JPS60209521A - メキタジン誘導体及び同誘導体からなる抗気管支痙攣剤 - Google Patents

メキタジン誘導体及び同誘導体からなる抗気管支痙攣剤

Info

Publication number
JPS60209521A
JPS60209521A JP60053210A JP5321085A JPS60209521A JP S60209521 A JPS60209521 A JP S60209521A JP 60053210 A JP60053210 A JP 60053210A JP 5321085 A JP5321085 A JP 5321085A JP S60209521 A JPS60209521 A JP S60209521A
Authority
JP
Japan
Prior art keywords
methyl
phenothiazine
compound
azoniabicyclo
octane
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP60053210A
Other languages
English (en)
Japanese (ja)
Other versions
JPH0548232B2 (enExample
Inventor
アレキサンドリオ　スビツシイ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Laboratorio Guidotti SpA
Original Assignee
Laboratorio Guidotti SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Laboratorio Guidotti SpA filed Critical Laboratorio Guidotti SpA
Publication of JPS60209521A publication Critical patent/JPS60209521A/ja
Publication of JPH0548232B2 publication Critical patent/JPH0548232B2/ja
Granted legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/007—Pulmonary tract; Aromatherapy
    • A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Otolaryngology (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP60053210A 1984-03-16 1985-03-16 メキタジン誘導体及び同誘導体からなる抗気管支痙攣剤 Granted JPS60209521A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT20082A/84 1984-03-16
IT20082/84A IT1173445B (it) 1984-03-16 1984-03-16 Agenti ad attivita' antibroncospastica e composizioni farmaceutiche che li contengono

Publications (2)

Publication Number Publication Date
JPS60209521A true JPS60209521A (ja) 1985-10-22
JPH0548232B2 JPH0548232B2 (enExample) 1993-07-20

Family

ID=11163657

Family Applications (1)

Application Number Title Priority Date Filing Date
JP60053210A Granted JPS60209521A (ja) 1984-03-16 1985-03-16 メキタジン誘導体及び同誘導体からなる抗気管支痙攣剤

Country Status (6)

Country Link
US (1) US4603132A (enExample)
EP (1) EP0159059B1 (enExample)
JP (1) JPS60209521A (enExample)
DE (1) DE3509460A1 (enExample)
ES (1) ES8603441A1 (enExample)
IT (1) IT1173445B (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI933167A7 (fi) * 1991-01-10 1993-07-09 Pfizer N-alkyylikinuklidiniumsuolat aineen P antagonisteina
IT1251161B (it) * 1991-08-07 1995-05-04 Derivati ammonio quaternari di (-) e (+)-3-(10 h-fenotiazin-10-ilmetil)-l-azabiciclo (2.2.2.)ottano e composizioni farmaceutiche che li contengono
DK1567164T3 (da) 2002-11-26 2009-05-18 Alexza Pharmaceuticals Inc Anvendelse af loxapin til fremstilling af et lægemiddel til behandling af smerte
EP1565184A1 (en) * 2002-11-26 2005-08-24 Alexza Molecular Delivery Corporation Treatment of headache with antipsychotics delivered by inhalation
FR2910814B1 (fr) * 2006-12-28 2011-06-17 Pf Medicament Utilisation du 10-°(r3)-1-azabicyclo°2.2.2!oct-3-ylmethyl!-10h- phenothiazine pour la preparation d'un medicament exercant une inhibition selective des recepteurs muscariniques m1,2,3

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3987042A (en) * 1969-03-03 1976-10-19 Claude Gueremy Phenothiazine derivative
GB1250534A (enExample) * 1969-03-03 1971-10-20

Also Published As

Publication number Publication date
IT8420082A1 (it) 1985-09-16
IT1173445B (it) 1987-06-24
ES541321A0 (es) 1985-12-16
ES8603441A1 (es) 1985-12-16
EP0159059B1 (en) 1988-12-14
EP0159059A1 (en) 1985-10-23
IT8420082A0 (it) 1984-03-16
JPH0548232B2 (enExample) 1993-07-20
DE3509460C2 (enExample) 1992-06-25
DE3509460A1 (de) 1985-09-19
US4603132A (en) 1986-07-29

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