JPS62132852A - チアムフエニコ−ル（１）の製法 - Google Patents

チアムフエニコ−ル（１）の製法

Info

Publication number
JPS62132852A
JPS62132852A JP61287879A JP28787986A JPS62132852A JP S62132852 A JPS62132852 A JP S62132852A JP 61287879 A JP61287879 A JP 61287879A JP 28787986 A JP28787986 A JP 28787986A JP S62132852 A JPS62132852 A JP S62132852A
Authority
JP
Japan
Prior art keywords
threo
aminodiol
hcl
tables
thiamphenicol
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP61287879A
Other languages
English (en)
Japanese (ja)
Inventor
ヘルムート・デイツク
ヴオルフ−デイートリツヒ・グラーデル
マチアス・ヴエーバー
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Roche Diagnostics GmbH
Original Assignee
Boehringer Mannheim GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=6287716&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JPS62132852(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Mannheim GmbH filed Critical Boehringer Mannheim GmbH
Publication of JPS62132852A publication Critical patent/JPS62132852A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C315/00—Preparation of sulfones; Preparation of sulfoxides
    • C07C315/04—Preparation of sulfones; Preparation of sulfoxides by reactions not involving the formation of sulfone or sulfoxide groups
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP61287879A 1985-12-05 1986-12-04 チアムフエニコ−ル（１）の製法 Pending JPS62132852A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3543021.4 1985-12-05
DE19853543021 DE3543021A1 (de) 1985-12-05 1985-12-05 Verbesserte verfahren zur herstellung von d-threo-1-(p-methylsulfonylphenyl) -2-dichloracetamido-propandiol-1,3-(thiamphenicol) sowie verwendung geeigneter zwischenprodukte

Publications (1)

Publication Number Publication Date
JPS62132852A true JPS62132852A (ja) 1987-06-16

Family

ID=6287716

Family Applications (1)

Application Number Title Priority Date Filing Date
JP61287879A Pending JPS62132852A (ja) 1985-12-05 1986-12-04 チアムフエニコ−ル（１）の製法

Country Status (6)

Country Link
US (1) US4945181A (enExample)
EP (1) EP0224902B1 (enExample)
JP (1) JPS62132852A (enExample)
AT (1) ATE42094T1 (enExample)
DE (2) DE3543021A1 (enExample)
ES (1) ES2008668B3 (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4796258B2 (ja) * 2000-04-11 2011-10-19 ザンボン グループ エス．ピー．エー． クラミジア・ニューモニエ感染症の治療に有用な医薬組成物を製造するためのチアムフェニコール及びその誘導体の使用

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH02771A (ja) * 1988-01-08 1990-01-05 Nippon Zeon Co Ltd チアンフェニコールの製造法
US5346828A (en) * 1991-03-27 1994-09-13 Celgene Corporation Stereoisomeric enrichment of 2-amino-3-hydroxy-3-phenylpropionic acids using d-threonine aldolase
EP1785414A1 (en) * 2005-11-09 2007-05-16 KRKA, tovarna zdravil, d.d., Novo mesto Process for the synthesis of intermediates of chloramphenicol or its analogues

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA526865A (en) * 1956-06-26 A. Gregory Walter Substituted sulfonylphenyl-amido-1,3-propanediols and process for preparing them
GB745900A (en) * 1951-10-01 1956-03-07 Sterling Drug Inc Acylaminodiols and method for preparing same
GB770277A (en) * 1952-08-23 1957-03-20 Parke Davis & Co Amino-propanediols and their derivatives
US2791595A (en) * 1953-01-14 1957-05-07 Parke Davis & Co Long chain esters of nitrophenylaminopropanediols and preparation thereof
US2742500A (en) * 1953-12-22 1956-04-17 Du Pont Resolution of phenylaminopropanediols and intermediates
US2726266A (en) * 1954-05-10 1955-12-06 Du Pont Antibacterial composition containing diastereoisomers of 1-(p-methylsul-fonylphenyl)-2-(alpha, alpha-dichlo-roacetamido)-1, 3-propanediol
CH589617A5 (enExample) * 1973-11-22 1977-07-15 Hoffmann La Roche
US4235892A (en) * 1979-02-05 1980-11-25 Schering Corporation, Patent Dept. 1-Aryl-2-acylamido-3-fluoro-1-propanols, methods for their use as antibacterial agents and compositions useful therefor
US4582918A (en) * 1984-09-19 1986-04-15 Schering Corporation Preparation of intermediates for (threo)-1-aryl-2-acylamido-3-fluoro-1-propanols

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4796258B2 (ja) * 2000-04-11 2011-10-19 ザンボン グループ エス．ピー．エー． クラミジア・ニューモニエ感染症の治療に有用な医薬組成物を製造するためのチアムフェニコール及びその誘導体の使用

Also Published As

Publication number Publication date
ATE42094T1 (de) 1989-04-15
DE3662786D1 (en) 1989-05-18
EP0224902B1 (de) 1989-04-12
US4945181A (en) 1990-07-31
EP0224902A1 (de) 1987-06-10
DE3543021A1 (de) 1987-06-11
DE3543021C2 (enExample) 1988-04-14
ES2008668B3 (es) 1989-08-01

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