JPWO2021160602A5 - - Google Patents
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- JPWO2021160602A5 JPWO2021160602A5 JP2022548400A JP2022548400A JPWO2021160602A5 JP WO2021160602 A5 JPWO2021160602 A5 JP WO2021160602A5 JP 2022548400 A JP2022548400 A JP 2022548400A JP 2022548400 A JP2022548400 A JP 2022548400A JP WO2021160602 A5 JPWO2021160602 A5 JP WO2021160602A5
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- JP
- Japan
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- invention described
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202062972484P | 2020-02-10 | 2020-02-10 | |
| US62/972,484 | 2020-02-10 | ||
| PCT/EP2021/053062 WO2021160602A1 (en) | 2020-02-10 | 2021-02-09 | Monoacylglycerol lipase modulators |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023512729A JP2023512729A (ja) | 2023-03-28 |
| JPWO2021160602A5 true JPWO2021160602A5 (enExample) | 2024-02-20 |
| JP7795466B2 JP7795466B2 (ja) | 2026-01-07 |
Family
ID=74595268
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022548400A Active JP7795466B2 (ja) | 2020-02-10 | 2021-02-09 | モノアシルグリセロールリパーゼ調節因子 |
Country Status (22)
| Country | Link |
|---|---|
| US (2) | US11708359B2 (enExample) |
| EP (1) | EP4103557B1 (enExample) |
| JP (1) | JP7795466B2 (enExample) |
| KR (1) | KR20220140581A (enExample) |
| CN (1) | CN115066422B (enExample) |
| AR (1) | AR121296A1 (enExample) |
| AU (1) | AU2021220539A1 (enExample) |
| BR (1) | BR112022015116A2 (enExample) |
| CA (1) | CA3169988A1 (enExample) |
| CL (1) | CL2022002136A1 (enExample) |
| CO (1) | CO2022011275A2 (enExample) |
| CR (1) | CR20220376A (enExample) |
| DO (1) | DOP2022000162A (enExample) |
| EC (1) | ECSP22062460A (enExample) |
| IL (1) | IL295447A (enExample) |
| JO (1) | JOP20220180A1 (enExample) |
| MX (1) | MX2022009804A (enExample) |
| PE (1) | PE20221576A1 (enExample) |
| PH (1) | PH12022552019A1 (enExample) |
| TW (1) | TW202140465A (enExample) |
| UY (1) | UY39066A (enExample) |
| WO (1) | WO2021160602A1 (enExample) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20220140581A (ko) | 2020-02-10 | 2022-10-18 | 얀센 파마슈티카 엔.브이. | 모노아실글리세롤 리파아제 조절제 |
| BR112022019178A2 (pt) | 2020-03-26 | 2022-11-01 | Janssen Pharmaceutica Nv | Aminociclobutanos como moduladores da monoacilglicerol lipase |
| BR112022019211A2 (pt) * | 2020-03-26 | 2023-03-07 | Janssen Pharmaceutica Nv | Azaspirociclos como moduladores de lipase de monoacilglicerol |
| JP7729832B2 (ja) | 2020-03-26 | 2025-08-26 | ヤンセン ファーマシューティカ エヌ.ベー. | モノアシルグリセロールリパーゼ調節因子としてのアリールピペリジン |
| US12115154B2 (en) | 2020-12-16 | 2024-10-15 | Srx Cardio, Llc | Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9) |
| JP2024532740A (ja) | 2021-08-09 | 2024-09-10 | ヤンセン ファーマシューティカ エヌ.ベー. | 自閉症スペクトラム障害に使用するためのモノアシルグリセロールリパーゼ調節因子 |
| CA3242372A1 (en) | 2021-12-29 | 2023-07-06 | Psy Therapeutics, Inc. | Inhibiting monoacylglycerol lipase (magl) |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2003244649A1 (en) | 2002-07-25 | 2004-02-23 | Pharmacia Italia Spa | Bicyclo-pyrazoles active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them |
