JPWO2022059779A5 - - Google Patents

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Publication number
JPWO2022059779A5
JPWO2022059779A5 JP2022550631A JP2022550631A JPWO2022059779A5 JP WO2022059779 A5 JPWO2022059779 A5 JP WO2022059779A5 JP 2022550631 A JP2022550631 A JP 2022550631A JP 2022550631 A JP2022550631 A JP 2022550631A JP WO2022059779 A5 JPWO2022059779 A5 JP WO2022059779A5
Authority
JP
Japan
Prior art keywords
benzothiazol
dihydrofuro
optionally substituted
imidazol
imidazo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2022550631A
Other languages
English (en)
Japanese (ja)
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JP7706775B2 (ja
JPWO2022059779A1 (https=
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/JP2021/034327 external-priority patent/WO2022059779A1/ja
Publication of JPWO2022059779A1 publication Critical patent/JPWO2022059779A1/ja
Publication of JPWO2022059779A5 publication Critical patent/JPWO2022059779A5/ja
Priority to JP2025106969A priority Critical patent/JP2025134941A/ja
Application granted granted Critical
Publication of JP7706775B2 publication Critical patent/JP7706775B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2022550631A 2020-09-18 2021-09-17 アミン誘導体 Active JP7706775B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025106969A JP2025134941A (ja) 2020-09-18 2025-06-25 アミン誘導体

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP2020157398 2020-09-18
JP2020157398 2020-09-18
JP2021122893 2021-07-28
JP2021122893 2021-07-28
PCT/JP2021/034327 WO2022059779A1 (ja) 2020-09-18 2021-09-17 アミン誘導体

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025106969A Division JP2025134941A (ja) 2020-09-18 2025-06-25 アミン誘導体

Publications (3)

Publication Number Publication Date
JPWO2022059779A1 JPWO2022059779A1 (https=) 2022-03-24
JPWO2022059779A5 true JPWO2022059779A5 (https=) 2024-09-19
JP7706775B2 JP7706775B2 (ja) 2025-07-14

Family

ID=80776131

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2022550631A Active JP7706775B2 (ja) 2020-09-18 2021-09-17 アミン誘導体
JP2025106969A Pending JP2025134941A (ja) 2020-09-18 2025-06-25 アミン誘導体

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025106969A Pending JP2025134941A (ja) 2020-09-18 2025-06-25 アミン誘導体

Country Status (10)

Country Link
US (1) US20230365589A1 (https=)
EP (1) EP4215534A4 (https=)
JP (2) JP7706775B2 (https=)
KR (1) KR20230069162A (https=)
CN (1) CN116209441A (https=)
AU (1) AU2021343770A1 (https=)
BR (1) BR112023003807A2 (https=)
CA (1) CA3191617A1 (https=)
MX (1) MX2023003245A (https=)
WO (1) WO2022059779A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2023008470A1 (ja) * 2021-07-28 2023-02-02 住友ファーマ株式会社 縮環アミン誘導体
WO2025170029A1 (ja) * 2024-02-09 2025-08-14 カルナバイオサイエンス株式会社 ジヒドロキナゾリノン誘導体

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20020084116A (ko) * 2000-02-07 2002-11-04 애보트 게엠베하 운트 콤파니 카게 2-벤조티아졸릴 우레아 유도체 및 이의 단백질 키나제억제제로서의 용도
EP1679308B1 (en) 2003-10-15 2013-07-24 Ube Industries, Ltd. Novel indazole derivative
WO2008021338A2 (en) * 2006-08-15 2008-02-21 Wyeth Tricyclic oxazolidone derivatives useful as pr modulators
JP2010163361A (ja) 2007-04-27 2010-07-29 Dainippon Sumitomo Pharma Co Ltd キノリン誘導体
KR20100010894A (ko) 2008-07-23 2010-02-02 가부시키가이샤 키노파마 Dyrk를 저해하는 화합물을 함유하는 의약 조성물
US8470835B2 (en) 2009-01-13 2013-06-25 Glaxo Group Limited Pyrimidinecarboxamide derivatives as inhibitors of Syk kinase
TW201039825A (en) 2009-02-20 2010-11-16 Astrazeneca Ab Cyclopropyl amide derivatives 983
CN102712601A (zh) * 2009-11-12 2012-10-03 赛尔维他股份公司 化合物、其制备方法、药物组合物、化合物的用途、用于调节或调控丝氨酸/苏氨酸激酶的方法以及丝氨酸/苏氨酸激酶调节剂
CA2816219C (en) 2010-11-01 2019-10-29 Portola Pharmaceuticals, Inc. Nicotinamides as syk modulators
UY34200A (es) 2011-07-21 2013-02-28 Bayer Ip Gmbh 3-(fluorovinil)pirazoles y su uso
US9446044B2 (en) 2011-08-19 2016-09-20 Diaxonhit DYRK1 inhibitors and uses thereof
WO2013043002A1 (en) 2011-09-23 2013-03-28 Yuhan Corporation Imide-containing benzothiazole derivative or its salt and pharmaceutical composition comprising the same
KR101916443B1 (ko) 2012-07-26 2018-11-08 글락소 그룹 리미티드 Pad4 억제제로서의 2-(아자인돌-2-일) 벤즈이미다졸
RS63405B1 (sr) 2013-10-25 2022-08-31 Blueprint Medicines Corp Inhibitori receptora faktora rasta fibroblasta
JP2015107945A (ja) 2013-12-05 2015-06-11 国立大学法人京都大学 神経新生に関する化合物及び医薬組成物
GB201401886D0 (en) * 2014-02-04 2014-03-19 Lytix Biopharma As Neurodegenerative therapies
JP2017516850A (ja) 2014-05-23 2017-06-22 エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft Jak阻害剤である5−クロロ−2−ジフルオロメトキシフェニルピラゾロピリミジン化合物
WO2016044641A2 (en) 2014-09-17 2016-03-24 Epizyme, Inc. Carm1 inhibitors and uses thereof
GB201617339D0 (en) 2016-10-12 2016-11-23 Lytix Biopharma As Therapeutic compounds
CN109206537B (zh) 2018-10-10 2021-04-09 华熙生物科技股份有限公司 一种乙酰化透明质酸钠的制备方法及其应用
US20230138851A1 (en) * 2020-01-30 2023-05-04 Carna Biosciences, Inc. Novel alkyne derivatives

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