KR100908350B1 - 남성의 사정을 지연시키기 위한 약학 조성물 - Google Patents

남성의 사정을 지연시키기 위한 약학 조성물 Download PDF

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Publication number
KR100908350B1
KR100908350B1 KR1020037012090A KR20037012090A KR100908350B1 KR 100908350 B1 KR100908350 B1 KR 100908350B1 KR 1020037012090 A KR1020037012090 A KR 1020037012090A KR 20037012090 A KR20037012090 A KR 20037012090A KR 100908350 B1 KR100908350 B1 KR 100908350B1
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South Korea
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tramadol
pharmaceutical composition
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ejaculation
pharmaceutically acceptable
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Korean (ko)
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KR20040052490A (ko
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데이비드 바-오
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디엠아이 바이오사이언스 인코포레이티드
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Assigned to 아이트 바이오사이언스, 아이엔씨. reassignment 아이트 바이오사이언스, 아이엔씨. 권리의 전부이전등록 Assignors: 디엠아이 바이오사이언시스 인코포레이티드
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis

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  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Reproductive Health (AREA)
  • Emergency Medicine (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Fats And Perfumes (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Liquid Crystal Substances (AREA)
  • Materials For Photolithography (AREA)
  • Medicinal Preparation (AREA)
KR1020037012090A 2001-03-16 2002-03-15 남성의 사정을 지연시키기 위한 약학 조성물 Expired - Fee Related KR100908350B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US27680601P 2001-03-16 2001-03-16
US60/276,806 2001-03-16
PCT/US2002/007928 WO2002074241A2 (en) 2001-03-16 2002-03-15 Method of delaying ejaculation

Publications (2)

Publication Number Publication Date
KR20040052490A KR20040052490A (ko) 2004-06-23
KR100908350B1 true KR100908350B1 (ko) 2009-07-20

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ID=23058139

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KR1020037012090A Expired - Fee Related KR100908350B1 (ko) 2001-03-16 2002-03-15 남성의 사정을 지연시키기 위한 약학 조성물

Country Status (17)

Country Link
US (2) US6974839B2 (https=)
EP (1) EP1397126B9 (https=)
JP (1) JP4377585B2 (https=)
KR (1) KR100908350B1 (https=)
CN (1) CN1289071C (https=)
AT (1) ATE326957T1 (https=)
AU (1) AU2002252361C1 (https=)
CA (2) CA2758923A1 (https=)
CY (1) CY1107478T1 (https=)
DE (1) DE60211689T2 (https=)
DK (1) DK1397126T5 (https=)
ES (1) ES2265495T3 (https=)
MX (1) MXPA03008372A (https=)
NZ (1) NZ528935A (https=)
PT (1) PT1397126E (https=)
WO (1) WO2002074241A2 (https=)
ZA (1) ZA200308067B (https=)

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EP1397126B9 (en) * 2001-03-16 2007-02-21 DMI Biosciences, Inc. Use of tramadol for delaying ejaculation
US8575169B2 (en) 2001-10-29 2013-11-05 Versi Group, Llc Method of treating sexual dysfunctions with delta opioid receptor agonist compounds
AU2003291302A1 (en) * 2002-11-06 2004-06-03 Azaya Therapeutics, Inc. Method for treatment of premature ejaculation in humans
WO2004078143A2 (en) * 2003-03-05 2004-09-16 The Brigham And Women's Hospital Inc. Methods for identification and uses of anti-inflammatory receptors for eicosapentaenoic acid analogs
BRPI0408454A (pt) 2003-03-21 2006-04-04 Nexmed Holdings Inc composição tópica, método de tratar a ejaculação precoce, e, uso da composição
AU2003903597A0 (en) * 2003-07-11 2003-07-24 Jakov Vaisman Treatment of premature ejaculation
JP5528705B2 (ja) * 2005-12-13 2014-06-25 トリニティ ラボラトリーズ インコーポレイテッド ヒトにおける早漏を治療するための方法
FR2907121B1 (fr) 2006-10-12 2012-05-04 Neorphys Nouveaux derives morphiniques
CN101674728A (zh) * 2007-02-12 2010-03-17 Dmi生物科学公司 降低曲马多的副作用
CN101657101B (zh) * 2007-02-12 2013-12-11 Dmi生物科学公司 并存早泄和勃起功能障碍的治疗
WO2008131256A1 (en) * 2007-04-19 2008-10-30 Trinity Laboratories Inc. Improved treatments for premature ejaculation in humans
US20090005319A1 (en) * 2007-07-01 2009-01-01 Barone Jr Frank V Topical compositions for delaying ejaculation and methods of using the same
KR101103118B1 (ko) * 2007-11-02 2012-01-04 동아제약주식회사 신규한 1,3-디히드로-5-이소벤조퓨란카르보니트릴 유도체 화합물 및 이를 함유하는 조루증 치료용 약학조성물
US8147848B2 (en) 2009-08-26 2012-04-03 Allergan, Inc. Method for treating premature ejaculation with a botulinum neurotoxin
GR1007315B (el) * 2010-04-19 2011-06-14 Uni-Pharma Κλεων Τσετης Φαρμακευτικα Εργαστηρια Αβεε Με Δ.Τ. Uni-Pharma Abee, Υγρομορφη παρεντερικης χορηγησης συνθεση που περιλαμβανει τραμαδολη hci και παρακεταμολη
US10702485B2 (en) 2011-07-09 2020-07-07 Syntrix Biosystems Inc. Compositions and methods for overcoming resistance to tramadol
US20180071269A1 (en) 2015-08-12 2018-03-15 Tianxin Wang Therapeutical methods, formulations and nutraceutical formulations
US11000488B2 (en) 2019-03-22 2021-05-11 Syntrix Biosystems Inc. Treating pain using desmetramadol

