JPWO2020263187A5 - - Google Patents
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- Publication number
- JPWO2020263187A5 JPWO2020263187A5 JP2021577361A JP2021577361A JPWO2020263187A5 JP WO2020263187 A5 JPWO2020263187 A5 JP WO2020263187A5 JP 2021577361 A JP2021577361 A JP 2021577361A JP 2021577361 A JP2021577361 A JP 2021577361A JP WO2020263187 A5 JPWO2020263187 A5 JP WO2020263187A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- substituted
- independently
- groups
- group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SG10201905890P | 2019-06-25 | ||
SG10201905890P | 2019-06-25 | ||
PCT/SG2020/050363 WO2020263187A1 (en) | 2019-06-25 | 2020-06-25 | Compounds for treatment of eye disorders |
Publications (2)
Publication Number | Publication Date |
---|---|
JP2022542645A JP2022542645A (ja) | 2022-10-06 |
JPWO2020263187A5 true JPWO2020263187A5 (es) | 2023-05-24 |
Family
ID=74062096
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2021577346A Pending JP2022543343A (ja) | 2019-06-25 | 2020-06-25 | がんの治療のための化合物 |
JP2021577361A Pending JP2022542645A (ja) | 2019-06-25 | 2020-06-25 | 眼障害の治療のための化合物 |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2021577346A Pending JP2022543343A (ja) | 2019-06-25 | 2020-06-25 | がんの治療のための化合物 |
Country Status (11)
Country | Link |
---|---|
US (2) | US20220242863A1 (es) |
EP (2) | EP3990458A1 (es) |
JP (2) | JP2022543343A (es) |
KR (1) | KR20220054286A (es) |
CN (2) | CN114450285B (es) |
AU (2) | AU2020301057A1 (es) |
BR (1) | BR112021026366A2 (es) |
CA (2) | CA3144226A1 (es) |
IL (2) | IL289221A (es) |
MX (2) | MX2022000099A (es) |
WO (2) | WO2020263187A1 (es) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN113354576B (zh) * | 2021-06-28 | 2022-08-12 | 黑龙江立科新材料有限公司 | 邻位烷氧基取代的吡啶类化合物的制备方法 |
Family Cites Families (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7078423B2 (en) * | 2002-07-18 | 2006-07-18 | Inotek Pharmaceuticals Corporation | 5-Aryltetrazole compounds, compositions thereof, and uses therefor |
EP1773826A4 (en) * | 2004-07-02 | 2009-06-03 | Exelixis Inc | MODULATORS OF C-MET AND THEIR METHOD OF USE |
DOP2006000051A (es) * | 2005-02-24 | 2006-08-31 | Lilly Co Eli | Inhibidores de vegf-r2 y métodos |
GB0507575D0 (en) * | 2005-04-14 | 2005-05-18 | Novartis Ag | Organic compounds |
KR100787131B1 (ko) * | 2006-07-04 | 2007-12-21 | 한국생명공학연구원 | Hif―1 활성을 저해하는 화합물, 이의 제조방법 및이를 유효성분으로 함유하는 약학적 조성물 |
CN101558068A (zh) * | 2006-10-16 | 2009-10-14 | 诺瓦提斯公司 | 用作蛋白激酶抑制剂的苯乙酰胺类 |
WO2008112695A2 (en) * | 2007-03-12 | 2008-09-18 | Irm Llc | Pyrazolo [3,4-d] pyrimidines and 1, 2, 5, 6-tetraaza- as- indacenes as protein kinase inhibitors for cancer treatment |
EP2903645A2 (en) * | 2012-10-05 | 2015-08-12 | Kadmon Corporation, LLC | Treatment of ocular disorders |
GB2508652A (en) * | 2012-12-07 | 2014-06-11 | Agency Science Tech & Res | Heterocyclic piperazine derivatives |
WO2015031613A1 (en) * | 2013-08-30 | 2015-03-05 | Ambit Biosciences Corporation | Biaryl acetamide compounds and methods of use thereof |
WO2015043492A1 (en) * | 2013-09-26 | 2015-04-02 | Sunshine Lake Pharma Co., Ltd. | Substituted urea derivatives and uses thereof in medicine |
CN105294680A (zh) * | 2014-06-25 | 2016-02-03 | 中国药科大学 | Vegfr-2不可逆抑制剂及其用途 |
WO2016004254A1 (en) * | 2014-07-01 | 2016-01-07 | The Regents Of The University Of California | Combined modulation of ire1 |
CN104876912B (zh) * | 2015-04-08 | 2017-07-21 | 苏州云轩医药科技有限公司 | Wnt信号通路抑制剂及其应用 |
KR102128018B1 (ko) * | 2017-05-12 | 2020-06-30 | 한국화학연구원 | 피라졸로 피리미딘 유도체, 이의 제조방법 및 이를 유효성분으로 함유하는 암, 자가면역질환 및 뇌질환의 예방 또는 치료용 약학적 조성물 |
SG11202005278PA (en) * | 2017-12-29 | 2020-07-29 | Agency Science Tech & Res | Compounds for treating eye diseases and methods thereof |
-
2020
- 2020-06-25 WO PCT/SG2020/050363 patent/WO2020263187A1/en unknown
- 2020-06-25 AU AU2020301057A patent/AU2020301057A1/en active Pending
- 2020-06-25 AU AU2020307293A patent/AU2020307293A1/en not_active Abandoned
- 2020-06-25 CN CN202080053620.5A patent/CN114450285B/zh active Active
- 2020-06-25 CA CA3144226A patent/CA3144226A1/en not_active Abandoned
- 2020-06-25 CN CN202080053621.XA patent/CN114466847A/zh active Pending
- 2020-06-25 MX MX2022000099A patent/MX2022000099A/es unknown
- 2020-06-25 KR KR1020227002304A patent/KR20220054286A/ko unknown
- 2020-06-25 BR BR112021026366A patent/BR112021026366A2/pt not_active Application Discontinuation
- 2020-06-25 US US17/596,976 patent/US20220242863A1/en active Pending
- 2020-06-25 WO PCT/SG2020/050362 patent/WO2020263186A1/en unknown
- 2020-06-25 JP JP2021577346A patent/JP2022543343A/ja active Pending
- 2020-06-25 MX MX2022000103A patent/MX2022000103A/es unknown
- 2020-06-25 US US17/596,988 patent/US20220315587A1/en active Pending
- 2020-06-25 CA CA3144228A patent/CA3144228A1/en not_active Abandoned
- 2020-06-25 EP EP20831505.1A patent/EP3990458A1/en active Pending
- 2020-06-25 JP JP2021577361A patent/JP2022542645A/ja active Pending
- 2020-06-25 EP EP20830624.1A patent/EP3990457A4/en active Pending
-
2021
- 2021-12-21 IL IL289221A patent/IL289221A/en unknown
- 2021-12-21 IL IL289201A patent/IL289201A/en unknown
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