JPS5297952A - Aminoalcohol derivatives and preparation thereof - Google Patents

Aminoalcohol derivatives and preparation thereof

Info

Publication number
JPS5297952A
JPS5297952A JP13785976A JP13785976A JPS5297952A JP S5297952 A JPS5297952 A JP S5297952A JP 13785976 A JP13785976 A JP 13785976A JP 13785976 A JP13785976 A JP 13785976A JP S5297952 A JPS5297952 A JP S5297952A
Authority
JP
Japan
Prior art keywords
preparation
aminoalcohol derivatives
aminoalcohol
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP13785976A
Other languages
English (en)
Other versions
JPS63435B2 (ja
Inventor
Ranberin Jiyorujiyu
Rooba Yozefu
Gire Kuroodo
Ronkushi Romeo
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Continental Pharma Inc
Original Assignee
Continental Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Continental Pharma Inc filed Critical Continental Pharma Inc
Publication of JPS5297952A publication Critical patent/JPS5297952A/ja
Publication of JPS63435B2 publication Critical patent/JPS63435B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
    • C07D211/14—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
    • C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D327/00—Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D327/02—Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms one oxygen atom and one sulfur atom
    • C07D327/06—Six-membered rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D335/00—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom
    • C07D335/04—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D335/06—Benzothiopyrans; Hydrogenated benzothiopyrans
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D337/00—Heterocyclic compounds containing rings of more than six members having one sulfur atom as the only ring hetero atom
    • C07D337/02—Seven-membered rings
    • C07D337/06—Seven-membered rings condensed with carbocyclic rings or ring systems
    • C07D337/08—Seven-membered rings condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D339/00—Heterocyclic compounds containing rings having two sulfur atoms as the only ring hetero atoms
    • C07D339/08—Six-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Hydrogenated Pyridines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
JP13785976A 1975-11-18 1976-11-18 Aminoalcohol derivatives and preparation thereof Granted JPS5297952A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7535217A FR2332010A1 (fr) 1975-11-18 1975-11-18 Amino-alcool heterocyclique, son sel et son procede de preparation

Publications (2)

Publication Number Publication Date
JPS5297952A true JPS5297952A (en) 1977-08-17
JPS63435B2 JPS63435B2 (ja) 1988-01-07

Family

ID=9162563

Family Applications (2)

Application Number Title Priority Date Filing Date
JP13785976A Granted JPS5297952A (en) 1975-11-18 1976-11-18 Aminoalcohol derivatives and preparation thereof
JP57002388A Expired JPS6017778B2 (ja) 1975-11-18 1982-01-12 アミノアルコ−ル誘導体およびその塩，並びにこれらの製造方法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP57002388A Expired JPS6017778B2 (ja) 1975-11-18 1982-01-12 アミノアルコ−ル誘導体およびその塩，並びにこれらの製造方法

Country Status (21)

Country Link
JP (2) JPS5297952A (ja)
AT (1) AT355566B (ja)
AU (1) AU510315B2 (ja)
BE (1) BE848496A (ja)
CA (1) CA1094088A (ja)
CH (2) CH623321A5 (ja)
DE (1) DE2651572C2 (ja)
DK (1) DK151330C (ja)
ES (1) ES453389A1 (ja)
FI (1) FI763265A (ja)
FR (1) FR2332010A1 (ja)
GB (1) GB1565080A (ja)
GR (1) GR62012B (ja)
IE (1) IE44265B1 (ja)
IL (1) IL50932A (ja)
MX (1) MX4881E (ja)
NL (1) NL180936C (ja)
NZ (1) NZ182665A (ja)
PT (1) PT65853B (ja)
SE (1) SE434744B (ja)
ZA (1) ZA766907B (ja)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6319916B1 (en) 1992-04-24 2001-11-20 Takeda Chemical Industries, Ltd. Heterocyclic compounds, their production and use

