JPS5995300A - コントロ−ルされた粒度の２−シアノ−４，５−エポキシ−３−オキソ−ステロイド類およびそれらの組成物 - Google Patents
コントロ−ルされた粒度の２−シアノ−４，５−エポキシ−３−オキソ−ステロイド類およびそれらの組成物Info
- Publication number
- JPS5995300A JPS5995300A JP58202482A JP20248283A JPS5995300A JP S5995300 A JPS5995300 A JP S5995300A JP 58202482 A JP58202482 A JP 58202482A JP 20248283 A JP20248283 A JP 20248283A JP S5995300 A JPS5995300 A JP S5995300A
- Authority
- JP
- Japan
- Prior art keywords
- cyano
- granular
- epoxy
- trilostane
- particles
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/001—Oxiranes
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Epoxy Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB8231278 | 1982-11-02 | ||
| GB8231278 | 1982-11-02 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS5995300A true JPS5995300A (ja) | 1984-06-01 |
| JPH0443078B2 JPH0443078B2 (Direct) | 1992-07-15 |
Family
ID=10533991
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP58202482A Granted JPS5995300A (ja) | 1982-11-02 | 1983-10-28 | コントロ−ルされた粒度の２−シアノ−４，５−エポキシ−３−オキソ−ステロイド類およびそれらの組成物 |
Country Status (12)
| Country | Link |
|---|---|
| EP (1) | EP0108606B1 (Direct) |
| JP (1) | JPS5995300A (Direct) |
| AT (1) | ATE38236T1 (Direct) |
| DE (1) | DE3378318D1 (Direct) |
| DK (1) | DK499683A (Direct) |
| ES (1) | ES526874A0 (Direct) |
| FI (1) | FI834025A7 (Direct) |
| GB (1) | GB2130588B (Direct) |
| GR (1) | GR79688B (Direct) |
| IE (1) | IE56205B1 (Direct) |
| NO (1) | NO833976L (Direct) |
| PT (1) | PT77593B (Direct) |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2003520803A (ja) * | 2000-01-18 | 2003-07-08 | マーゲツツ，ジヨージ | ホルモンレセプターの調節 |
| JP2004529142A (ja) * | 2001-04-09 | 2004-09-24 | ステグラム・ファーマシューティカルズ・リミテッド | ヒトおよび動物におけるコルチゾールおよび他の副腎ホルモンの異常濃度に伴う臨床状態の処置としてのこれらのホルモン濃度の間歇的低下 |
| JP2006523665A (ja) * | 2003-04-16 | 2006-10-19 | マーゲッツ，ジョージ | アンギオテンシンｉｉ関連疾患の治療 |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8328929D0 (en) * | 1983-10-29 | 1983-11-30 | Sterwin Ag | Steroid compounds |
| US6458811B1 (en) | 1996-03-26 | 2002-10-01 | Eli Lilly And Company | Benzothiophenes formulations containing same and methods |
| EP2462959B1 (en) | 2005-07-12 | 2016-06-22 | Ampio Pharmaceuticals, Inc. | Methods and products for treatment of diseases |
| GB2627797A (en) * | 2023-03-02 | 2024-09-04 | Norbrook Lab Ltd | Trilostane formulation |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3296255A (en) * | 1963-11-29 | 1967-01-03 | Sterling Drug Inc | 2-cyano steroids |
| GB1123770A (en) * | 1966-11-15 | 1968-08-14 | Sterling Drug Inc | 2-cyano-3-oxo-steroids |
| FR2408345A1 (fr) * | 1976-11-30 | 1979-06-08 | Besins Jean Louis | Nouvelle composition a action anti-conceptionnelle |
| US4062954A (en) * | 1976-12-27 | 1977-12-13 | Sterling Drug Inc. | Process for using a steroid compound |
| US4160027A (en) * | 1977-12-20 | 1979-07-03 | Sterling Drug Inc. | Steroid cyanoketones and intermediates |
| GB8328929D0 (en) | 1983-10-29 | 1983-11-30 | Sterwin Ag | Steroid compounds |
-
1983
- 1983-10-28 JP JP58202482A patent/JPS5995300A/ja active Granted
- 1983-10-28 ES ES526874A patent/ES526874A0/es active Granted
- 1983-11-01 NO NO833976A patent/NO833976L/no unknown
- 1983-11-01 GB GB08329173A patent/GB2130588B/en not_active Expired
- 1983-11-01 DK DK499683A patent/DK499683A/da not_active Application Discontinuation
- 1983-11-02 FI FI834025A patent/FI834025A7/fi not_active Application Discontinuation
- 1983-11-02 IE IE2563/83A patent/IE56205B1/en not_active IP Right Cessation
- 1983-11-02 PT PT77593A patent/PT77593B/pt not_active IP Right Cessation
- 1983-11-02 AT AT83306665T patent/ATE38236T1/de not_active IP Right Cessation
- 1983-11-02 EP EP83306665A patent/EP0108606B1/en not_active Expired
- 1983-11-02 DE DE8383306665T patent/DE3378318D1/de not_active Expired
- 1983-11-02 GR GR72848A patent/GR79688B/el unknown
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2003520803A (ja) * | 2000-01-18 | 2003-07-08 | マーゲツツ，ジヨージ | ホルモンレセプターの調節 |
| JP2004529142A (ja) * | 2001-04-09 | 2004-09-24 | ステグラム・ファーマシューティカルズ・リミテッド | ヒトおよび動物におけるコルチゾールおよび他の副腎ホルモンの異常濃度に伴う臨床状態の処置としてのこれらのホルモン濃度の間歇的低下 |
| JP2006523665A (ja) * | 2003-04-16 | 2006-10-19 | マーゲッツ，ジョージ | アンギオテンシンｉｉ関連疾患の治療 |
Also Published As
| Publication number | Publication date |
|---|---|
| GB8329173D0 (en) | 1983-12-07 |
| FI834025L (fi) | 1984-05-03 |
| FI834025A0 (fi) | 1983-11-02 |
| NO833976L (no) | 1984-05-03 |
| ATE38236T1 (de) | 1988-11-15 |
| EP0108606A1 (en) | 1984-05-16 |
| GB2130588B (en) | 1986-08-13 |
| IE56205B1 (en) | 1991-05-22 |
| PT77593A (en) | 1983-12-01 |
| DE3378318D1 (en) | 1988-12-01 |
| EP0108606B1 (en) | 1988-10-26 |
| IE832563L (en) | 1984-05-02 |
| ES8504486A1 (es) | 1985-05-01 |
| GR79688B (Direct) | 1984-10-31 |
| DK499683A (da) | 1984-05-03 |
| DK499683D0 (da) | 1983-11-01 |
| FI834025A7 (fi) | 1984-05-03 |
| ES526874A0 (es) | 1985-05-01 |
| GB2130588A (en) | 1984-06-06 |
| JPH0443078B2 (Direct) | 1992-07-15 |
| PT77593B (en) | 1986-03-18 |
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