl)- phenylamino]-methyl}-1-methyl-1H-benzimidazol-5-carbonyl)-pyridin-2-yl-amino]-propionsäure-ethylester-Methansulfonat und dessen Verwendung als Arzneimittel
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WO2006125042A1 (en) * 2005-05-19 2006-11-23 Boehringer Ingelheim International Gmbh Method for the treatment of drug-induced sexual dysfunction
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US20070105869A1 (en) * 2005-11-08 2007-05-10 Stephane Pollentier Use of flibanserin for the treatment of pre-menopausal sexual desire disorders
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US20120040008A1 (en) * 2010-08-11 2012-02-16 Ashish Chatterji Pharmaceutical compositions of metabotropic glutamate 5 receptor (mglu5) antagonists
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EP2834224B1 (en) * 2012-04-02 2018-06-06 MSN Laboratories Limited Process for the preparation of benzimidazole derivatives and salts thereof
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Also Published As

Publication number Publication date
EP1499298A1 (de) 2005-01-26
US20050095293A1 (en) 2005-05-05
BR0308188A (pt) 2004-12-21
NO20043998L (no) 2004-10-05
JP2005526738A (ja) 2005-09-08
MEP43508A (en) 2011-02-10
EP1818047A2 (de) 2007-08-15
AU2003229555A1 (en) 2003-09-16
WO2003074032A1 (de) 2003-09-12
EP1818047A3 (de) 2008-08-06
DE10209982A1 (de) 2003-09-25

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