KR20010043216A - 1-(6-클로로나프트-2-일설포닐)-4-[4-(4-피리딜)벤조일]피페라진의 입도가 감소된 제형 - Google Patents

1-(6-클로로나프트-2-일설포닐)-4-[4-(4-피리딜)벤조일]피페라진의 입도가 감소된 제형 Download PDF

Info

Publication number
KR20010043216A
KR20010043216A KR1020007012149A KR20007012149A KR20010043216A KR 20010043216 A KR20010043216 A KR 20010043216A KR 1020007012149 A KR1020007012149 A KR 1020007012149A KR 20007012149 A KR20007012149 A KR 20007012149A KR 20010043216 A KR20010043216 A KR 20010043216A
Authority
KR
South Korea
Prior art keywords
chloronaphth
pyridyl
benzoyl
piperazine
ylsulfonyl
Prior art date
Application number
KR1020007012149A
Other languages
English (en)
Korean (ko)
Inventor
애쉬포드매리앤
제임즈라저
Original Assignee
다비드 에 질레스
아스트라제네카 아베
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 다비드 에 질레스, 아스트라제네카 아베 filed Critical 다비드 에 질레스
Publication of KR20010043216A publication Critical patent/KR20010043216A/ko

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
KR1020007012149A 1998-05-02 1999-04-27 1-(6-클로로나프트-2-일설포닐)-4-[4-(4-피리딜)벤조일]피페라진의 입도가 감소된 제형 KR20010043216A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB9809350.3 1998-05-02
GBGB9809350.3A GB9809350D0 (en) 1998-05-02 1998-05-02 Novel salt
PCT/GB1999/001316 WO1999057112A1 (en) 1998-05-02 1999-04-27 Reduced particle size form of 1-(6-chloronaphth-2- ylsulphonyl) -4-[4-(4pyridyl) benzoyl] piperazine

Publications (1)

Publication Number Publication Date
KR20010043216A true KR20010043216A (ko) 2001-05-25

Family

ID=10831311

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020007012149A KR20010043216A (ko) 1998-05-02 1999-04-27 1-(6-클로로나프트-2-일설포닐)-4-[4-(4-피리딜)벤조일]피페라진의 입도가 감소된 제형

Country Status (16)

Country Link
EP (1) EP1084118A1 (ja)
JP (1) JP2002513789A (ja)
KR (1) KR20010043216A (ja)
CN (1) CN1308629A (ja)
AU (1) AU3719699A (ja)
BR (1) BR9910176A (ja)
CA (1) CA2331041A1 (ja)
EE (1) EE200000638A (ja)
GB (1) GB9809350D0 (ja)
HU (1) HUP0102394A3 (ja)
IL (1) IL139405A0 (ja)
NO (1) NO20005498D0 (ja)
PL (1) PL343705A1 (ja)
SK (1) SK16522000A3 (ja)
WO (1) WO1999057112A1 (ja)
ZA (1) ZA200006036B (ja)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69833036T2 (de) * 1997-09-30 2006-06-22 Daiichi Pharmaceutical Co., Ltd. Sulfonylderivate
TWI290136B (en) 2000-04-05 2007-11-21 Daiichi Seiyaku Co Ethylenediamine derivatives
WO2003000657A1 (fr) 2001-06-20 2003-01-03 Daiichi Pharmaceutical Co., Ltd. Derives de diamine
DK1569912T3 (en) 2002-12-03 2015-06-29 Pharmacyclics Inc 2- (2-hydroxybiphenyl-3-yl) -1h-benzoimidazole-5-carboxamidine derivatives as factor VIIa inhibitors.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA56197C2 (uk) * 1996-11-08 2003-05-15 Зенека Лімітед Гетероциклічні похідні
ATE334975T1 (de) * 1997-05-30 2006-08-15 Takeda Pharmaceutical Sulfonamidderivate, ihre herstellung und verwendung
DE69833036T2 (de) * 1997-09-30 2006-06-22 Daiichi Pharmaceutical Co., Ltd. Sulfonylderivate