| EP2090576A1 (en) | 2008-02-01 | 2009-08-19 | Merz Pharma GmbH & Co.KGaA | 6-halo-pyrazolo[1,5-a]pyridines, a process for their preparation and their use as metabotropic glutamate receptor (mGluR) modulators |
| EP2760450A1 (en) | 2011-09-30 | 2014-08-06 | Janssen Pharmaceutica, N.V. | Monoacylglycerol lipase inhibitors for the treatment of metabolic diseases and related disorders |
| JP6832342B2 (ja) | 2016-03-31 | 2021-02-24 | 武田薬品工業株式会社 | 複素環化合物 |
| EA036637B1 (ru) | 2016-03-31 | 2020-12-02 | Такеда Фармасьютикал Компани Лимитед | Гетероциклические спиросоединения, ингибирующие моноацилглицерин-липазу |
| GB201613163D0 (en) | 2016-07-29 | 2016-09-14 | Autifony Therapeutics Ltd | Novel compounds |
| EP3689879B1 (en) | 2017-09-29 | 2025-02-12 | Takeda Pharmaceutical Company Limited | Heterocyclic compound |
| WO2020211798A1 (zh) | 2019-04-16 | 2020-10-22 | 上海翰森生物医药科技有限公司 | 含二并环类衍生物抑制剂、其制备方法和应用 |
| KR20220140581A (ko) * | 2020-02-10 | 2022-10-18 | 얀센 파마슈티카 엔.브이. | 모노아실글리세롤 리파아제 조절제 |
| BR112022019178A2 (pt) | 2020-03-26 | 2022-11-01 | Janssen Pharmaceutica Nv | Aminociclobutanos como moduladores da monoacilglicerol lipase |
| BR112022019211A2 (pt) | 2020-03-26 | 2023-03-07 | Janssen Pharmaceutica Nv | Azaspirociclos como moduladores de lipase de monoacilglicerol |
| JP7729832B2 (ja) | 2020-03-26 | 2025-08-26 | ヤンセン ファーマシューティカ エヌ.ベー. | モノアシルグリセロールリパーゼ調節因子としてのアリールピペリジン |
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2021
- 2021-02-09 KR KR1020227031216A patent/KR20220140581A/ko not_active Withdrawn
- 2021-02-09 PH PH1/2022/552019A patent/PH12022552019A1/en unknown
- 2021-02-09 US US17/171,559 patent/US11708359B2/en active Active
- 2021-02-09 CN CN202180013762.3A patent/CN115066422B/zh active Active
- 2021-02-09 PE PE2022001698A patent/PE20221576A1/es unknown
- 2021-02-09 IL IL295447A patent/IL295447A/en unknown
- 2021-02-09 EP EP21705124.2A patent/EP4103557B1/en active Active
- 2021-02-09 CA CA3169988A patent/CA3169988A1/en active Pending
- 2021-02-09 MX MX2022009804A patent/MX2022009804A/es unknown
- 2021-02-09 CR CR20220376A patent/CR20220376A/es unknown
- 2021-02-09 JP JP2022548400A patent/JP7795466B2/ja active Active
- 2021-02-09 AR ARP210100333A patent/AR121296A1/es not_active Application Discontinuation
- 2021-02-09 WO PCT/EP2021/053062 patent/WO2021160602A1/en not_active Ceased
- 2021-02-09 UY UY0001039066A patent/UY39066A/es unknown
- 2021-02-09 AU AU2021220539A patent/AU2021220539A1/en active Pending
- 2021-02-09 BR BR112022015116A patent/BR112022015116A2/pt unknown
- 2021-02-09 JO JOP/2022/0180A patent/JOP20220180A1/ar unknown
- 2021-02-09 TW TW110104960A patent/TW202140465A/zh unknown
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2022
- 2022-08-08 CL CL2022002136A patent/CL2022002136A1/es unknown
- 2022-08-09 EC ECSENADI202262460A patent/ECSP22062460A/es unknown
- 2022-08-10 DO DO2022000162A patent/DOP2022000162A/es unknown
- 2022-08-10 CO CONC2022/0011275A patent/CO2022011275A2/es unknown
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2023
- 2023-06-02 US US18/328,242 patent/US20230382902A1/en not_active Abandoned