KR100708444B1 - 치환된 벤즈이미다졸, 이들의 제조방법 및 기생원생동물에 대한 약제로서의 용도 - Google Patents

치환된 벤즈이미다졸, 이들의 제조방법 및 기생원생동물에 대한 약제로서의 용도 Download PDF

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KR100708444B1
KR100708444B1 KR1020017013296A KR20017013296A KR100708444B1 KR 100708444 B1 KR100708444 B1 KR 100708444B1 KR 1020017013296 A KR1020017013296 A KR 1020017013296A KR 20017013296 A KR20017013296 A KR 20017013296A KR 100708444 B1 KR100708444 B1 KR 100708444B1
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South Korea
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ameria
compound
active compound
mol
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KR20020008839A (ko
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그라이프기젤라
하버코른악셀
바스너베른트
리브폴커
마홀트알브레흐트
스퇼팅죄른
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바이엘 악티엔게젤샤프트
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C07D491/056—Ortho-condensed systems with two or more oxygen atoms as ring hetero atoms in the oxygen-containing ring

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
KR1020017013296A 1999-05-05 2000-04-26 치환된 벤즈이미다졸, 이들의 제조방법 및 기생원생동물에 대한 약제로서의 용도 Expired - Fee Related KR100708444B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19920551A DE19920551A1 (de) 1999-05-05 1999-05-05 Substituierte Benzimidazole, ihre Herstellung und ihre Verwendung als Mittel gegen parasitäre Protozoen
DE19920551.5 1999-05-05
PCT/EP2000/003714 WO2000068225A1 (de) 1999-05-05 2000-04-26 Substituierte benzimidazole, ihre herstellung und ihre verwendung als mittel gegen parasitäre protozoen

Publications (2)

Publication Number Publication Date
KR20020008839A KR20020008839A (ko) 2002-01-31
KR100708444B1 true KR100708444B1 (ko) 2007-04-18

Family

ID=7906972

Family Applications (1)

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KR1020017013296A Expired - Fee Related KR100708444B1 (ko) 1999-05-05 2000-04-26 치환된 벤즈이미다졸, 이들의 제조방법 및 기생원생동물에 대한 약제로서의 용도

Country Status (17)

Country Link
US (1) US6569881B1 (enExample)
EP (1) EP1177191B1 (enExample)
JP (1) JP2002544129A (enExample)
KR (1) KR100708444B1 (enExample)
CN (1) CN1130359C (enExample)
AT (1) ATE256124T1 (enExample)
AU (1) AU761553B2 (enExample)
BR (1) BR0010699A (enExample)
CA (1) CA2372664C (enExample)
DE (2) DE19920551A1 (enExample)
DK (1) DK1177191T3 (enExample)
ES (1) ES2213024T3 (enExample)
HK (1) HK1046143B (enExample)
HU (1) HUP0201035A3 (enExample)
NZ (1) NZ515243A (enExample)
WO (1) WO2000068225A1 (enExample)
ZA (1) ZA200107985B (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10049468A1 (de) * 2000-10-06 2002-04-11 Bayer Ag N-Alkoxyalkyl-substituierte Benzimidazole, ihre Herstellung und ihre Verwendung als Mittel gegen parasitäre Protozoen
DE10131149A1 (de) * 2001-06-28 2003-01-16 Bayer Ag Substituierte Benzinmidazole zur Bekämpfung von Endoparasiten
DE102004042958A1 (de) * 2004-09-02 2006-03-09 Bayer Healthcare Ag Neue antiparasitäre Kombination von Wirkstoffen
DE102005000746A1 (de) * 2005-01-05 2006-07-13 Bayer Healthcare Ag Bekämpfung der Histomoniasis
DE102009038950A1 (de) 2009-08-26 2011-03-03 Bayer Animal Health Gmbh Neue antiparasitäre Kombination von Wirkstoffen
RU2477129C1 (ru) * 2011-07-19 2013-03-10 Государственное научное учреждение Северо-Кавказский зональный научно-исследовательский ветеринарный институт (ГНУ СКЗНИВИ) Российской академии сельскохозяйственных наук Способ лечения кокцидиоза (эймериоза) сельскохозяйственных животных и птиц
CN105237480B (zh) * 2015-08-14 2017-12-05 三峡大学 一种2‑三氟甲基苯并咪唑化合物及其制备方法
CN115768426B (zh) * 2020-07-03 2025-03-07 日本农药株式会社 球虫病防治剂和球虫病防治剂的使用方法

