JPS58201763A - インド−ルアセトキシ酢酸エステル - Google Patents
インド−ルアセトキシ酢酸エステルInfo
- Publication number
- JPS58201763A JPS58201763A JP8286182A JP8286182A JPS58201763A JP S58201763 A JPS58201763 A JP S58201763A JP 8286182 A JP8286182 A JP 8286182A JP 8286182 A JP8286182 A JP 8286182A JP S58201763 A JPS58201763 A JP S58201763A
- Authority
- JP
- Japan
- Prior art keywords
- acid ester
- indoleacetoxyacetic
- formula
- indolacetoxyacetic
- acetate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP8286182A JPS58201763A (ja) | 1982-05-17 | 1982-05-17 | インド−ルアセトキシ酢酸エステル |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP8286182A JPS58201763A (ja) | 1982-05-17 | 1982-05-17 | インド−ルアセトキシ酢酸エステル |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS58201763A true JPS58201763A (ja) | 1983-11-24 |
| JPH0212221B2 JPH0212221B2 (enrdf_load_stackoverflow) | 1990-03-19 |
Family
ID=13786116
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP8286182A Granted JPS58201763A (ja) | 1982-05-17 | 1982-05-17 | インド−ルアセトキシ酢酸エステル |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JPS58201763A (enrdf_load_stackoverflow) |
Cited By (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6207700B1 (en) | 1999-01-07 | 2001-03-27 | Vanderbilt University | Amide derivatives for antiangiogenic and/or antitumorigenic use |
| US6306890B1 (en) | 1999-08-30 | 2001-10-23 | Vanderbilt University | Esters derived from indolealkanols and novel amides derived from indolealkylamides that are selective COX-2 inhibitors |
| US6762182B1 (en) | 1999-01-07 | 2004-07-13 | Vanderbilt University | Converting cox inhibition compounds that are not COX-2 selective inhibitors to derivatives that are COX-2 selective inhibitors |
| US7736624B2 (en) | 2006-06-19 | 2010-06-15 | Univ Vanderbilt | Methods and compositions for diagnostic and therapeutic targeting of COX-2 |
| US8168656B2 (en) | 2004-04-26 | 2012-05-01 | Vanderbilt University | Indoleacetic acid and indenacetic acid derivatives as therapeutic agents with reduced gastrointestinal toxicity |
| US9346803B2 (en) | 2011-10-17 | 2016-05-24 | Vanderbilt University | Indomethacin analogs for the treatment of castrate-resistant prostate cancer |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5147708A (ja) * | 1974-10-23 | 1976-04-23 | Hitachi Ltd | Denshanontenkairo |
| JPS58164570A (ja) * | 1982-02-26 | 1983-09-29 | トロポンベルケ・ゲゼルシヤフト・ミツト・ベシユレンクテル・ハフツング・ウント・カンパニ−・コマンジツト・ゲゼルシヤフト | アセメタシンの製造法 |
-
1982
- 1982-05-17 JP JP8286182A patent/JPS58201763A/ja active Granted
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5147708A (ja) * | 1974-10-23 | 1976-04-23 | Hitachi Ltd | Denshanontenkairo |
| JPS58164570A (ja) * | 1982-02-26 | 1983-09-29 | トロポンベルケ・ゲゼルシヤフト・ミツト・ベシユレンクテル・ハフツング・ウント・カンパニ−・コマンジツト・ゲゼルシヤフト | アセメタシンの製造法 |
Cited By (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6207700B1 (en) | 1999-01-07 | 2001-03-27 | Vanderbilt University | Amide derivatives for antiangiogenic and/or antitumorigenic use |
| US6399647B2 (en) | 1999-01-07 | 2002-06-04 | Vanderbilt University | Amide derivatives for antiangiogenic and/or antitumorigenic use |
| US6762182B1 (en) | 1999-01-07 | 2004-07-13 | Vanderbilt University | Converting cox inhibition compounds that are not COX-2 selective inhibitors to derivatives that are COX-2 selective inhibitors |
| US6306890B1 (en) | 1999-08-30 | 2001-10-23 | Vanderbilt University | Esters derived from indolealkanols and novel amides derived from indolealkylamides that are selective COX-2 inhibitors |
| US8168656B2 (en) | 2004-04-26 | 2012-05-01 | Vanderbilt University | Indoleacetic acid and indenacetic acid derivatives as therapeutic agents with reduced gastrointestinal toxicity |
| US7736624B2 (en) | 2006-06-19 | 2010-06-15 | Univ Vanderbilt | Methods and compositions for diagnostic and therapeutic targeting of COX-2 |
| US8143302B2 (en) | 2006-06-19 | 2012-03-27 | Vanderbilt University | Methods and compositions for diagnostic and therapeutic targeting of COX-2 |
| US8865130B2 (en) | 2006-06-19 | 2014-10-21 | Vanderbilt University | Methods and compositions for diagnostic and therapeutic targeting of COX-2 |
| US9346803B2 (en) | 2011-10-17 | 2016-05-24 | Vanderbilt University | Indomethacin analogs for the treatment of castrate-resistant prostate cancer |
| US9895351B2 (en) | 2011-10-17 | 2018-02-20 | Vanderbilt University | Indomethacin analogs for the treatment of castrate-resistant prostate cancer |
| US10398678B2 (en) | 2011-10-17 | 2019-09-03 | Vanderbilt University | Indomethacin analogs for the treatment of castrate-resistant prostate cancer |
| US11738004B2 (en) | 2011-10-17 | 2023-08-29 | Vanderbilt University | Indomethacin analogs for the treatment of castrate-resistant prostate cancer |
Also Published As
| Publication number | Publication date |
|---|---|
| JPH0212221B2 (enrdf_load_stackoverflow) | 1990-03-19 |
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