JPWO2021201036A5 - - Google Patents
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- JPWO2021201036A5 JPWO2021201036A5 JP2022512589A JP2022512589A JPWO2021201036A5 JP WO2021201036 A5 JPWO2021201036 A5 JP WO2021201036A5 JP 2022512589 A JP2022512589 A JP 2022512589A JP 2022512589 A JP2022512589 A JP 2022512589A JP WO2021201036 A5 JPWO2021201036 A5 JP WO2021201036A5
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- JP
- Japan
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- optionally substituted
- methyl
- group
- carbon atoms
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- Prior art date
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2020065410 | 2020-03-31 | ||
| JP2020065410 | 2020-03-31 | ||
| PCT/JP2021/013694 WO2021201036A1 (ja) | 2020-03-31 | 2021-03-30 | ヒドロキシピロリジン誘導体およびその医薬用途 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JPWO2021201036A1 JPWO2021201036A1 (https=) | 2021-10-07 |
| JPWO2021201036A5 true JPWO2021201036A5 (https=) | 2024-04-26 |
| JP7684282B2 JP7684282B2 (ja) | 2025-05-27 |
Family
ID=77927631
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022512589A Active JP7684282B2 (ja) | 2020-03-31 | 2021-03-30 | ヒドロキシピロリジン誘導体およびその医薬用途 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20230312542A1 (https=) |
| EP (1) | EP4129402A4 (https=) |
| JP (1) | JP7684282B2 (https=) |
| CN (1) | CN115298173A (https=) |
| WO (1) | WO2021201036A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20240327392A1 (en) * | 2021-06-25 | 2024-10-03 | Albius Sciences Alpha Private Limited | Heterocycloalkyl-substituted polyheteroazole derivatives as medicaments for treating and/or preventing rs virus infections |
| KR20240148807A (ko) * | 2022-03-22 | 2024-10-11 | 옵쉐스트바 스 아그라니첸너이아트볫스트벤너스찌유 "빅-즈다로비예쥐보트니흐" | 메데토미딘 및 그 유도체의 제조 방법 |
| CN119677735A (zh) * | 2022-05-11 | 2025-03-21 | 基因泰克公司 | 作为vhl配体的苯并噻唑化合物 |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2425288A1 (en) | 2000-10-11 | 2002-05-02 | Sander G. Mills | Pyrrolidine modulators of ccr5 chemokine receptor activity |
| AU2006223482A1 (en) | 2005-03-14 | 2006-09-21 | Janssen Pharmaceutica, N.V. | Process for the preparation of opioid modulators |
| EP2238128B1 (en) | 2007-12-26 | 2012-08-22 | Sanofi | Heterocyclic pyrazole-carboxamides as p2y12 antagonists |
| PL2242759T3 (pl) | 2008-02-06 | 2013-06-28 | Astrazeneca Ab | Związki |
| EP2384328B1 (en) | 2008-11-27 | 2013-02-13 | Boehringer Ingelheim International GmbH | 6,7,8,9-tetrahydro-5h-1,4,7,10a-tetraaza-cyclohept[f]indene derivatives, pharmaceutical compositions containing these compounds, their use and process for preparing them |
| US8673954B2 (en) * | 2009-02-27 | 2014-03-18 | Enanta Pharmaceuticals, Inc. | Benzimidazole derivatives |
| EA020031B1 (ru) * | 2009-06-11 | 2014-08-29 | Эббви Бахамаз Лтд. | Противовирусные соединения |
| AU2010274001A1 (en) * | 2009-07-16 | 2012-02-23 | Vertex Pharmaceuticals Incorporated | Benzimidazole analogues for the treatment or prevention of Flavivirus infections |
| EP2305660A1 (en) | 2009-09-25 | 2011-04-06 | Almirall, S.A. | New thiadiazole derivatives |
| WO2011084402A1 (en) | 2009-12-21 | 2011-07-14 | Merck Sharp & Dohme Corp. | Tyrosine kinase inhibitors |
| EP2752410B1 (en) | 2011-10-25 | 2016-08-31 | Shionogi & Co., Ltd. | Heterocycle derivative having pgd2 receptor antagonist activity |
| KR102668696B1 (ko) * | 2012-01-12 | 2024-05-29 | 예일 유니버시티 | E3 유비퀴틴 리가아제에 의한 표적 단백질 및 다른 폴리펩티드의 증진된 분해를 위한 화합물 및 방법 |
| US9783527B2 (en) | 2014-09-16 | 2017-10-10 | Abbvie Inc. | Indazole ureas and method of use |
| WO2019084026A1 (en) * | 2017-10-24 | 2019-05-02 | Genentech, Inc. | (4-HYDROXYPYRROLIDIN-2-YL) -HETEROCYCLIC COMPOUNDS AND METHODS OF USE |
| IL281188B2 (en) * | 2018-09-07 | 2025-08-01 | Arvinas Operations Inc | Polycyclic compounds and methods for the targeted degradation of rapidly accelerated fibrosarcoma polypeptides |
-
2021
- 2021-03-30 JP JP2022512589A patent/JP7684282B2/ja active Active
- 2021-03-30 CN CN202180026438.5A patent/CN115298173A/zh active Pending
- 2021-03-30 US US17/915,794 patent/US20230312542A1/en active Pending
- 2021-03-30 WO PCT/JP2021/013694 patent/WO2021201036A1/ja not_active Ceased
- 2021-03-30 EP EP21778705.0A patent/EP4129402A4/en not_active Withdrawn
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