JPS57136559A - Nitrosourea compound and its preparation - Google Patents
Nitrosourea compound and its preparationInfo
- Publication number
- JPS57136559A JPS57136559A JP194982A JP194982A JPS57136559A JP S57136559 A JPS57136559 A JP S57136559A JP 194982 A JP194982 A JP 194982A JP 194982 A JP194982 A JP 194982A JP S57136559 A JPS57136559 A JP S57136559A
- Authority
- JP
- Japan
- Prior art keywords
- compound
- groups
- preparation
- urea
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Landscapes
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
NEW MATERIAL:The compound of formulaI(R1 is 1W12C straight-chain alkyl which may have lower aliphatic acyloxy group; R2 is 5W8C alkyl having ≥4 OH groups, or a residue obtained by removing 1-position OH group from a monosaccharide or a disaccharide, wherein said OH groups may be acylated.)
EXAMPLE: 1-(2-Chloroethyl)-1-nitroso-3-methyl-3-(1-deoxy-D-glycitolyl)urea.
USE: Antitumor agent. It has excellent antileukemic and antitumor activities, and is useful as a medicine having high safety.
PROCESS: The compound of formulaIis prepared by reacting the urea derivative of formula II with nitrous acid pref. in the presence of formic acid, acetic acid, etc. at 0W5°C.
COPYRIGHT: (C)1982,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP194982A JPS5830303B2 (en) | 1982-01-08 | 1982-01-08 | Nitrosourea compounds and their production method |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP194982A JPS5830303B2 (en) | 1982-01-08 | 1982-01-08 | Nitrosourea compounds and their production method |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS57136559A true JPS57136559A (en) | 1982-08-23 |
JPS5830303B2 JPS5830303B2 (en) | 1983-06-28 |
Family
ID=11515853
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP194982A Expired JPS5830303B2 (en) | 1982-01-08 | 1982-01-08 | Nitrosourea compounds and their production method |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5830303B2 (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102134207A (en) * | 2011-01-14 | 2011-07-27 | 厦门大学 | Urea compound and preparation method and application thereof |
-
1982
- 1982-01-08 JP JP194982A patent/JPS5830303B2/en not_active Expired
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102134207A (en) * | 2011-01-14 | 2011-07-27 | 厦门大学 | Urea compound and preparation method and application thereof |
Also Published As
Publication number | Publication date |
---|---|
JPS5830303B2 (en) | 1983-06-28 |
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