JPS5540612A - 3"-acetyl-4"-isovaleryltylosin - Google Patents
3"-acetyl-4"-isovaleryltylosinInfo
- Publication number
- JPS5540612A JPS5540612A JP11302378A JP11302378A JPS5540612A JP S5540612 A JPS5540612 A JP S5540612A JP 11302378 A JP11302378 A JP 11302378A JP 11302378 A JP11302378 A JP 11302378A JP S5540612 A JPS5540612 A JP S5540612A
- Authority
- JP
- Japan
- Prior art keywords
- acetyl
- formula
- tylosin
- methanol
- isovaleryltylosin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- OKKJLVBELUTLKV-UHFFFAOYSA-N Methanol Chemical compound OC OKKJLVBELUTLKV-UHFFFAOYSA-N 0.000 abstract 6
- WFDIJRYMOXRFFG-UHFFFAOYSA-N Acetic anhydride Chemical compound CC(=O)OC(C)=O WFDIJRYMOXRFFG-UHFFFAOYSA-N 0.000 abstract 3
- 229930194936 Tylosin Natural products 0.000 abstract 2
- 239000004182 Tylosin Substances 0.000 abstract 2
- 125000000218 acetic acid group Chemical group C(C)(=O)* 0.000 abstract 2
- 230000000844 anti-bacterial effect Effects 0.000 abstract 2
- WBPYTXDJUQJLPQ-VMXQISHHSA-N tylosin Chemical compound O([C@@H]1[C@@H](C)O[C@H]([C@@H]([C@H]1N(C)C)O)O[C@@H]1[C@@H](C)[C@H](O)CC(=O)O[C@@H]([C@H](/C=C(\C)/C=C/C(=O)[C@H](C)C[C@@H]1CC=O)CO[C@H]1[C@@H]([C@H](OC)[C@H](O)[C@@H](C)O1)OC)CC)[C@H]1C[C@@](C)(O)[C@@H](O)[C@H](C)O1 WBPYTXDJUQJLPQ-VMXQISHHSA-N 0.000 abstract 2
- 229960004059 tylosin Drugs 0.000 abstract 2
- 235000019375 tylosin Nutrition 0.000 abstract 2
- FREZLSIGWNCSOQ-UHFFFAOYSA-N 3-methylbutanoyl 3-methylbutanoate Chemical compound CC(C)CC(=O)OC(=O)CC(C)C FREZLSIGWNCSOQ-UHFFFAOYSA-N 0.000 abstract 1
- 241000894006 Bacteria Species 0.000 abstract 1
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 abstract 1
- 239000000654 additive Substances 0.000 abstract 1
- 150000001412 amines Chemical class 0.000 abstract 1
- 239000003242 anti bacterial agent Substances 0.000 abstract 1
- 229940088710 antibiotic agent Drugs 0.000 abstract 1
- 230000003115 biocidal effect Effects 0.000 abstract 1
- 235000019658 bitter taste Nutrition 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 150000007529 inorganic bases Chemical class 0.000 abstract 1
- -1 isovaleryl Chemical group 0.000 abstract 1
- 239000003120 macrolide antibiotic agent Substances 0.000 abstract 1
- 239000000463 material Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000003960 organic solvent Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000006188 syrup Substances 0.000 abstract 1
- 235000020357 syrup Nutrition 0.000 abstract 1
- LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 abstract 1
- 238000007669 thermal treatment Methods 0.000 abstract 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 abstract 1
Landscapes
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (15)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP11302378A JPS5540612A (en) | 1978-09-14 | 1978-09-14 | 3"-acetyl-4"-isovaleryltylosin |
| SE7907547A SE445739B (sv) | 1978-09-14 | 1979-09-11 | 3", 4"-diacyltylosinderivat |
| IT25677/79A IT1123137B (it) | 1978-09-14 | 1979-09-12 | "3",4"-diaciltilosina e procedimento per la sua produzione |
| FR7922759A FR2436150A1 (fr) | 1978-09-14 | 1979-09-12 | Derives de 3'',4''-diacyltylosine utiles comme medicaments |
| CH830879A CH642381A5 (de) | 1978-09-14 | 1979-09-13 | Dialkanoyltylosinderivate. |
| CA335,557A CA1133899A (en) | 1978-09-14 | 1979-09-13 | 3", 4"-diacyltylosin derivatives |
| HU79TO1116A HU181976B (en) | 1978-09-14 | 1979-09-13 | Process for preparing 3",4"-diacyl-tylosin derivatives |
| GB7931717A GB2031418B (en) | 1978-09-14 | 1979-09-13 | 3'',4''-diacyl derivatives of tylosin |
| DK382979A DK153492C (da) | 1978-09-14 | 1979-09-13 | Fremgangsmaade til fremstilling af 3ae, 4ae-diacyltylosinderivater |
| US06/075,661 US4268665A (en) | 1978-09-14 | 1979-09-14 | Derivatives of antibiotic tylosin |
| DE19792937267 DE2937267A1 (de) | 1978-09-14 | 1979-09-14 | 3'',4''-diacyltylosinderivate |
| NL7906894A NL7906894A (nl) | 1978-09-14 | 1979-09-14 | 3",4"-diacyltylosinederivaten. |
| AT0607479A AT366699B (de) | 1978-09-14 | 1979-09-14 | Verfahren zur herstellung von 3'', 4''-diacyltylosinderivaten |
| AT0518080A AT367432B (de) | 1978-09-14 | 1980-10-20 | Verfahren zur herstellung von neuen 3",4"diacyltylosinderivaten |
| DK446985A DK156071C (da) | 1978-09-14 | 1985-10-02 | Fremgangsmaade til fremstilling af 3,3'',4''-triacyltylosinderivater |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP11302378A JPS5540612A (en) | 1978-09-14 | 1978-09-14 | 3"-acetyl-4"-isovaleryltylosin |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS5540612A true JPS5540612A (en) | 1980-03-22 |
| JPS6155517B2 JPS6155517B2 (en, 2012) | 1986-11-28 |
Family
ID=14601497
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP11302378A Granted JPS5540612A (en) | 1978-09-14 | 1978-09-14 | 3"-acetyl-4"-isovaleryltylosin |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JPS5540612A (en, 2012) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH0375315U (en, 2012) * | 1989-11-28 | 1991-07-29 |
-
1978
- 1978-09-14 JP JP11302378A patent/JPS5540612A/ja active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| JPS6155517B2 (en, 2012) | 1986-11-28 |
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