JPWO2022127869A5 - - Google Patents

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Publication number
JPWO2022127869A5
JPWO2022127869A5 JP2023576366A JP2023576366A JPWO2022127869A5 JP WO2022127869 A5 JPWO2022127869 A5 JP WO2022127869A5 JP 2023576366 A JP2023576366 A JP 2023576366A JP 2023576366 A JP2023576366 A JP 2023576366A JP WO2022127869 A5 JPWO2022127869 A5 JP WO2022127869A5
Authority
JP
Japan
Prior art keywords
alkyl
cycloalkyl
phenyl
heterocyclyl
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023576366A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024522210A5 (https=
JP2024522210A (ja
Publication date
Priority claimed from CN202011495497.0A external-priority patent/CN114644633B/zh
Application filed filed Critical
Publication of JP2024522210A publication Critical patent/JP2024522210A/ja
Publication of JP2024522210A5 publication Critical patent/JP2024522210A5/ja
Publication of JPWO2022127869A5 publication Critical patent/JPWO2022127869A5/ja
Pending legal-status Critical Current

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JP2023576366A 2020-12-18 2021-12-16 複素環系jak阻害剤 Pending JP2024522210A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN202011495497.0 2020-12-18
CN202011495497.0A CN114644633B (zh) 2020-12-18 2020-12-18 杂环类jak抑制剂
PCT/CN2021/138842 WO2022127869A1 (zh) 2020-12-18 2021-12-16 杂环类jak抑制剂

Publications (3)

Publication Number Publication Date
JP2024522210A JP2024522210A (ja) 2024-06-11
JP2024522210A5 JP2024522210A5 (https=) 2026-03-09
JPWO2022127869A5 true JPWO2022127869A5 (https=) 2026-03-09

Family

ID=81990162

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023576366A Pending JP2024522210A (ja) 2020-12-18 2021-12-16 複素環系jak阻害剤

Country Status (7)

Country Link
US (1) US20240246984A1 (https=)
EP (1) EP4310088A4 (https=)
JP (1) JP2024522210A (https=)
CN (1) CN114644633B (https=)
AU (1) AU2021398704A1 (https=)
CA (1) CA3222404A1 (https=)
WO (1) WO2022127869A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2024539280A (ja) 2021-10-25 2024-10-28 カイメラ セラピューティクス, インコーポレイテッド Tyk2分解剤およびそれらの使用

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20090306067A1 (en) * 2006-04-10 2009-12-10 Harald Engelhardt 2, 4-diaminopyrimidide derivates and their use for the treatment of cancer
EP2528918B1 (en) * 2010-01-29 2014-09-10 Nerviano Medical Sciences S.r.l. 6,7-dihydroimidazo[1,5-a]pyrazin-8(5h)-one derivatives as protein kinase modulators
WO2016061751A1 (en) * 2014-10-22 2016-04-28 Merck Sharp & Dohme Corp. Ethyl n-boc piperidinyl pyrazolo pyridones as janus kinase inhibitors
MX2020002869A (es) * 2017-09-15 2020-07-24 Aduro Biotech Inc Compuestos de pirazolopirimidinona y usos de los mismos.
WO2019074962A1 (en) * 2017-10-10 2019-04-18 Syros Pharmaceuticals, Inc. PYRROLOTRIAZINE COMPOUNDS AND METHODS FOR INHIBITING TAM KINASES
JP2022510980A (ja) * 2018-11-30 2022-01-28 江▲蘇▼豪森▲薬▼▲業▼集▲団▼有限公司 ヘテロ芳香族誘導体調節因子、その製造方法及び使用
JP7617030B2 (ja) * 2019-05-08 2025-01-17 ビマラン バイオサイエンシーズ,インク. Jak阻害剤

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