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2512817A1 (fr) * 1981-09-17 1983-03-18 Roussel Uclaf Nouveaux derives de l'aminomethyl 1h-indole-4-methanol et leurs sels, leur procede de preparation, leur application a titre de medicaments, les compositions les renfermant et leurs intermediaires de preparation
US4562200A (en) * 1983-06-30 1985-12-31 American Home Products Corporation 5(Indolyl) and 5(2,3-dihydroindolyl) substituted aminoethanols and their use as anti-hypertensives
US4521606A (en) * 1983-06-30 1985-06-04 American Home Products Corp. 5-Indolyl substituted aminoethanols
US4622399A (en) * 1983-06-30 1986-11-11 American Home Products Corporation Bicyclo-heterocyclic nitrogen substituted aminoethanol derivatives
US5705515A (en) * 1994-04-26 1998-01-06 Merck & Co., Inc. Substituted sulfonamides as selective β-3 agonists for the treatment of diabetes and obesity
US5541197A (en) * 1994-04-26 1996-07-30 Merck & Co., Inc. Substituted sulfonamides as selective β3 agonists for the treatment of diabetes and obesity
US5561142A (en) * 1994-04-26 1996-10-01 Merck & Co., Inc. Substituted sulfonamides as selective β3 agonists for the treatment of diabetes and obesity
US5656661A (en) * 1994-07-27 1997-08-12 The Procter & Gamble Company Dihydrobenzofuran and related compounds useful as anti-inflammatory agents
US5684002A (en) * 1994-09-07 1997-11-04 The Procter & Gamble Company Dihydorbenzofuran and related compounds useful as anti-inflammatory agents
EP0882707B1 (en) 1996-01-10 2003-10-08 Asahi Kasei Kabushiki Kaisha Novel tricyclic compounds and drug compositions containing the same
US5672620A (en) * 1996-02-01 1997-09-30 The Procter & Gamble Company Dihydrobenzofuran and related compounds useful as anti-inflammatory agents
US5684031A (en) * 1996-02-01 1997-11-04 The Procter & Gamble Company Dihydrobenzofuran and related compounds useful as anti-inflammatory agents
FR2758820B1 (fr) * 1997-01-30 1999-02-26 Synthelabo Derives de alpha-azacyclomethyl-benzofurane, leur preparation et leur application en therapeutique
AU6218598A (en) * 1997-01-30 1998-08-25 Synthelabo Alpha-azacyclomethyl benzothiophene and alpha-azacyclomethyl benzofurane derivatives, preparation and therapeutic application
DE997458T1 (de) * 1997-07-03 2001-03-01 Asahi Chemical Ind Tricyclische verbindungen mit gesättigten ringen und diese enthaltende medizinische zubereitungen
DK1277736T3 (da) 2000-04-28 2007-10-01 Asahi Kasei Pharma Corp Hidtil ukendte bicykliske forbindelser
EP1935882B1 (en) 2001-10-25 2011-02-09 Asahi Kasei Pharma Corporation Bicyclic compounds
JPWO2010041568A1 (ja) 2008-10-09 2012-03-08 旭化成ファーマ株式会社 インダゾール誘導体
KR20110050734A (ko) 2008-10-09 2011-05-16 아사히 가세이 파마 가부시키가이샤 인다졸 화합물

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1013224A (en) * 1962-06-21 1965-12-15 Ici Ltd Heterocyclic aminoethanols
US3255249A (en) * 1963-04-26 1966-06-07 Ici Ltd 2-branched lower alkyl-amino-1-(indan-, hydrogenated indan- and hydrogenated naphth-2-yl) lower alkanols
CH442302A (de) * 1964-04-17 1967-08-31 Sandoz Ag Verfahren zur Herstellung eines neuen Indolderivates
FR2138488A1 (en) * 1971-05-27 1973-01-05 Lipha 1-(5-indanyl)-omega-aminoalkanes - with tranquillizing activity