Also Published As

Publication number Publication date
SK16522000A3 (sk) 2001-05-10
WO1999057112A1 (en) 1999-11-11
EE200000638A (et) 2002-04-15
HUP0102394A2 (hu) 2001-12-28
HUP0102394A3 (en) 2003-01-28
ZA200006036B (en) 2002-01-25
IL139405A0 (en) 2001-11-25
NO20005498L (no) 2000-11-01
JP2002513789A (ja) 2002-05-14
BR9910176A (pt) 2001-01-09
GB9809350D0 (en) 1998-07-01
NO20005498D0 (no) 2000-11-01
CN1308629A (zh) 2001-08-15
CA2331041A1 (en) 1999-11-11
EP1084118A1 (en) 2001-03-21
AU3719699A (en) 1999-11-23
PL343705A1 (en) 2001-08-27

Similar Documents

Publication Publication Date Title
CA2552786C (en) Crystalline polymorph of a bisulfate salt of a thrombin receptor antagonist
EP0288973B1 (en) Benzothiazolinone derivatives, their production and pharmaceutical composition
CN103119030A (zh) 基质金属蛋白酶抑制剂
CZ293126B6 (cs) Léčivo k léčení schizofrenie, deprese, neuróz a psychóz
RU2385325C2 (ru) Способ получения сульфата атазанавира
BG102948A (bg) Пиразинони като инхибитори на тромбин
JP2015232046A (ja) 第Xa因子阻害剤の結晶形態
PL207651B1 (pl) Pochodne diazepanu lub ich sole i zawierające je kompozycja farmaceutyczna oraz inhibitor aktywowanego czynnika krzepnięcia krwi X
EA015376B1 (ru) СОЛИ ПРОИЗВОДНЫХ 6-ГЕТЕРОАРИЛ-(1,2,3,4,4a,10b)-ГЕКСАГИДРОФЕНАНТРИДИНА И ИХ ПРИМЕНЕНИЕ
TW200402416A (en) Novel piperidine derivatives
EP2138482A1 (en) Bicyclic heterocyclic compound
AU687128B2 (en) Prodrugs of an inhibitor of HIV protease
JP4230453B2 (ja) 1−メチル−2−(4−アミジノフェニルアミノメチル)−ベンズイミダゾール−5−イル−カルボン酸−(n−2−ピリジル−n−2−ヒドロキシカルボニルエチル)−アミドの新規プロドラッグ、それらの製造及び医薬組成物としてのそれらの使用
EP0228959B1 (en) Aminostyryl compound, leukotriene antagonistic composition containing the same as effective ingredients and method of antagonizing srs by employing the same
KR20040015087A (ko) 만성 관절 류마티즘 치료제
JP4248245B2 (ja) 6−フェニルベンゾナフチリジン
WO2000048996A2 (de) Beta-alaninderivate
KR19980703601A (ko) 당단백질 IIb/IIIa 길항제
KR20220152293A (ko) Covid-19 관련 병태의 치료 방법
KR20010043216A (ko) 1-(6-클로로나프트-2-일설포닐)-4-[4-(4-피리딜)벤조일]피페라진의 입도가 감소된 제형
JPS63225355A (ja) 1,4−ジヒドロピリジン誘導体
WO2001017990A1 (en) Heterocyclic derivatives as inhibitors of factor xa
CZ20004037A3 (cs) Forma l-(6-chlornaft-2-ylsulfonyl)-4-[4-(4- pyridyl)benzoyl]piperazinu se zmenšenu velikostí částic a farmaceutická kompozice tuto formu obsahující
MXPA00010676A (en) Reduced particle size form of 1-(6-chloronaphth-2- ylsulphonyl) -4-[4-(4pyridyl) benzoyl]piperazine
CN113105391B (zh) 一种具有镇痛活性的高乌甲素衍生物及其制备方法和应用

Legal Events

Date Code Title Description
WITN Application deemed withdrawn, e.g. because no request for examination was filed or no examination fee was paid