JPS6219438B2 - - Google Patents

Info

Publication number
JPS6219438B2
JPS6219438B2 JP57065232A JP6523282A JPS6219438B2 JP S6219438 B2 JPS6219438 B2 JP S6219438B2 JP 57065232 A JP57065232 A JP 57065232A JP 6523282 A JP6523282 A JP 6523282A JP S6219438 B2 JPS6219438 B2 JP S6219438B2
Authority
JP
Japan
Prior art keywords
deoxy
hydrogen
acetyl
ethyl acetate
mixture
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP57065232A
Other languages
English (en)
Japanese (ja)
Other versions
JPS57181096A (en
Inventor
Adamu Nageru Aasaa
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
PFIZER
Original Assignee
PFIZER
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by PFIZER filed Critical PFIZER
Publication of JPS57181096A publication Critical patent/JPS57181096A/ja
Publication of JPS6219438B2 publication Critical patent/JPS6219438B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40—Esters thereof
    • C07F9/4003—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/4006—Esters of acyclic acids which can have further substituents on alkyl

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
JP57065232A 1981-04-20 1982-04-19 4''-deoxy-4''-methylene oleandomycin and derivatives Granted JPS57181096A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/255,620 US4336368A (en) 1981-04-20 1981-04-20 4 Deoxy-4-methylene oleandomycin and derivatives thereof

Publications (2)

Publication Number Publication Date
JPS57181096A JPS57181096A (en) 1982-11-08
JPS6219438B2 true JPS6219438B2 (https=) 1987-04-28

Family

ID=22969153

Family Applications (1)

Application Number Title Priority Date Filing Date
JP57065232A Granted JPS57181096A (en) 1981-04-20 1982-04-19 4''-deoxy-4''-methylene oleandomycin and derivatives

Country Status (8)

Country Link
US (1) US4336368A (https=)
EP (1) EP0063489B1 (https=)
JP (1) JPS57181096A (https=)
AT (1) ATE8147T1 (https=)
DE (1) DE3260297D1 (https=)
DK (1) DK152133C (https=)
GR (1) GR76472B (https=)
IE (1) IE52912B1 (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4429116A (en) * 1982-12-27 1984-01-31 Pfizer Inc. Alkylated oleandomycin containing compounds
US4640910A (en) * 1985-11-12 1987-02-03 Abbott Laboratories Erythromycin A silylated compounds and method of use
DE3782994T2 (de) * 1986-09-18 1993-04-08 Taisho Pharma Co Ltd Erythromycin-a-derivate und verfahren zu ihrer herstellung.
SI9010556B (sl) * 1990-03-21 1998-10-31 Pliva Oleandomicin oksimi in postopek za njihovo pripravo
US5872229A (en) 1995-11-21 1999-02-16 Abbott Laboratories Process for 6-O-alkylation of erythromycin derivatives
US5929219A (en) 1997-09-10 1999-07-27 Abbott Laboratories 9-hydrazone and 9-azine erythromycin derivatives and a process of making the same
US6732014B2 (en) 2001-02-27 2004-05-04 Crane Co. System for accomplishing product detection
US8548625B2 (en) 2001-08-23 2013-10-01 Crane Merchandising Systems, Inc. Optical vend sensing system for product delivery detection

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4085119A (en) * 1977-02-04 1978-04-18 Pfizer Inc. 4-Substituted amino derivatives of oleandomycin
US4090017A (en) * 1977-02-04 1978-05-16 Pfizer Inc. 4-Deoxy-4-substituted amino derivatives of oleandomycin
US4124755A (en) * 1978-01-03 1978-11-07 Pfizer Inc. 11-Alkanoyl-4"-deoxy-4"-isonitrilo-oleandomycin derivatives
US4166901A (en) * 1978-01-03 1979-09-04 Pfizer Inc. 4"-Deoxy-4"-arylglyoxamido- and aroylthioformamido derivatives of oleandomycin and its esters

Also Published As

Publication number Publication date
DE3260297D1 (en) 1984-08-02
DK173182A (da) 1982-10-21
JPS57181096A (en) 1982-11-08
EP0063489B1 (en) 1984-06-27
DK152133C (da) 1988-07-11
DK152133B (da) 1988-02-01
IE52912B1 (en) 1988-04-13
EP0063489A1 (en) 1982-10-27
GR76472B (https=) 1984-08-10
US4336368A (en) 1982-06-22
ATE8147T1 (de) 1984-07-15
IE820916L (en) 1982-10-20

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