KR20070083705A - 티로신 키나제 수용체 ｃ­ｆｍｓ를 억제하기 위한4-(4-메틸피페라진-1-일메틸)-ｎ-[4-메틸-3-(4-(피리딘-3-일)피리미딘-2-일아미노)페닐]-벤즈아미드의 용도 - Google Patents

티로신 키나제 수용체 ｃ­ｆｍｓ를 억제하기 위한4-(4-메틸피페라진-1-일메틸)-ｎ-[4-메틸-3-(4-(피리딘-3-일)피리미딘-2-일아미노)페닐]-벤즈아미드의 용도 Download PDF

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Publication number
KR20070083705A
KR20070083705A KR1020077008716A KR20077008716A KR20070083705A KR 20070083705 A KR20070083705 A KR 20070083705A KR 1020077008716 A KR1020077008716 A KR 1020077008716A KR 20077008716 A KR20077008716 A KR 20077008716A KR 20070083705 A KR20070083705 A KR 20070083705A
Authority
KR
South Korea
Prior art keywords
compound
fms
csf
carcinoma
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
KR1020077008716A
Other languages
English (en)
Korean (ko)
Inventor
안드레아 루이스 듀어
티모시 피터 휴스
알란 브루스 리온스
Original Assignee
메드벳 싸이언스 피티와이. 리미티드
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 메드벳 싸이언스 피티와이. 리미티드 filed Critical 메드벳 싸이언스 피티와이. 리미티드
Publication of KR20070083705A publication Critical patent/KR20070083705A/ko
Ceased legal-status Critical Current

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
KR1020077008716A 2004-10-18 2005-10-17 티로신 키나제 수용체 ｃ­ｆｍｓ를 억제하기 위한4-(4-메틸피페라진-1-일메틸)-ｎ-[4-메틸-3-(4-(피리딘-3-일)피리미딘-2-일아미노)페닐]-벤즈아미드의 용도 Ceased KR20070083705A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US61974404P 2004-10-18 2004-10-18
US60/619,744 2004-10-18

Publications (1)

Publication Number Publication Date
KR20070083705A true KR20070083705A (ko) 2007-08-24

Family

ID=36202610

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020077008716A Ceased KR20070083705A (ko) 2004-10-18 2005-10-17 티로신 키나제 수용체 ｃ­ｆｍｓ를 억제하기 위한4-(4-메틸피페라진-1-일메틸)-ｎ-[4-메틸-3-(4-(피리딘-3-일)피리미딘-2-일아미노)페닐]-벤즈아미드의 용도

Country Status (19)

Country Link
US (1) US20080255139A1 (https=)
EP (1) EP1804800B1 (https=)
JP (1) JP2008516898A (https=)
KR (1) KR20070083705A (https=)
CN (1) CN101035535A (https=)
AT (1) ATE492277T1 (https=)
AU (1) AU2005297321A1 (https=)
BR (1) BRPI0517083A (https=)
CA (1) CA2580976A1 (https=)
DE (1) DE602005025514D1 (https=)
IL (1) IL182419A0 (https=)
MA (1) MA28946B1 (https=)
MX (1) MX2007004660A (https=)
NO (1) NO20072501L (https=)
NZ (1) NZ554009A (https=)
RU (1) RU2007118420A (https=)
TN (1) TNSN07141A1 (https=)
WO (1) WO2006042362A1 (https=)
ZA (1) ZA200702316B (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009058968A2 (en) * 2007-10-31 2009-05-07 Janssen Pharmaceutica N.V. Biomarker for assessing response to fms treatment
CN107530430A (zh) * 2015-01-13 2018-01-02 国立大学法人京都大学 用于预防和/或治疗肌萎缩性侧索硬化症的药剂

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4837237A (en) * 1985-07-09 1989-06-06 Fred Hutchinson Cancer Research Center Therapy using glucosidase processing inhibitors
DE60212836T2 (de) * 2001-05-16 2007-01-25 Gpc Biotech Ag Pyridylpyrimidin-derivate als wirksame verbindungen gegen prionen-krankheiten
WO2004026930A2 (en) * 2002-06-26 2004-04-01 The Ohio State University Research Foundation The method for reducing inflammation using sti-571 or its salt

Also Published As

Publication number Publication date
AU2005297321A1 (en) 2006-04-27
MA28946B1 (fr) 2007-10-01
DE602005025514D1 (de) 2011-02-03
NO20072501L (no) 2007-05-15
NZ554009A (en) 2010-09-30
JP2008516898A (ja) 2008-05-22
IL182419A0 (en) 2007-09-20
TNSN07141A1 (en) 2008-11-21
EP1804800B1 (en) 2010-12-22
ZA200702316B (en) 2008-09-25
WO2006042362A1 (en) 2006-04-27
CA2580976A1 (en) 2006-04-27
EP1804800A4 (en) 2008-03-19
BRPI0517083A (pt) 2008-09-30
ATE492277T1 (de) 2011-01-15
EP1804800A1 (en) 2007-07-11
RU2007118420A (ru) 2008-11-27
CN101035535A (zh) 2007-09-12
MX2007004660A (es) 2007-10-17
US20080255139A1 (en) 2008-10-16

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