JPS643166A - Production of thiol - Google Patents
Production of thiolInfo
- Publication number
- JPS643166A JPS643166A JP15750187A JP15750187A JPS643166A JP S643166 A JPS643166 A JP S643166A JP 15750187 A JP15750187 A JP 15750187A JP 15750187 A JP15750187 A JP 15750187A JP S643166 A JPS643166 A JP S643166A
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- formula
- compound
- reaction
- useful
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
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- Furan Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
PURPOSE: To obtain a thiol which is useful as an intermediate of medicines advantageously through a substantially one-step process without isolation of the intermediate by allowing hydrochloric acid to react with a reaction product from 2,2-disubstituted-thiazolidine and a nitroethene derivative.
CONSTITUTION: The reaction between a compound of formula I (R1 is 1W4C alkyl; R2 is 1W4C alkyl, acetate) and another compound of formula II (R3 is 1W4C alkyl; P is eliminable group) in a solvent, preferably water and/or lower alcohol, is followed by action of hydrochloric acid on the reaction mixture to give a subject compound of formula IV, which is useful as an intermediate of a compound of formula III (R1, R2 are H, 1W4C alkyl; R3, alk are 1W4C alkyl) which is used as a medicine. Thus, the reaction process, operations are much improved, installation costs are saved, and the yield of the product exceeds 80%. The compound of formula I is readily prepared from an sulfate ester of 2-aminoalcohol and has high stability.
COPYRIGHT: (C)1989,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP62-157501A JPH013166A (en) | 1987-06-26 | Method for producing thiols |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP62-157501A JPH013166A (en) | 1987-06-26 | Method for producing thiols |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS643166A true JPS643166A (en) | 1989-01-06 |
JPH013166A JPH013166A (en) | 1989-01-06 |
Family
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