Citations (1)

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US5929122A (en) 1996-10-09 1999-07-27 Gruenenthal Gmbh Combination preparation containing tramadol and a calcium channel antagonist

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AU657351B2 (en) 1991-09-06 1995-03-09 Mcneilab, Inc. Compositions comprising a tramadol material and any of codeine, oxycodone or hydrocodone and their use
CA2095523C (en) 1991-09-06 2004-06-22 Robert B. Raffa Composition comprising a tramadol material and acetaminophen and its use
US5223541A (en) 1991-09-13 1993-06-29 Mcneilab, Inc. Tramadol n-oxide material, enantiomers and compositions thereof, and their use
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DE4329794C2 (de) 1993-09-03 1997-09-18 Gruenenthal Gmbh Tramadolsalz enthaltende Arzneimittel mit verzögerter Wirkstofffreisetzung
IT1264965B1 (it) 1993-11-12 1996-10-17 Giorgio Cavallini Uso di alfa 1-bloccanti nel trattamento della eiaculazione precoce
US6017963A (en) * 1995-11-14 2000-01-25 Euro-Celtique, S.A. Formulation for intranasal administration
DE19547766A1 (de) 1995-12-20 1997-06-26 Gruenenthal Gmbh 1-Phenyl-2-dimethylaminomethyl-cyclohexan-1-ol-verbindungen als pharmazeutische Wirkstoffe
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US5929122A (en) 1996-10-09 1999-07-27 Gruenenthal Gmbh Combination preparation containing tramadol and a calcium channel antagonist

Also Published As

Publication number Publication date
HK1068549A1 (en) 2005-04-29
JP2004532828A (ja) 2004-10-28
DE60211689D1 (de) 2006-06-29
EP1397126A2 (en) 2004-03-17
WO2002074241A2 (en) 2002-09-26
WO2002074241A3 (en) 2003-12-24
ES2265495T3 (es) 2007-02-16
ZA200308067B (en) 2005-03-30
DE60211689T2 (de) 2007-01-11
US20020132857A1 (en) 2002-09-19
CN1520289A (zh) 2004-08-11
DK1397126T5 (da) 2007-05-21
AU2002252361C1 (en) 2006-03-30
MXPA03008372A (es) 2004-11-12
EP1397126B2 (en) 2006-05-31
NZ528935A (en) 2004-10-29
CA2440920C (en) 2012-01-24
CA2758923A1 (en) 2002-09-26
EP1397126B9 (en) 2007-02-21
US20060106113A1 (en) 2006-05-18
CN1289071C (zh) 2006-12-13
ATE326957T1 (de) 2006-06-15
KR20040052490A (ko) 2004-06-23
US6974839B2 (en) 2005-12-13
DK1397126T3 (da) 2006-10-02
JP4377585B2 (ja) 2009-12-02
EP1397126B1 (en) 2006-05-24
CA2440920A1 (en) 2002-09-26
PT1397126E (pt) 2006-10-31
EP1397126A4 (en) 2005-02-16
CY1107478T1 (el) 2013-03-13
AU2002252361B2 (en) 2005-09-08

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