JPS6334152B2 - - Google Patents

Info

Publication number
JPS6334152B2
JPS6334152B2 JP60043555A JP4355585A JPS6334152B2 JP S6334152 B2 JPS6334152 B2 JP S6334152B2 JP 60043555 A JP60043555 A JP 60043555A JP 4355585 A JP4355585 A JP 4355585A JP S6334152 B2 JPS6334152 B2 JP S6334152B2
Authority
JP
Japan
Prior art keywords
fluoro
piperazinyl
pyrimidinyl
formula
fluorophenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP60043555A
Other languages
English (en)
Japanese (ja)
Other versions
JPS6175A (ja
Inventor
Pii Ieuitsuchi Josefu
Jii Robetsuku Junia Uorutaa
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Co
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of JPS6175A publication Critical patent/JPS6175A/ja
Publication of JPS6334152B2 publication Critical patent/JPS6334152B2/ja
Granted legal-status Critical Current

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP60043555A 1984-03-06 1985-03-05 神経弛緩剤、１‐フルオロフェニルブチル‐４‐（５‐ハロ‐２‐ピリミジニル）ピペラジン誘導体 Granted JPS6175A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US58658084A 1984-03-06 1984-03-06
US586580 1984-03-06
US683309 1984-12-18

Publications (2)

Publication Number Publication Date
JPS6175A JPS6175A (ja) 1986-01-06
JPS6334152B2 true JPS6334152B2 (cs) 1988-07-08

Family

ID=24346326

Family Applications (1)

Application Number Title Priority Date Filing Date
JP60043555A Granted JPS6175A (ja) 1984-03-06 1985-03-05 神経弛緩剤、１‐フルオロフェニルブチル‐４‐（５‐ハロ‐２‐ピリミジニル）ピペラジン誘導体

Country Status (1)

Country Link
JP (1) JPS6175A (cs)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE8701375D0 (sv) * 1987-04-02 1987-04-02 Leo Ab Novel pyridyl- and pyrimidyl derivatives
HU206109B (en) * 1987-10-26 1992-08-28 Pfizer Process for producing heterocyclic carbonylpropyl pyrimidinyl piperazine derivatives and pharmaceutical compositions comprising same
GB9721780D0 (en) * 1997-10-14 1997-12-10 Glaxo Group Ltd Process for the synthesis of chloropurine intermediates
CN101679400B (zh) * 2007-05-14 2013-04-17 爱思开生物制药株式会社 氨基甲酰氧基芳基链烷芳基哌嗪化合物，含该化合物的药物组合物以及通过给予该化合物治疗疼痛、焦虑和抑郁的方法
JP2015514135A (ja) * 2012-04-14 2015-05-18 イントラ−セルラー・セラピーズ・インコーポレイテッドＩｎｔｒａ−Ｃｅｌｌｕｌａｒ Ｔｈｅｒａｐｉｅｓ， Ｉｎｃ． 新規組成物および方法

Also Published As

Publication number Publication date
JPS6175A (ja) 1986-01-06

Similar Documents

Publication Publication Date Title
US4605655A (en) Antipsychotic 1-fluorophenylbutyl-4-(2-pyrimidinyl)piperazine derivatives
JP3880842B2 (ja) １−〔（４−クロロフェニル）フェニルメチル〕ピペラジンの鏡像体およびその製造法
US6498168B2 (en) Muscarinic antagonists
KR870001045B1 (ko) 2-[4-[(4,4-디알킬-2,6-피페리딘디온-1-일)부틸]피페라지닐] 피리미딘류의 제조방법
JPS6084282A (ja) １−ヘテロアリ−ル−４−〔（２．５−ピロリジンジオン−１−イル）アルキル〕ピペラジン誘導体
JP2000505795A (ja) 置換シクロアザンから誘導された新規芳香族ピペラジン、それらの調製法、医薬組成物、および薬剤としての使用
CZ362092A3 (en) Piperazinyl cyclohexanol and piperidinyl cyclohexanol derivative, process of its preparation and a pharmaceutical preparation containing thereof
HU227973B1 (hu) Indazolamidok és az ezeket tartalmazó gyógyszerek
HU185157B (en) Process for the preparation of 8-arylalkyl-3-phenyl-3-nortropanols and acid addition salts thereof
JPH0567637B2 (cs)
Yevich et al. Synthesis and biological characterization of. alpha.-(4-fluorophenyl)-4-(5-fluoro-2-pyrimidinyl)-1-piperazinebutanol and analogs as potential atypical antipsychotic agents
DE68910451T2 (de) 1,4-benzoxazin- und 1,4-benzothiazin-derivate und verfahren zu deren herstellung.
JPS6334152B2 (cs)
HU195509B (en) Process for producing pyridinyl-piperazine derivatives and pharmaceutical compositions containing them as active agents
CA1177830A (en) Hexahydro-trans- and tetrahydropyridoindole neuroleptic agents
JPWO2003002532A1 (ja) 縮合環式基を有する環状ジアミン化合物
FR2744451A1 (fr) Nouvelles imidazolidinones, pyrimidinones, et 1,3-diazepin-2 -ones, leur preparation et leurs applications en therapeutique
Balle et al. Synthesis and structure–affinity relationship investigations of 5-aminomethyl and 5-carbamoyl analogues of the antipsychotic sertindole. A new class of selective α1 adrenoceptor antagonists
JP2021104931A (ja) 含窒素複素環を有するジベンゾアゼピン誘導体
WO2005073183A1 (ja) アリールスルフィド誘導体
MXPA06013520A (es) Tetrahironaftilpiperazinas como antagonistas, agonistas inversos y agonistas parciales de 5-ht1b.
JP2571903B2 (ja) 新規アミノアルキルクロモン、その製造方法及びそれを含む薬学的組成物
JPS5838277A (ja) スピロチアゾリジニルピペラジン誘導体
CA2324268A1 (en) Aromaheterocyclic derivatives
HUP9903913A2 (hu) Szelektív dopamin D4 receptor ligandum troponil-piperazinok, eljárás előállításukra, azokat tartalmazó gyógyszerkészítmények és alkalmazásuk

Legal Events

Date Code Title Description
R250 Receipt of annual fees

Free format text: JAPANESE INTERMEDIATE CODE: R250

EXPY Cancellation because of completion of term