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6319916B1 (en) 1992-04-24 2001-11-20 Takeda Chemical Industries, Ltd. Heterocyclic compounds, their production and use

Also Published As

Publication number Publication date
BE848496A (fr) 1977-05-18
SE434744B (sv) 1984-08-13
DK151330C (da) 1988-04-25
AU1977976A (en) 1978-05-25
AU510315B2 (en) 1980-06-19
JPS63435B2 (ja) 1988-01-07
NZ182665A (en) 1978-11-13
JPS57145843A (en) 1982-09-09
JPS6017778B2 (ja) 1985-05-07
SE7612554L (sv) 1977-05-19
IE44265B1 (en) 1981-09-23
FI763265A (ja) 1977-05-19
NL7612794A (nl) 1977-05-23
GR62012B (en) 1979-02-15
FR2332010B1 (ja) 1979-06-29
NL180936B (nl) 1986-12-16
ZA766907B (en) 1977-10-26
PT65853A (fr) 1976-12-01
MX4881E (es) 1982-11-30
ES453389A1 (es) 1977-11-16
IL50932A (en) 1984-01-31
ATA854376A (de) 1979-08-15
DK151330B (da) 1987-11-23
DE2651572A1 (de) 1977-06-08
IE44265L (en) 1977-05-18
CH623321A5 (en) 1981-05-29
DK517076A (da) 1977-05-19
AT355566B (de) 1980-03-10
FR2332010A1 (fr) 1977-06-17
IL50932A0 (en) 1977-01-31
GB1565080A (en) 1980-04-16
NL180936C (nl) 1987-05-18
DE2651572C2 (de) 1982-05-19
PT65853B (fr) 1978-05-15
CH622770A5 (en) 1981-04-30
CA1094088A (en) 1981-01-20

Similar Documents

Publication Publication Date Title
JPS52106877A (en) Novel pyridinecarboxyamides and their preparation
JPS5297952A (en) Aminoalcohol derivatives and preparation thereof
JPS5289662A (en) Novel polyhalogenoosteroid and preparation thereof
GB1538240A (en) O-2-isocephem compounds and their preparation
JPS5219670A (en) Chromann44ons and preparation method thereof
JPS5262399A (en) Polyamideterpolymer and preparation thereof
IL49516A (en) 3-amino-4-deoxo-4-imino and amino-rifamycins and their preparation
JPS51138609A (en) 12222tetrafluoroethyll fluoromethilether and its preparation
IL50657A (en) 11-deoxy-16-aryl- -tetranor-prosta-cis-5-ene-13-yneoic acid derivatives and their preparation
JPS5248674A (en) Benzisoquinolines and preparation method thereof
IL50080A0 (en) New azabicycloheptanes and their preparation
JPS51138667A (en) Anthraquinoneebissamizine and preparation*
JPS5212175A (en) Triazaspirodecanone derivatives and preparation method thereof
IL58505A0 (en) 16,16-disubstituted androst-5-ene derivatives and their preparation
JPS51143630A (en) Nnbenzyll2* 22dimethoxyyacetamide and preparation
JPS5217478A (en) New homophthalimide derivatives and preparation method thereof
IL50536A (en) N-((5-methoxy-6-haloindol-3-yl) ethyl) alkanoylamides and their preparation
JPS5212158A (en) Epoxyandrostane and preparation thereof
JPS5257310A (en) Antiihemophilia agent and preparation thereof
JPS5251364A (en) Thiazolizine derivatives and preparation thereof
NZ182426A (en) Aroyl-phenylindene and aroyl-phenyl-naphthalene derivatives
JPS5219649A (en) Novel triaminoo androstane derivatives and preparation thereof
IL50820A0 (en) Novel rifamycin derivatives and their preparation
JPS51125338A (en) Diphenylether derivatives and preparation thereof
JPS523060A (en) Paraachlorophenoxyisobutyric acid derivatives and preparation thereof