JPS56142282A - Penem-3-carboxylic acid derivative and its preparation - Google Patents
Penem-3-carboxylic acid derivative and its preparationInfo
- Publication number
- JPS56142282A JPS56142282A JP3001380A JP3001380A JPS56142282A JP S56142282 A JPS56142282 A JP S56142282A JP 3001380 A JP3001380 A JP 3001380A JP 3001380 A JP3001380 A JP 3001380A JP S56142282 A JPS56142282 A JP S56142282A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- alkyl
- group
- carboxylic acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 abstract 5
- 125000000217 alkyl group Chemical group 0.000 abstract 4
- 125000006239 protecting group Chemical group 0.000 abstract 3
- JYBFBEHQCOUIFO-SYPWQXSBSA-N (5r)-7-oxo-3-sulfanylidene-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid Chemical compound S1C(=S)C(C(=O)O)N2C(=O)C[C@H]21 JYBFBEHQCOUIFO-SYPWQXSBSA-N 0.000 abstract 1
- 241000894006 Bacteria Species 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 239000004599 antimicrobial Substances 0.000 abstract 1
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 244000052616 bacterial pathogen Species 0.000 abstract 1
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 239000000463 material Substances 0.000 abstract 1
- 230000001717 pathogenic effect Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
- C07D205/09—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
- C07F7/1804—Compounds having Si-O-C linkages
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (16)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP3001380A JPS56142282A (en) | 1980-03-10 | 1980-03-10 | Penem-3-carboxylic acid derivative and its preparation |
AU68172/81A AU6817281A (en) | 1980-03-10 | 1981-03-09 | 2-penem-3-carboxylic acid derivatives |
SE8101464A SE8101464L (sv) | 1980-03-10 | 1981-03-09 | 2-penem-3-karboxylsyraderivat, deras framstellning och anvendning |
GB8107415A GB2074563B (en) | 1980-03-10 | 1981-03-10 | 2-penem-3-carboxylic acid derivatives their preparation and use |
BE0/204081A BE887886A (fr) | 1980-03-10 | 1981-03-10 | Derivés de l'acide 2-peneme-3-carboxylique leur preparation et leur application thérapeutique. |
FR8104709A FR2477547A1 (fr) | 1980-03-10 | 1981-03-10 | Derives de l'acide 2-peneme-3-carboxylique, leur preparation et leur application therapeutique |
DE19813109086 DE3109086A1 (de) | 1980-03-10 | 1981-03-10 | 2-penem-3-carbonsaeure-derivate, verfahren zu ihrer herstellung und ihre verwendung |
ES500253A ES8205808A1 (es) | 1980-03-10 | 1981-03-10 | Un procedimiento para la preparacion de nuevos derivados del acido 2-penem-3-carboxilico. |
IT67330/81A IT1172228B (it) | 1980-03-10 | 1981-03-10 | Derivati dell acido 2 penem 3 carbossilico loro preparazione ed impiego come antibiotici |
PL23007481A PL230074A1 (enrdf_load_stackoverflow) | 1980-03-10 | 1981-03-10 | |
ZA00811567A ZA811567B (en) | 1980-03-10 | 1981-03-10 | 2-penem-3-carboxylic acid derivatives, their preparation and use |
DK108581A DK108581A (da) | 1980-03-10 | 1981-03-10 | 2-penem-3-carboxylsyre-derivater og fremgangsmaade til fremstiling heraf |
DD81228171A DD157801A5 (de) | 1980-03-10 | 1981-03-10 | Verfahren zur herstellung von 2-penem-3-karbonsaeure-abkoemmlingen |
CH1634/81A CH653034A5 (de) | 1980-03-10 | 1981-03-10 | 2-thioxopenam-3-carbonsaeurederivate sowie ihre tautomere und diese erstgenannten verbindungen enthaltendes pharmazeutisches praeparat. |
NL8101167A NL8101167A (nl) | 1980-03-10 | 1981-03-10 | 2-penem-3-carbonzuurverbindingen, hun bereiding en gebruik. |
US06/582,152 US4639441A (en) | 1980-03-10 | 1984-02-24 | 2-penem-3-carboxylic acid derivatives and use |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP3001380A JPS56142282A (en) | 1980-03-10 | 1980-03-10 | Penem-3-carboxylic acid derivative and its preparation |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS56142282A true JPS56142282A (en) | 1981-11-06 |
JPH0134994B2 JPH0134994B2 (enrdf_load_stackoverflow) | 1989-07-21 |
Family
ID=12291973
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP3001380A Granted JPS56142282A (en) | 1980-03-10 | 1980-03-10 | Penem-3-carboxylic acid derivative and its preparation |
Country Status (4)
Country | Link |
---|---|
JP (1) | JPS56142282A (enrdf_load_stackoverflow) |
AU (1) | AU6817281A (enrdf_load_stackoverflow) |
BE (1) | BE887886A (enrdf_load_stackoverflow) |
ZA (1) | ZA811567B (enrdf_load_stackoverflow) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ATE112778T1 (de) * | 1982-11-29 | 1994-10-15 | Schering Corp | Verfahren zur herstellung von penem-verbindungen. |
US4619783A (en) * | 1983-06-10 | 1986-10-28 | Pfizer Inc. | Process and intermediates for the preparation of penem derivatives |
US4725678A (en) * | 1983-06-10 | 1988-02-16 | Pfizer Inc. | Azetidinone intermediates for the preparation of penem derivatives |
US4595539A (en) * | 1983-06-10 | 1986-06-17 | Pfizer Inc. | Preparation of penem derivatives and azetidinone intermediates |
JPH09202789A (ja) * | 1995-11-20 | 1997-08-05 | Suntory Ltd | ペネム誘導体およびこれを含有する抗菌剤 |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS53137951A (en) * | 1977-05-09 | 1978-12-01 | Ciba Geigy Ag | Thiaaaza compound having betaalactum ring |
-
1980
- 1980-03-10 JP JP3001380A patent/JPS56142282A/ja active Granted
-
1981
- 1981-03-09 AU AU68172/81A patent/AU6817281A/en not_active Abandoned
- 1981-03-10 ZA ZA00811567A patent/ZA811567B/xx unknown
- 1981-03-10 BE BE0/204081A patent/BE887886A/fr not_active IP Right Cessation
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS53137951A (en) * | 1977-05-09 | 1978-12-01 | Ciba Geigy Ag | Thiaaaza compound having betaalactum ring |
Also Published As
Publication number | Publication date |
---|---|
JPH0134994B2 (enrdf_load_stackoverflow) | 1989-07-21 |
ZA811567B (en) | 1982-04-28 |
BE887886A (fr) | 1981-09-10 |
AU6817281A (en) | 1981-09-17 |
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