KR20050074493A - 칼륨 채널 및/또는 피질 뉴우런 작용 조절제로서 유용한ｎ-페닐안트라닐산 및/또는 2-벤즈이미다졸론의 유도체 - Google Patents
칼륨 채널 및/또는 피질 뉴우런 작용 조절제로서 유용한ｎ-페닐안트라닐산 및/또는 2-벤즈이미다졸론의 유도체 Download PDFInfo
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- KR20050074493A KR20050074493A KR1020057006856A KR20057006856A KR20050074493A KR 20050074493 A KR20050074493 A KR 20050074493A KR 1020057006856 A KR1020057006856 A KR 1020057006856A KR 20057006856 A KR20057006856 A KR 20057006856A KR 20050074493 A KR20050074493 A KR 20050074493A
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Classifications
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
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- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
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- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
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- Vascular Medicine (AREA)
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- Psychology (AREA)
- Urology & Nephrology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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|---|---|---|---|
| US41952502P | 2002-10-21 | 2002-10-21 | |
| US60/419,525 | 2002-10-21 |
Publications (1)
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| KR20050074493A true KR20050074493A (ko) | 2005-07-18 |
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Family Applications (1)
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| EP (1) | EP1553932A2 (https=) |
| JP (1) | JP2006513154A (https=) |
| KR (1) | KR20050074493A (https=) |
| AU (1) | AU2003272068A1 (https=) |
| CA (1) | CA2503075A1 (https=) |
| WO (1) | WO2004035037A2 (https=) |
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| US7632866B2 (en) | 2002-10-21 | 2009-12-15 | Ramot At Tel Aviv University | Derivatives of N-phenylanthranilic acid and 2-benzimidazolone as potassium channel and/or neuron activity modulators |
| US8765815B2 (en) | 2007-09-20 | 2014-07-01 | Ramot At Tel-Aviv University Ltd. | N-phenyl anthranilic acid derivatives and uses thereof |
| GB0723794D0 (en) | 2007-12-05 | 2008-01-16 | Lectus Therapeutics Ltd | Potassium ion channel modulators and uses thereof |
| GB0813403D0 (en) * | 2008-07-22 | 2008-08-27 | Lectus Therapeutics Ltd | Potassium ion channel modulators & uses thereof |
| CA3077659A1 (en) | 2017-10-09 | 2019-04-18 | Ramot At Tel-Aviv University Ltd. | Modulators of potassium ion and trpv1 channels and uses thereof |
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| JPS5032189A (https=) * | 1973-07-20 | 1975-03-28 | ||
| JPS5095285A (https=) * | 1973-12-26 | 1975-07-29 | ||
| JPH05132431A (ja) * | 1990-03-28 | 1993-05-28 | Nippon Oil & Fats Co Ltd | 高分子化薬剤およびその製造法 |
| US5565483A (en) * | 1995-06-07 | 1996-10-15 | Bristol-Myers Squibb Company | 3-substituted oxindole derivatives as potassium channel modulators |
| ITMI962356A1 (it) * | 1996-11-13 | 1998-05-13 | Uni Degli Studi Di Brescia D I | Uso di composti derivati da molecole ad attivita' antinfiammatoria di tipo non steroideo per la prevenzione e il trattamento di |
| CA2290509A1 (en) * | 1997-07-01 | 1999-01-14 | Warner-Lambert Company | 2-(4-bromo or 4-iodo phenylamino) benzoic acid derivatives and their use as mek inhibitors |
| US6291442B1 (en) * | 1998-02-03 | 2001-09-18 | The General Hospital Corporation | Pharmacological modulators of voltage-gated potassium ion channels |
| EP1144387A1 (en) * | 1998-12-04 | 2001-10-17 | Neurosearch A/S | New benzimidazolone-, benzoxazolone-, or benzothiazolone derivatives as ion channel modulating agents |
| US6472165B1 (en) * | 1999-08-03 | 2002-10-29 | Arzneimittelwerk Dresden Gmbh | Modulatory binding site in potassium channels for screening and finding new active ingredients |
| US6713454B1 (en) * | 1999-09-13 | 2004-03-30 | Nobex Corporation | Prodrugs of etoposide and etoposide analogs |
| US6413507B1 (en) * | 1999-12-23 | 2002-07-02 | Shearwater Corporation | Hydrolytically degradable carbamate derivatives of poly (ethylene glycol) |
| AU5702201A (en) * | 2000-04-13 | 2001-10-30 | Mayo Foundation | Abeta<sub>42</sub> lowering agents |
| US6429223B1 (en) * | 2000-06-23 | 2002-08-06 | Medinox, Inc. | Modified forms of pharmacologically active agents and uses therefor |
| TWI287984B (en) * | 2000-10-17 | 2007-10-11 | Wyeth Corp | Pharmaceutical composition for modulating bladder function |
| GB0026838D0 (en) * | 2000-11-02 | 2000-12-20 | Glaxo Group Ltd | Treatment method |
| US6593349B2 (en) * | 2001-03-19 | 2003-07-15 | Icagen, Inc. | Bisarylamines as potassium channel openers |
| US8765815B2 (en) * | 2007-09-20 | 2014-07-01 | Ramot At Tel-Aviv University Ltd. | N-phenyl anthranilic acid derivatives and uses thereof |
-
2003
- 2003-10-21 KR KR1020057006856A patent/KR20050074493A/ko not_active Ceased
- 2003-10-21 JP JP2004544675A patent/JP2006513154A/ja active Pending
- 2003-10-21 WO PCT/IL2003/000855 patent/WO2004035037A2/en not_active Ceased
- 2003-10-21 EP EP03753909A patent/EP1553932A2/en not_active Withdrawn
- 2003-10-21 CA CA002503075A patent/CA2503075A1/en not_active Abandoned
- 2003-10-21 AU AU2003272068A patent/AU2003272068A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2004035037A2 (en) | 2004-04-29 |
| CA2503075A1 (en) | 2004-04-29 |
| AU2003272068A1 (en) | 2004-05-04 |
| JP2006513154A (ja) | 2006-04-20 |
| AU2003272068A8 (en) | 2004-05-04 |
| WO2004035037A3 (en) | 2004-06-03 |
| EP1553932A2 (en) | 2005-07-20 |
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