KR101919259B1 - 3-아릴옥시퀴놀린 유도체의 제조 방법 - Google Patents

3-아릴옥시퀴놀린 유도체의 제조 방법 Download PDF

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Publication number
KR101919259B1
KR101919259B1 KR1020177008909A KR20177008909A KR101919259B1 KR 101919259 B1 KR101919259 B1 KR 101919259B1 KR 1020177008909 A KR1020177008909 A KR 1020177008909A KR 20177008909 A KR20177008909 A KR 20177008909A KR 101919259 B1 KR101919259 B1 KR 101919259B1
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KR
South Korea
Prior art keywords
group
derivative
present
solvent
aryloxyquinoline
Prior art date
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KR1020177008909A
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English (en)
Korean (ko)
Other versions
KR20170044201A (ko
Inventor
마사오 야마구치
료지 와다
Original Assignee
닛뽕소다 가부시키가이샤
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Publication of KR20170044201A publication Critical patent/KR20170044201A/ko
Application granted granted Critical
Publication of KR101919259B1 publication Critical patent/KR101919259B1/ko

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20Oxygen atoms
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A01N43/42Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B61/00Other general methods

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Epidemiology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Quinoline Compounds (AREA)
KR1020177008909A 2014-10-06 2015-10-02 3-아릴옥시퀴놀린 유도체의 제조 방법 KR101919259B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JPJP-P-2014-206000 2014-10-06
JP2014206000 2014-10-06
PCT/JP2015/078019 WO2016056475A1 (ja) 2014-10-06 2015-10-02 3-アリールオキシキノリン誘導体の製造方法

Publications (2)

Publication Number Publication Date
KR20170044201A KR20170044201A (ko) 2017-04-24
KR101919259B1 true KR101919259B1 (ko) 2018-11-15

Family

ID=55653087

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020177008909A KR101919259B1 (ko) 2014-10-06 2015-10-02 3-아릴옥시퀴놀린 유도체의 제조 방법

Country Status (5)

Country Link
JP (2) JPWO2016056475A1 (ja)
KR (1) KR101919259B1 (ja)
CN (1) CN107108509A (ja)
IL (1) IL251471B (ja)
WO (1) WO2016056475A1 (ja)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1917245A1 (de) * 2005-08-21 2008-05-07 Abbott GmbH & Co. KG Heterocyclische verbindungen und ihre verwendung als bindungspartner für 5-ht5-rezeptoren
WO2010058314A1 (en) * 2008-11-18 2010-05-27 Pfizer Inc. Hydroxyquinolin-2(1h)-ones and derivatives thereof
SI2522658T1 (sl) * 2010-01-04 2018-12-31 Nippon Soda Co., Ltd. Dušik-vsebujoča heterociklična spojina in kmetijski/hortikulturni germicid
JP2014166991A (ja) * 2013-01-31 2014-09-11 Nippon Soda Co Ltd 含窒素ヘテロ環化合物および農園芸用殺菌剤

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
"Optimization of the Reaction Conditions for Synthesis of 3-(aryloxy)quinoline Derivatives via Friedlander’s Cyclization Reaction", Bull. Korean Chem. Soc., 2013, Vol.34, No.6, pp.1848-1852*

Also Published As

Publication number Publication date
CN107108509A (zh) 2017-08-29
JP2019006804A (ja) 2019-01-17
JPWO2016056475A1 (ja) 2017-07-06
IL251471B (en) 2020-07-30
KR20170044201A (ko) 2017-04-24
WO2016056475A1 (ja) 2016-04-14
JP6621888B2 (ja) 2019-12-18
IL251471A0 (en) 2017-05-29

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