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1122988A (en) 1964-10-22 1968-08-07 Fisons Pest Control Ltd Benzimidazole derivatives
GB1163262A (en) 1966-01-13 1969-09-04 Fisons Pest Control Ltd Substituted Benzimidazoles and Biocidally Active Compositions
NL7013343A (enExample) * 1969-09-26 1971-03-30
JPS6019908B2 (ja) * 1980-04-30 1985-05-18 カネボウ株式会社 １，３−ジオキソレン−２−オン誘導体
FR2521141A1 (fr) 1982-02-09 1983-08-12 Rhone Poulenc Agrochimie Nouveaux derives du cyano-2 benzimidazole, leur preparation et leur utilisation comme fongicides
JPS58152879A (ja) * 1982-03-05 1983-09-10 Mitsubishi Chem Ind Ltd ４−ブロムメチル−５−メチル−１，３−ジオキソ−ル−２−オンの製法
US4434173A (en) * 1982-08-23 1984-02-28 Pfizer Inc. Bis-esters of 4,5-di(hydroxymethyl)-2-oxo-1,3-dioxole as antibacterial agents
US4448732A (en) * 1982-09-07 1984-05-15 Pfizer Inc. 2-Oxo-1,3-dioxol-4-ylmethyl esters of penicillanic acid 1,1-dioxide
FR2559150B1 (fr) 1984-02-06 1986-06-27 Rhone Poulenc Agrochimie Nouveaux derives du cyano-2 benzimidazole, leur preparation et leur utilisation comme fongicides
FR2572401B1 (fr) 1984-10-26 1986-12-26 Rhone Poulenc Agrochimie Nouveaux derives du cyano-2 benzimidazole, leur preparation et leur utilisation comme fongicides et acaricides
FR2594437A1 (fr) 1986-02-19 1987-08-21 Rhone Poulenc Agrochimie Nouveaux derives du cyano-2 benzimidazole, leur preparation, les compositions les contenant et leur utilisation comme fongicide
US4859684A (en) 1986-09-15 1989-08-22 Janssen Pharmaceutica N.V. (1H-imidazol-1-ylmethyl) substituted benzimidazole derivatives and use thereof in treating androgen dependent disorders
DE4237617A1 (de) * 1992-11-06 1994-05-11 Bayer Ag Verwendung von substituierten Benzimidazolen
US5331003A (en) 1993-03-26 1994-07-19 Eli Lilly And Company Anticoccidial methods

Also Published As

Publication number Publication date
ATE256124T1 (de) 2003-12-15
HUP0201035A3 (en) 2006-03-28
CA2372664C (en) 2009-09-22
CA2372664A1 (en) 2000-11-16
KR20020008839A (ko) 2002-01-31
WO2000068225A1 (de) 2000-11-16
EP1177191B1 (de) 2003-12-10
HK1046143B (zh) 2004-10-21
ES2213024T3 (es) 2004-08-16
HUP0201035A2 (en) 2002-08-28
AU5392600A (en) 2000-11-21
US6569881B1 (en) 2003-05-27
AU761553B2 (en) 2003-06-05
JP2002544129A (ja) 2002-12-24
CN1130359C (zh) 2003-12-10
NZ515243A (en) 2004-09-24
DK1177191T3 (da) 2004-04-05
BR0010699A (pt) 2002-02-05
EP1177191A1 (de) 2002-02-06
DE50004731D1 (de) 2004-01-22
DE19920551A1 (de) 2000-11-09
HK1046143A1 (en) 2002-12-27
CN1349529A (zh) 2002-05-15
ZA200107985B (en) 2002-12-24

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