JPWO2021160602A5 - - Google Patents

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Publication number
JPWO2021160602A5
JPWO2021160602A5 JP2022548400A JP2022548400A JPWO2021160602A5 JP WO2021160602 A5 JPWO2021160602 A5 JP WO2021160602A5 JP 2022548400 A JP2022548400 A JP 2022548400A JP 2022548400 A JP2022548400 A JP 2022548400A JP WO2021160602 A5 JPWO2021160602 A5 JP WO2021160602A5
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JP
Japan
Prior art keywords
invention described
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022548400A
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English (en)
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JP2023512729A (ja
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2021/053062 external-priority patent/WO2021160602A1/en
Publication of JP2023512729A publication Critical patent/JP2023512729A/ja
Publication of JPWO2021160602A5 publication Critical patent/JPWO2021160602A5/ja
Pending legal-status Critical Current

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Claims (1)

  1. 明細書に記載の発明。

JP2022548400A 2020-02-10 2021-02-09 モノアシルグリセロールリパーゼ調節因子 Pending JP2023512729A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202062972484P 2020-02-10 2020-02-10
US62/972,484 2020-02-10
PCT/EP2021/053062 WO2021160602A1 (en) 2020-02-10 2021-02-09 Monoacylglycerol lipase modulators

Publications (2)

Publication Number Publication Date
JP2023512729A JP2023512729A (ja) 2023-03-28
JPWO2021160602A5 true JPWO2021160602A5 (ja) 2024-02-20

Family

ID=74595268

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022548400A Pending JP2023512729A (ja) 2020-02-10 2021-02-09 モノアシルグリセロールリパーゼ調節因子

Country Status (21)

Country Link
US (2) US11708359B2 (ja)
EP (1) EP4103557A1 (ja)
JP (1) JP2023512729A (ja)
KR (1) KR20220140581A (ja)
CN (1) CN115066422A (ja)
AR (1) AR121296A1 (ja)
AU (1) AU2021220539A1 (ja)
BR (1) BR112022015116A2 (ja)
CA (1) CA3169988A1 (ja)
CL (1) CL2022002136A1 (ja)
CO (1) CO2022011275A2 (ja)
CR (1) CR20220376A (ja)
DO (1) DOP2022000162A (ja)
EC (1) ECSP22062460A (ja)
IL (1) IL295447A (ja)
JO (1) JOP20220180A1 (ja)
MX (1) MX2022009804A (ja)
PE (1) PE20221576A1 (ja)
TW (1) TW202140465A (ja)
UY (1) UY39066A (ja)
WO (1) WO2021160602A1 (ja)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20220140581A (ko) 2020-02-10 2022-10-18 얀센 파마슈티카 엔.브이. 모노아실글리세롤 리파아제 조절제
WO2021191384A1 (en) 2020-03-26 2021-09-30 Janssen Pharmaceutica Nv Aryl piperidines as monoacylglycerol lipase modulators
CA3176113A1 (en) 2020-03-26 2021-09-30 Janssen Pharmaceutica Nv Aminocyclobutanes as monoacylglycerol lipase modulators
BR112022019211A2 (pt) 2020-03-26 2023-03-07 Janssen Pharmaceutica Nv Azaspirociclos como moduladores de lipase de monoacilglicerol
KR20240046538A (ko) 2021-08-09 2024-04-09 얀센 파마슈티카 엔브이 자폐증 스펙트럼 장애에 사용하기 위한 모노아실글리세롤 리파제 조절제

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA05000945A (es) 2002-07-25 2005-05-16 Pharmacia Italia Spa Biciclo-pirazoles activos como inhibidores de la cinasa, procedimientos para su preparacion y composiciones farmaceuticas que los contienen.
EP2090576A1 (en) 2008-02-01 2009-08-19 Merz Pharma GmbH & Co.KGaA 6-halo-pyrazolo[1,5-a]pyridines, a process for their preparation and their use as metabotropic glutamate receptor (mGluR) modulators
EP2760450A1 (en) * 2011-09-30 2014-08-06 Janssen Pharmaceutica, N.V. Monoacylglycerol lipase inhibitors for the treatment of metabolic diseases and related disorders
US10610520B2 (en) 2016-03-31 2020-04-07 Takeda Pharmaceutical Company Limited Heterocyclic compound
JP6788683B2 (ja) 2016-03-31 2020-11-25 武田薬品工業株式会社 複素環化合物
JP7189143B2 (ja) * 2017-09-29 2022-12-13 武田薬品工業株式会社 複素環化合物
CN112272670B (zh) 2019-04-16 2023-12-12 上海翰森生物医药科技有限公司 含二并环类衍生物抑制剂、其制备方法和应用
KR20220140581A (ko) 2020-02-10 2022-10-18 얀센 파마슈티카 엔.브이. 모노아실글리세롤 리파아제 조절제
WO2021191384A1 (en) 2020-03-26 2021-09-30 Janssen Pharmaceutica Nv Aryl piperidines as monoacylglycerol lipase modulators
CA3176113A1 (en) 2020-03-26 2021-09-30 Janssen Pharmaceutica Nv Aminocyclobutanes as monoacylglycerol lipase modulators
BR112022019211A2 (pt) 2020-03-26 2023-03-07 Janssen Pharmaceutica Nv Azaspirociclos como moduladores de lipase de monoacilglicerol

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