JPS5835190A - ペネム−３−カルボン酸誘導体 - Google Patents

ペネム−３−カルボン酸誘導体

Info

Publication number
JPS5835190A
JPS5835190A JP56133203A JP13320381A JPS5835190A JP S5835190 A JPS5835190 A JP S5835190A JP 56133203 A JP56133203 A JP 56133203A JP 13320381 A JP13320381 A JP 13320381A JP S5835190 A JPS5835190 A JP S5835190A
Authority
JP
Japan
Prior art keywords
group
hydroxyethyl
penem
hydrogen atom
carboxylic acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP56133203A
Other languages
English (en)
Japanese (ja)
Other versions
JPS6324515B2 (cs
Inventor
Isao Kawamoto
勲 川本
Tetsuo Miyadera
宮寺　哲男
Masao Sugimura
杉村　征夫
Teruo Tanaka
輝夫 田中
Toshihiko Hashimoto
俊彦 橋本
Kimio Iino
公夫 飯野
Shinichi Sugawara
真一 菅原
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sankyo Co Ltd
Original Assignee
Sankyo Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Co Ltd filed Critical Sankyo Co Ltd
Priority to JP56133203A priority Critical patent/JPS5835190A/ja
Priority to GB08224330A priority patent/GB2105329B/en
Priority to DE19823231596 priority patent/DE3231596A1/de
Priority to FR8214580A priority patent/FR2512027A1/fr
Priority to IT68039/82A priority patent/IT1156494B/it
Priority to CH5058/82A priority patent/CH654308A5/de
Publication of JPS5835190A publication Critical patent/JPS5835190A/ja
Publication of JPS6324515B2 publication Critical patent/JPS6324515B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP56133203A 1981-08-25 1981-08-25 ペネム−３−カルボン酸誘導体 Granted JPS5835190A (ja)

Priority Applications (6)

Application Number Priority Date Filing Date Title
JP56133203A JPS5835190A (ja) 1981-08-25 1981-08-25 ペネム−３−カルボン酸誘導体
GB08224330A GB2105329B (en) 1981-08-25 1982-08-25 Penem-3-carboxylic acid derivatives their preparation and their use as antimicrobial agents
DE19823231596 DE3231596A1 (de) 1981-08-25 1982-08-25 Penem-3-carbonsaeurederivate, verfahren zu deren herstellung und diese enthaltende pharmazeutische zusammensetzungen
FR8214580A FR2512027A1 (fr) 1981-08-25 1982-08-25 Derives d'acide peneme-3-carboxylique, leur preparation et leur utilisation comme agents antimicrobiens
IT68039/82A IT1156494B (it) 1981-08-25 1982-08-25 Derivati dell acido penem 3 carbossilico loro preparazione ed uso come agenti antimicrobici
CH5058/82A CH654308A5 (de) 1981-08-25 1982-08-25 Penem-3-carbonsaeurederivate und deren herstellung.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP56133203A JPS5835190A (ja) 1981-08-25 1981-08-25 ペネム−３−カルボン酸誘導体

Publications (2)

Publication Number Publication Date
JPS5835190A true JPS5835190A (ja) 1983-03-01
JPS6324515B2 JPS6324515B2 (cs) 1988-05-20

Family

ID=15099135

Family Applications (1)

Application Number Title Priority Date Filing Date
JP56133203A Granted JPS5835190A (ja) 1981-08-25 1981-08-25 ペネム−３−カルボン酸誘導体

Country Status (6)

Country Link
JP (1) JPS5835190A (cs)
CH (1) CH654308A5 (cs)
DE (1) DE3231596A1 (cs)
FR (1) FR2512027A1 (cs)
GB (1) GB2105329B (cs)
IT (1) IT1156494B (cs)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5921692A (ja) * 1982-07-29 1984-02-03 Sankyo Co Ltd 経口ペネム化合物及びその製法

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0110280B1 (en) * 1982-11-29 1994-10-12 Schering Corporation Process for the production of penem compounds
US4791198A (en) * 1984-07-05 1988-12-13 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha Beta-lactam compound and preparation thereof
US4861877A (en) * 1984-07-05 1989-08-29 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha Process for preparing 4-acetoxy-3-hydroxyethylazetidin-2-one derivatives
GB8915392D0 (en) * 1989-07-05 1989-08-23 Erba Carlo Spa Process for penems
US5416208A (en) * 1989-07-05 1995-05-16 Farmitalia Carlo Erba S R L Process for penems

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS53137951A (en) * 1977-05-09 1978-12-01 Ciba Geigy Ag Thiaaaza compound having betaalactum ring
JPS55153789A (en) * 1979-04-11 1980-11-29 Sankyo Co Ltd Penem-3-carboxylic acid derivative and its preparation
JPS572290A (en) * 1980-06-03 1982-01-07 Sankyo Co Ltd Production of penem-3-carboxylic derivative

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4168314A (en) * 1977-11-17 1979-09-18 Merck & Co., Inc. 6-(1'-Hydroxyethyl)-2-aminoethylthio-pen-2-em-3-carboxylic acid
EP0003960B1 (de) * 1978-02-02 1983-06-29 Ciba-Geigy Ag 6-Substituierte Thia-Azaverbindungen, ihre Herstellung und diese enthaltende pharmazeutische Präparate
CA1212105A (en) * 1980-04-30 1986-09-30 Shoji Ikeda Ampicillin esters and production thereof
US4411906A (en) * 1981-11-25 1983-10-25 Schering Corporation (5R,6S,8R)-6-(1-Hydroxyethyl)-2-(2-fluoroethylthio)-penem-3-carboxylates

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS53137951A (en) * 1977-05-09 1978-12-01 Ciba Geigy Ag Thiaaaza compound having betaalactum ring
JPS55153789A (en) * 1979-04-11 1980-11-29 Sankyo Co Ltd Penem-3-carboxylic acid derivative and its preparation
JPS572290A (en) * 1980-06-03 1982-01-07 Sankyo Co Ltd Production of penem-3-carboxylic derivative

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5921692A (ja) * 1982-07-29 1984-02-03 Sankyo Co Ltd 経口ペネム化合物及びその製法

Also Published As

Publication number Publication date
DE3231596A1 (de) 1983-03-10
FR2512027B1 (cs) 1984-12-14
GB2105329B (en) 1985-05-30
IT8268039A0 (it) 1982-08-25
IT1156494B (it) 1987-02-04
CH654308A5 (de) 1986-02-14
DE3231596C2 (cs) 1989-03-09
FR2512027A1 (fr) 1983-03-04
GB2105329A (en) 1983-03-23
JPS6324515B2 (cs) 1988-05-20

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