JPWO2020262603A5 - - Google Patents
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- Publication number
- JPWO2020262603A5 JPWO2020262603A5 JP2021527768A JP2021527768A JPWO2020262603A5 JP WO2020262603 A5 JPWO2020262603 A5 JP WO2020262603A5 JP 2021527768 A JP2021527768 A JP 2021527768A JP 2021527768 A JP2021527768 A JP 2021527768A JP WO2020262603 A5 JPWO2020262603 A5 JP WO2020262603A5
- Authority
- JP
- Japan
- Prior art keywords
- amino
- group
- phenyl
- trifluoromethyl
- cyclopropanecarboxylic acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2019122077 | 2019-06-28 | ||
| JP2019122077 | 2019-06-28 | ||
| PCT/JP2020/025187 WO2020262603A1 (ja) | 2019-06-28 | 2020-06-26 | Ｅｐ２アンタゴニスト |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JPWO2020262603A1 JPWO2020262603A1 (https=) | 2020-12-30 |
| JPWO2020262603A5 true JPWO2020262603A5 (https=) | 2023-06-27 |
| JP7647552B2 JP7647552B2 (ja) | 2025-03-18 |
Family
ID=74060242
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021527768A Active JP7647552B2 (ja) | 2019-06-28 | 2020-06-26 | Ｅｐ２アンタゴニスト |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20220388955A1 (https=) |
| EP (1) | EP3992176B1 (https=) |
| JP (1) | JP7647552B2 (https=) |
| KR (1) | KR20220030219A (https=) |
| CN (1) | CN114026068A (https=) |
| AU (1) | AU2020306387A1 (https=) |
| BR (1) | BR112021026397A2 (https=) |
| CA (1) | CA3144201A1 (https=) |
| ES (1) | ES3048491T3 (https=) |
| IL (1) | IL289252A (https=) |
| MX (1) | MX2021015654A (https=) |
| PH (1) | PH12021553155A1 (https=) |
| TW (1) | TW202114985A (https=) |
| WO (1) | WO2020262603A1 (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2024016314A (ja) * | 2020-12-24 | 2024-02-07 | 小野薬品工業株式会社 | 一般式（ｉ－ａ）で示される化合物、その薬学的に許容される塩、またはそれらの水和物と免疫チェックポイント阻害薬および／またはｅｐ４受容体拮抗薬との組み合わせ |
| TW202241846A (zh) * | 2020-12-24 | 2022-11-01 | 日商小野藥品工業股份有限公司 | 具有ｅｐ拮抗活性之化合物的鹽、溶劑合物及結晶 |
| JP2024016311A (ja) * | 2020-12-24 | 2024-02-07 | 小野薬品工業株式会社 | Ｅｐ２アンタゴニスト |
| EP4359399A4 (en) | 2021-06-24 | 2025-04-23 | Reservoir Neuroscience, Inc. | EP2 antagonist compounds |
| JP7205657B1 (ja) | 2021-08-10 | 2023-01-17 | 小野薬品工業株式会社 | Ｅｐ４アンタゴニストの製造方法 |
| CN115417772B (zh) * | 2022-09-26 | 2024-07-19 | 无锡双启科技有限公司 | 一种3-硝基-4-氟苯甲醚的制备方法 |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4618702A (en) | 1985-01-24 | 1986-10-21 | E. I. Du Pont De Nemours And Company | Manufacture of butanedicarboxylic acid esters |
| EP0218728A1 (en) | 1985-04-03 | 1987-04-22 | Yamanouchi Pharmaceutical Co. Ltd. | Phenylene derivatives |
| IL140930A0 (en) * | 1998-08-07 | 2002-02-10 | Emisphere Tech Inc | Compounds and compositions for delivering active agents |
| ES2298168T3 (es) * | 1999-12-16 | 2008-05-16 | Emisphere Technologies, Inc. | Compuestos y composiciones para suministrar agentes activos. |
| US7601712B2 (en) * | 2003-09-17 | 2009-10-13 | Ono Pharmaceutical Co., Ltd. | Carboxylic acid compounds and medicinal compositions containing the same as the active ingredient |
| RU2006125441A (ru) * | 2003-12-15 | 2008-01-27 | Джапан Тобакко Инк. (Jp) | Производные циклопропана и их фармацевтическое применение |
| WO2005080367A1 (en) * | 2004-02-12 | 2005-09-01 | Pharmagene Laboratories Limited | Ep2 receptor agonists |
| JP5017103B2 (ja) | 2004-06-17 | 2012-09-05 | トランスフオーム・フアーマシユーチカルズ・インコーポレーテツド | 薬剤共結晶組成物および関連した使用方法 |
| WO2007052843A1 (ja) | 2005-11-04 | 2007-05-10 | Takeda Pharmaceutical Company Limited | 複素環アミド化合物およびその用途 |
| KR20070052843A (ko) | 2005-11-18 | 2007-05-23 | 로열 플래닛 캄퍼니 리미티드 | 가상현실 쇼핑 시스템 |
| JP2008152097A (ja) | 2006-12-19 | 2008-07-03 | Nikon Corp | 連続撮影制御方法および撮像装置 |
| EP2003118A1 (de) | 2007-06-13 | 2008-12-17 | Bayer Schering Pharma Aktiengesellschaft | Zimtsäurederivate als Modulatoren des EP2-Rezeptors |
| TWI410410B (zh) * | 2007-08-10 | 2013-10-01 | Ono Pharmaceutical Co | Phenylacetic acid compounds |
| JP2012177618A (ja) | 2011-02-25 | 2012-09-13 | Nsk Ltd | レゾルバ装置 |
| EP2721011B1 (en) | 2011-06-20 | 2017-09-06 | Emory University | Prostaglandin receptor ep2 antagonists, derivatives, compositions, and uses related thereto |
| CA2867527A1 (en) * | 2012-05-03 | 2013-11-07 | Takeda Gmbh | Novel ep2 receptor agonists |
-
2020
- 2020-06-24 TW TW109121578A patent/TW202114985A/zh unknown
- 2020-06-26 EP EP20832376.6A patent/EP3992176B1/en active Active
- 2020-06-26 CN CN202080047042.4A patent/CN114026068A/zh active Pending
- 2020-06-26 WO PCT/JP2020/025187 patent/WO2020262603A1/ja not_active Ceased
- 2020-06-26 CA CA3144201A patent/CA3144201A1/en active Pending
- 2020-06-26 PH PH1/2021/553155A patent/PH12021553155A1/en unknown
- 2020-06-26 BR BR112021026397A patent/BR112021026397A2/pt not_active Application Discontinuation
- 2020-06-26 KR KR1020217042562A patent/KR20220030219A/ko not_active Withdrawn
- 2020-06-26 AU AU2020306387A patent/AU2020306387A1/en not_active Abandoned
- 2020-06-26 JP JP2021527768A patent/JP7647552B2/ja active Active
- 2020-06-26 MX MX2021015654A patent/MX2021015654A/es unknown
- 2020-06-26 ES ES20832376T patent/ES3048491T3/es active Active
- 2020-06-26 US US17/621,137 patent/US20220388955A1/en active Pending
-
2021
- 2021-12-22 IL IL289252A patent/IL289252A/en unknown
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