JPWO2022078352A5 - - Google Patents
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- JPWO2022078352A5 JPWO2022078352A5 JP2023523059A JP2023523059A JPWO2022078352A5 JP WO2022078352 A5 JPWO2022078352 A5 JP WO2022078352A5 JP 2023523059 A JP2023523059 A JP 2023523059A JP 2023523059 A JP2023523059 A JP 2023523059A JP WO2022078352 A5 JPWO2022078352 A5 JP WO2022078352A5
- Authority
- JP
- Japan
- Prior art keywords
- crystalline form
- disease
- ray powder
- powder diffraction
- peaks
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN2020120814 | 2020-10-14 | ||
| CNPCT/CN2020/120814 | 2020-10-14 | ||
| PCT/CN2021/123387 WO2022078352A1 (en) | 2020-10-14 | 2021-10-13 | Crystal forms of glp-1r agonists and uses thereof |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| JP2023546125A JP2023546125A (ja) | 2023-11-01 |
| JP2023546125A5 JP2023546125A5 (https=) | 2024-10-21 |
| JPWO2022078352A5 true JPWO2022078352A5 (https=) | 2024-10-21 |
| JP7769695B2 JP7769695B2 (ja) | 2025-11-13 |
Family
ID=78401981
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023523059A Active JP7769695B2 (ja) | 2020-10-14 | 2021-10-13 | Ｇｌｐ－１ｒアゴニストの結晶形態およびその使用 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US12516041B2 (https=) |
| EP (1) | EP4228753B1 (https=) |
| JP (1) | JP7769695B2 (https=) |
| CN (1) | CN116710446B (https=) |
| AU (1) | AU2021359493A1 (https=) |
| CA (1) | CA3195264A1 (https=) |
| ES (1) | ES3041328T3 (https=) |
| TW (1) | TWI912388B (https=) |
| WO (1) | WO2022078352A1 (https=) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20210069000A (ko) * | 2019-12-02 | 2021-06-10 | 현대약품 주식회사 | Glp-1 수용체 작용제 |
| KR20240068737A (ko) | 2021-09-27 | 2024-05-17 | 테른스 파마슈티칼스, 인크. | Glp-1r 효능제로서의 벤즈이미다졸 카복실산 |
| AU2022375634A1 (en) | 2021-10-25 | 2024-06-06 | Terns Pharmaceuticals, Inc. | Compounds as glp-1r agonists |
| KR20240150488A (ko) | 2022-02-23 | 2024-10-15 | 테른스 파마슈티칼스, 인크. | Glp-1r 작용제로서의 화합물 |
| CN117362282B (zh) * | 2022-07-07 | 2026-04-21 | 杭州德睿智药科技有限公司 | Glp-1r激动剂的盐及其制备方法和应用 |
| AU2023310481A1 (en) * | 2022-07-18 | 2025-03-06 | Mindrank Therapeutics (Suzhou) New Drug Research And Development Co., Ltd | Polymorphic form of glp-1r agonist, preparation method therefor and use thereof |
| US20240398794A1 (en) | 2023-04-07 | 2024-12-05 | Terns Pharmaceuticals, Inc. | COMBINATIONS OF GLP-1R AND THRß AGONISTS AND METHODS OF USE THEREOF |
| TW202521533A (zh) | 2023-09-14 | 2025-06-01 | 香港商歌禮製藥(中國)有限公司 | Glp-1r 激動劑及其治療方法 |
| US12291530B1 (en) | 2023-11-24 | 2025-05-06 | Ascletis Pharma (China) Co., Limited | GLP-1R agonist and therapeutic method thereof |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3773919A (en) | 1969-10-23 | 1973-11-20 | Du Pont | Polylactide-drug mixtures |
| US4485045A (en) | 1981-07-06 | 1984-11-27 | Research Corporation | Synthetic phosphatidyl cholines useful in forming liposomes |
| US4544545A (en) | 1983-06-20 | 1985-10-01 | Trustees University Of Massachusetts | Liposomes containing modified cholesterol for organ targeting |
| US5013556A (en) | 1989-10-20 | 1991-05-07 | Liposome Technology, Inc. | Liposomes with enhanced circulation time |
| US7727983B2 (en) | 2008-03-07 | 2010-06-01 | Transtech Pharma, Inc. | Oxadiazoanthracene compounds for the treatment of diabetes |
| AR083878A1 (es) * | 2010-11-15 | 2013-03-27 | Boehringer Ingelheim Int | Terapia antidiabetica vasoprotectora y cardioprotectora, linagliptina, metodo de tratamiento |
| EP3555064B9 (en) * | 2016-12-16 | 2023-03-01 | Pfizer Inc. | Glp-1 receptor agonists and uses thereof |
| ES2943510T3 (es) * | 2018-06-15 | 2023-06-13 | Pfizer | Agonistas del receptor GLP-1 y usos del mismo |
| CR20210341A (es) * | 2018-11-22 | 2021-11-25 | Qilu Regor Therapeutics Inc | Agonistas de glp-ir y usos de los mismos |
| US10954221B2 (en) * | 2019-04-12 | 2021-03-23 | Qilu Regor Therapeutics Inc. | GLP-1R agonists and uses thereof |
| AU2020256647B2 (en) * | 2019-04-12 | 2025-07-31 | Qilu Regor Therapeutics Inc. | GLP-1R agonists and uses thereof |
-
2021
- 2021-10-13 TW TW110138006A patent/TWI912388B/zh active
- 2021-10-13 CA CA3195264A patent/CA3195264A1/en active Pending
- 2021-10-13 WO PCT/CN2021/123387 patent/WO2022078352A1/en not_active Ceased
- 2021-10-13 CN CN202180082321.9A patent/CN116710446B/zh active Active
- 2021-10-13 ES ES21798552T patent/ES3041328T3/es active Active
- 2021-10-13 AU AU2021359493A patent/AU2021359493A1/en active Pending
- 2021-10-13 JP JP2023523059A patent/JP7769695B2/ja active Active
- 2021-10-13 EP EP21798552.2A patent/EP4228753B1/en active Active
- 2021-10-13 US US18/031,380 patent/US12516041B2/en active Active
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