JPS60105651A - 2−ヒドロキシ−5−〔1−ヒドロキシ−2−(4−フエニル−2−ブチル)アミノエチル〕ベンズアミドの製造法 - Google Patents

2−ヒドロキシ−5−〔1−ヒドロキシ−2−(4−フエニル−2−ブチル)アミノエチル〕ベンズアミドの製造法

Info

Publication number
JPS60105651A
JPS60105651A JP59202903A JP20290384A JPS60105651A JP S60105651 A JPS60105651 A JP S60105651A JP 59202903 A JP59202903 A JP 59202903A JP 20290384 A JP20290384 A JP 20290384A JP S60105651 A JPS60105651 A JP S60105651A
Authority
JP
Japan
Prior art keywords
hydroxy
benzamide
phenyl
active ingredient
hydrochloride
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP59202903A
Other languages
English (en)
Japanese (ja)
Inventor
アンジエロ マライ
ギウセツペ セリ
マリオ パイニ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SHIYARUPAA SpA PAA IND PHARM
Original Assignee
SHIYARUPAA SpA PAA IND PHARM
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SHIYARUPAA SpA PAA IND PHARM filed Critical SHIYARUPAA SpA PAA IND PHARM
Publication of JPS60105651A publication Critical patent/JPS60105651A/ja
Pending legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/60Salicylic acid; Derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C1/00Preparation of hydrocarbons from one or more compounds, none of them being a hydrocarbon
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00Preparation of carboxylic acid amides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00Preparation of carboxylic acid amides
    • C07C231/12Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/28Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton
    • C07C237/30Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton having the nitrogen atom of the carboxamide group bound to hydrogen atoms or to acyclic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00Preparation of carboxylic acid esters

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP59202903A 1983-09-27 1984-09-27 2−ヒドロキシ−5−〔1−ヒドロキシ−2−(4−フエニル−2−ブチル)アミノエチル〕ベンズアミドの製造法 Pending JPS60105651A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT23005A/83 1983-09-27
IT23005/83A IT1194406B (it) 1983-09-27 1983-09-27 Procedimento per la preparazione di 2-idrossi-5-01-idrossi-2-((4-fenil-2-butil)ammino) etil benzammide

Publications (1)

Publication Number Publication Date
JPS60105651A true JPS60105651A (ja) 1985-06-11

Family

ID=11202777

Family Applications (1)

Application Number Title Priority Date Filing Date
JP59202903A Pending JPS60105651A (ja) 1983-09-27 1984-09-27 2−ヒドロキシ−5−〔1−ヒドロキシ−2−(4−フエニル−2−ブチル)アミノエチル〕ベンズアミドの製造法

Country Status (7)

Country Link
JP (1) JPS60105651A (it)
BE (1) BE900663A (it)
CH (1) CH661923A5 (it)
DE (1) DE3435349A1 (it)
FR (1) FR2552427B1 (it)
GB (1) GB2149399B (it)
IT (1) IT1194406B (it)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2017098520A1 (en) * 2015-12-09 2017-06-15 prscDAVALURI RAMAMOHAN RAO Process for the preparation of labetalol hydrochloride
CN112225674B (zh) * 2020-10-28 2021-12-03 天津大学 盐酸拉贝洛尔晶型化合物及其制备方法和应用

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS4843341A (it) * 1971-10-02 1973-06-22

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1266058A (it) * 1969-07-08 1972-03-08
ZA794872B (en) * 1978-09-20 1980-11-26 Schering Corp A phenylalkylaminoethylsalicylamide,its preparation and pharmaceutical compositions containing it

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS4843341A (it) * 1971-10-02 1973-06-22

Also Published As

Publication number Publication date
DE3435349C2 (it) 1989-09-21
IT8323005A0 (it) 1983-09-27
FR2552427A1 (fr) 1985-03-29
FR2552427B1 (fr) 1988-03-25
BE900663A (fr) 1985-01-16
GB2149399B (en) 1987-05-13
GB8424100D0 (en) 1984-10-31
IT1194406B (it) 1988-09-22
DE3435349A1 (de) 1985-04-18
CH661923A5 (it) 1987-08-31
GB2149399A (en) 1985-06-12
IT8323005A1 (it) 1985-03-27

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