JPS62185068A - 置換ピロリジン―２―オン化合物、その製造方法及びそれを含む向知性薬 - Google Patents
置換ピロリジン―２―オン化合物、その製造方法及びそれを含む向知性薬Info
- Publication number
- JPS62185068A JPS62185068A JP62018790A JP1879087A JPS62185068A JP S62185068 A JPS62185068 A JP S62185068A JP 62018790 A JP62018790 A JP 62018790A JP 1879087 A JP1879087 A JP 1879087A JP S62185068 A JPS62185068 A JP S62185068A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- oxo
- unsubstituted
- group
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/24—Oxygen or sulfur atoms
- C07D207/26—2-Pyrrolidones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyrrole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Steroid Compounds (AREA)
- Solid-Sorbent Or Filter-Aiding Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH346/86-6 | 1986-01-30 | ||
| CH34686 | 1986-01-30 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS62185068A true JPS62185068A (ja) | 1987-08-13 |
| JPH0558631B2 JPH0558631B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1993-08-27 |
Family
ID=4184917
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP62018790A Granted JPS62185068A (ja) | 1986-01-30 | 1987-01-30 | 置換ピロリジン―２―オン化合物、その製造方法及びそれを含む向知性薬 |
Country Status (21)
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2002051836A1 (fr) * | 2000-12-27 | 2002-07-04 | Kyowa Hakko Kogyo Co., Ltd. | Inhibiteur de dipeptidyl peptidase iv |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FI95572C (fi) * | 1987-06-22 | 1996-02-26 | Eisai Co Ltd | Menetelmä lääkeaineena käyttökelpoisen piperidiinijohdannaisten tai sen farmaseuttisen suolan valmistamiseksi |
| EP4101561A1 (de) | 2021-06-08 | 2022-12-14 | Meusburger Georg GmbH & Co. KG | Zentriereinrichtung für ein formwerkzeug mit gleichzeitig tragenden wälzkörpereinheiten |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5488264A (en) * | 1977-12-23 | 1979-07-13 | Troponwerke Gmbh & Co Kg | 22oxoo11pyrrolidine acetic acid derivatives* their manufacture and use |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1039113A (en) * | 1964-08-06 | 1966-08-17 | Ucb Sa | New n-substituted lactams |
| US4144246A (en) * | 1976-11-15 | 1979-03-13 | Parke, Davis & Company | Pyrrolidineacetic acid esters |
| BE864269A (fr) * | 1977-03-03 | 1978-06-16 | Parke Davis & Co | Nouveaux n-(aminoalkyl substitue)-2-oxo-1-pyrrolidine-acetamides et procedes pour les produire |
| DE3361609D1 (en) * | 1982-03-24 | 1986-02-06 | Prodes Sa | New n-((2-oxo-1-pyrrolidinyl)acetyl)piperazines, the methods of producing such new compounds and their salts as well as pharmaceutical preparations for therapeutic use containing these compounds or salts |
-
1987
- 1987-01-21 PH PH34749A patent/PH23078A/en unknown
- 1987-01-26 EP EP87810045A patent/EP0236263B1/de not_active Expired - Lifetime
- 1987-01-26 DE DE8787810045T patent/DE3783247D1/de not_active Expired - Fee Related
- 1987-01-26 ES ES87810045T patent/ES2053578T3/es not_active Expired - Lifetime
- 1987-01-26 AT AT87810045T patent/ATE84033T1/de not_active IP Right Cessation
- 1987-01-26 FI FI870329A patent/FI870329A7/fi not_active IP Right Cessation
- 1987-01-27 IL IL81394A patent/IL81394A/xx not_active IP Right Cessation
- 1987-01-28 DD DD87299511A patent/DD260066A5/de unknown
- 1987-01-28 CA CA000528330A patent/CA1312081C/en not_active Expired - Lifetime
- 1987-01-28 PT PT84204A patent/PT84204B/pt not_active IP Right Cessation
- 1987-01-29 HU HU87277A patent/HU202862B/hu not_active IP Right Cessation
- 1987-01-29 NZ NZ219101A patent/NZ219101A/xx unknown
- 1987-01-29 IE IE23087A patent/IE61100B1/en not_active IP Right Cessation
- 1987-01-29 ZA ZA87650A patent/ZA87650B/xx unknown
- 1987-01-29 DK DK047187A patent/DK47187A/da not_active Application Discontinuation
- 1987-01-29 AU AU68097/87A patent/AU599951B2/en not_active Ceased
- 1987-01-29 NO NO870374A patent/NO870374L/no unknown
- 1987-01-30 JP JP62018790A patent/JPS62185068A/ja active Granted
- 1987-01-30 KR KR870000728A patent/KR870007159A/ko not_active Ceased
-
1989
- 1989-06-19 US US07/370,093 patent/US4945092A/en not_active Expired - Fee Related
-
1993
- 1993-03-19 GR GR920402948T patent/GR3007411T3/el unknown
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5488264A (en) * | 1977-12-23 | 1979-07-13 | Troponwerke Gmbh & Co Kg | 22oxoo11pyrrolidine acetic acid derivatives* their manufacture and use |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2002051836A1 (fr) * | 2000-12-27 | 2002-07-04 | Kyowa Hakko Kogyo Co., Ltd. | Inhibiteur de dipeptidyl peptidase iv |
Also Published As
| Publication number | Publication date |
|---|---|
| HU202862B (en) | 1991-04-29 |
| FI870329A0 (fi) | 1987-01-26 |
| PH23078A (en) | 1989-04-10 |
| AU6809787A (en) | 1987-08-06 |
| ATE84033T1 (de) | 1993-01-15 |
| EP0236263A2 (de) | 1987-09-09 |
| HUT43058A (en) | 1987-09-28 |
| ZA87650B (en) | 1987-09-30 |
| NO870374D0 (no) | 1987-01-29 |
| NZ219101A (en) | 1990-03-27 |
| ES2053578T3 (es) | 1994-08-01 |
| NO870374L (no) | 1987-07-31 |
| CA1312081C (en) | 1992-12-29 |
| DK47187D0 (da) | 1987-01-29 |
| PT84204A (en) | 1987-02-01 |
| PT84204B (pt) | 1989-09-14 |
| DD260066A5 (de) | 1988-09-14 |
| US4945092A (en) | 1990-07-31 |
| DE3783247D1 (de) | 1993-02-11 |
| KR870007159A (ko) | 1987-08-17 |
| EP0236263B1 (de) | 1992-12-30 |
| DK47187A (da) | 1987-07-31 |
| FI870329A7 (fi) | 1987-07-31 |
| JPH0558631B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1993-08-27 |
| IL81394A (en) | 1991-08-16 |
| AU599951B2 (en) | 1990-08-02 |
| EP0236263A3 (en) | 1989-04-19 |
| IE61100B1 (en) | 1994-10-05 |
| IL81394A0 (en) | 1987-08-31 |
| GR3007411T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1993-07-30 |
| IE870230L (en) | 1987-07-30 |
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