KR101919259B1 - 3-아릴옥시퀴놀린 유도체의 제조 방법 - Google Patents
3-아릴옥시퀴놀린 유도체의 제조 방법 Download PDFInfo
- Publication number
- KR101919259B1 KR101919259B1 KR1020177008909A KR20177008909A KR101919259B1 KR 101919259 B1 KR101919259 B1 KR 101919259B1 KR 1020177008909 A KR1020177008909 A KR 1020177008909A KR 20177008909 A KR20177008909 A KR 20177008909A KR 101919259 B1 KR101919259 B1 KR 101919259B1
- Authority
- KR
- South Korea
- Prior art keywords
- group
- derivative
- present
- solvent
- aryloxyquinoline
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
- A01N43/42—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B61/00—Other general methods
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Epidemiology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Plant Pathology (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Quinoline Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2014206000 | 2014-10-06 | ||
JPJP-P-2014-206000 | 2014-10-06 | ||
PCT/JP2015/078019 WO2016056475A1 (ja) | 2014-10-06 | 2015-10-02 | 3-アリールオキシキノリン誘導体の製造方法 |
Publications (2)
Publication Number | Publication Date |
---|---|
KR20170044201A KR20170044201A (ko) | 2017-04-24 |
KR101919259B1 true KR101919259B1 (ko) | 2018-11-15 |
Family
ID=55653087
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
KR1020177008909A KR101919259B1 (ko) | 2014-10-06 | 2015-10-02 | 3-아릴옥시퀴놀린 유도체의 제조 방법 |
Country Status (5)
Country | Link |
---|---|
JP (2) | JPWO2016056475A1 (ja) |
KR (1) | KR101919259B1 (ja) |
CN (1) | CN107108509A (ja) |
IL (1) | IL251471B (ja) |
WO (1) | WO2016056475A1 (ja) |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2007022946A1 (de) * | 2005-08-21 | 2007-03-01 | Abbott Gmbh & Co. Kg | Heterocyclische verbindungen und ihre verwendung als bindungspartner für 5-ht5-rezeptoren |
WO2010058314A1 (en) * | 2008-11-18 | 2010-05-27 | Pfizer Inc. | Hydroxyquinolin-2(1h)-ones and derivatives thereof |
DK2522658T3 (en) * | 2010-01-04 | 2018-11-19 | Nippon Soda Co | NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS AND AGRICULTURAL / Horticulture Bactericidal Agents |
JP2014166991A (ja) * | 2013-01-31 | 2014-09-11 | Nippon Soda Co Ltd | 含窒素ヘテロ環化合物および農園芸用殺菌剤 |
-
2015
- 2015-10-02 JP JP2016553078A patent/JPWO2016056475A1/ja active Pending
- 2015-10-02 KR KR1020177008909A patent/KR101919259B1/ko active IP Right Grant
- 2015-10-02 CN CN201580053799.3A patent/CN107108509A/zh active Pending
- 2015-10-02 WO PCT/JP2015/078019 patent/WO2016056475A1/ja active Application Filing
-
2017
- 2017-03-30 IL IL251471A patent/IL251471B/en active IP Right Grant
-
2018
- 2018-09-03 JP JP2018164142A patent/JP6621888B2/ja active Active
Non-Patent Citations (1)
Title |
---|
"Optimization of the Reaction Conditions for Synthesis of 3-(aryloxy)quinoline Derivatives via Friedlander’s Cyclization Reaction", Bull. Korean Chem. Soc., 2013, Vol.34, No.6, pp.1848-1852* |
Also Published As
Publication number | Publication date |
---|---|
JPWO2016056475A1 (ja) | 2017-07-06 |
KR20170044201A (ko) | 2017-04-24 |
IL251471A0 (en) | 2017-05-29 |
JP2019006804A (ja) | 2019-01-17 |
CN107108509A (zh) | 2017-08-29 |
JP6621888B2 (ja) | 2019-12-18 |
WO2016056475A1 (ja) | 2016-04-14 |
IL251471B (en) | 2020-07-30 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
US10125122B2 (en) | Method for preparing methyl (Z)-3-[[[4-[methyl[2-(4-methyl-1-piperazinyl)acetyl]amino]phenyl]amino]phenylmethylene)oxindole-6-carboxylate (intedanib, nintedanib) | |
Rad-Moghadam et al. | Synthesis of novel pyrano [3, 2-c] quinoline-2, 5-diones using an acidic ionic liquid catalyst | |
Ninomiya et al. | Total synthesis of actinorhodin | |
Xie et al. | Intrinsically safe and shelf-stable diazo-transfer reagent for fast synthesis of diazo compounds | |
WO2020127945A1 (en) | Process and intermediates for the synthesis of voxelotor | |
Hawaiz et al. | One-pot three-component synthesis of some new azo-pyrazoline derivatives | |
Asahara et al. | Cyclodextrin host as a supramolecular catalyst in nonpolar solvents: stereoselective synthesis of (E)-3-alkylideneoxindoles | |
Kalita et al. | FeCl 3· 6H 2 O catalyzed aqueous media domino synthesis of 5-monoalkylbarbiturates: water as both reactant and solvent | |
Liu et al. | Synthesis, Crystal Structure, and Fungicidal Activity of Novel 1, 5‐Diaryl‐1H‐Pyrazol‐3‐Oxy Derivatives Containing Oxyacetic Acid or Oxy (2‐thioxothiazolidin‐3‐yl) ethanone Moieties | |
CN107629001B (zh) | 一种抗癌药物乐伐替尼的合成方法 | |
KR101919259B1 (ko) | 3-아릴옥시퀴놀린 유도체의 제조 방법 | |
Xu et al. | Modular synthesis of (E)-cinnamaldehydes directly from allylarenes via a metal-free DDQ-mediated oxidative process | |
WO2011086570A1 (en) | Process for preparation of cyanoalkylpropionate derivatives | |
JP7117968B2 (ja) | ヒドロキシ酸の製造方法。 | |
Osipov et al. | Synthesis of 8-substituted 1, 5-diazabicyclo [3.2. 1] octane derivatives via double aza-Michael addition of homopiperazine to 3-trifluoroacetyl-4H-chromenes | |
KR20130090360A (ko) | 물 또는 다양한 산을 첨가제로 이용한 새로운 마이클-첨가 반응을 통하여 화합물을 제조하는 방법 | |
EP4434970A1 (en) | Method for producing halovinyl imidazole compound | |
US11267787B2 (en) | Method for producing quinolin-4(1H)-one derivative | |
CN109422690A (zh) | 一种制备1-烷基-3-烷基吡唑-5-甲酸酯的方法 | |
BR112021016834A2 (pt) | Método de produção de um éster de ácido dicarboxílico a,ss-insaturado representado pela fórmula geral | |
JPH0240365A (ja) | N‐ヒドロキシピラゾールの製法 | |
US9029591B2 (en) | Gem-dinitro ester compound as energetic material and preparation method thereof | |
CN105440042B (zh) | 一种pp796中间体嘧啶三唑的合成方法 | |
CN109369606A (zh) | 一种乙酰化二苯并-1,3-二氧杂环辛类化合物的制备方法与作为抗菌药物的应用 | |
CN105801487B (zh) | 一种4-甲氨基安替比林的制备方法 |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
A201 | Request for examination | ||
E902 | Notification of reason for refusal | ||
E701 | Decision to grant or registration of patent right |