JPS5042021A - - Google Patents

Info

Publication number
JPS5042021A
JPS5042021A JP49075928A JP7592874A JPS5042021A JP S5042021 A JPS5042021 A JP S5042021A JP 49075928 A JP49075928 A JP 49075928A JP 7592874 A JP7592874 A JP 7592874A JP S5042021 A JPS5042021 A JP S5042021A
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP49075928A
Other versions
JPS5314080B2 (ja
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from IT2706673A external-priority patent/IT1043857B/it
Priority claimed from IT1977474A external-priority patent/IT1054154B/it
Application filed filed Critical
Publication of JPS5042021A publication Critical patent/JPS5042021A/ja
Publication of JPS5314080B2 publication Critical patent/JPS5314080B2/ja
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18Bridged systems
JP7592874A 1973-07-25 1974-07-04 Expired JPS5314080B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT2706673A IT1043857B (it) 1973-07-25 1973-07-25 Derivati delle rifapicime procedimento della loro sintesi e loro impiego quali intermeni per la produzione di sofamicine
IT1977474A IT1054154B (it) 1974-01-24 1974-01-24 Procedimento per la preparazione di ossazino rifamione

Publications (2)

Publication Number Publication Date
JPS5042021A true JPS5042021A (ja) 1975-04-16
JPS5314080B2 JPS5314080B2 (ja) 1978-05-15

Family

ID=26327298

Family Applications (2)

Application Number Title Priority Date Filing Date
JP7592774A Expired JPS5339440B2 (ja) 1973-07-25 1974-07-04
JP7592874A Expired JPS5314080B2 (ja) 1973-07-25 1974-07-04

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP7592774A Expired JPS5339440B2 (ja) 1973-07-25 1974-07-04

Country Status (25)

Country Link
US (3) US3963705A (ja)
JP (2) JPS5339440B2 (ja)
AR (2) AR207762A1 (ja)
AT (2) AT334530B (ja)
BE (2) BE815122A (ja)
CA (2) CA1024139A (ja)
CH (2) CH615683A5 (ja)
DD (2) DD112133A5 (ja)
DE (2) DE2428387A1 (ja)
DK (2) DK284874A (ja)
ES (2) ES429060A1 (ja)
FI (2) FI153574A (ja)
FR (2) FR2257297B1 (ja)
GB (2) GB1454801A (ja)
HU (2) HU167983B (ja)
IE (2) IE39388B1 (ja)
IN (2) IN138735B (ja)
NL (2) NL7409892A (ja)
NO (2) NO142305C (ja)
PH (1) PH13691A (ja)
PL (1) PL91647B1 (ja)
RO (1) RO63865A (ja)
SE (2) SE393112B (ja)
SU (2) SU613725A3 (ja)
YU (2) YU36720B (ja)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5473799A (en) * 1977-11-16 1979-06-13 Kanebo Ltd Preparation of 1,3-oxazino (5,6-c) rifamycin derivative
JPS5473798A (en) * 1977-11-15 1979-06-13 Kanebo Ltd Novel 1,3-oxazino (5,6-c) rifamycin derivative
JPS5484600A (en) * 1977-12-15 1979-07-05 Kanebo Ltd Preparation of 1,3-oxazino 5,6-c rifamycin derivative
JPS5776597A (en) * 1980-10-30 1982-05-13 Kiyouritsu Kurieiteibu Asoshie Electric musical instrument

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR207762A1 (es) * 1973-07-25 1976-10-29 Archifar Ind Chim Trentino Procedimiento para la preparacion de 3-((4-metil-1-piperazin-1-il)-imino)-metil-rifamicina sv o rifampicina
GB1576886A (en) * 1977-04-20 1980-10-15 Lepetit Spa Rifamycin derivatives
US4179439A (en) * 1977-07-01 1979-12-18 Intreprinderea De Antibiotice Iasi Rifamycins and method for their preparation
GB1594134A (en) * 1977-11-25 1981-07-30 Holco Investment Inc Rifamycins
JPS58115705U (ja) * 1982-02-01 1983-08-08 株式会社ニコン カメラのフアインダ光学系
GB8308166D0 (en) * 1983-03-24 1983-05-05 Erba Farmitalia Preparation of azinomethyl-rifamycins
GB8318072D0 (en) * 1983-07-04 1983-08-03 Lepetit Spa Water-soluble rifampicin derivatives
DE69735383T2 (de) * 1996-11-19 2007-02-15 Georgetown University Methode zur Inhibierung von HEREGULIN und seines Rezeptors sowie Verwendung zur Inhibierung von Krebszellen
US20090275594A1 (en) * 2008-05-05 2009-11-05 Macielag Mark J 3-hydrazone piperazinyl rifamycin derivatives useful as antimicrobial agents
CN103755723B (zh) * 2014-02-07 2016-04-20 天津大学 一种利福平i晶型的制备方法
CN103951677B (zh) * 2014-03-17 2016-04-06 四川省长征药业股份有限公司 利福喷丁的制备方法
CN106632394A (zh) * 2016-11-15 2017-05-10 南京工业大学 一种利用釜式反应装置与微通道反应装置串联反应制备利福平的方法
CN106749326A (zh) * 2016-11-28 2017-05-31 南京工业大学 一种由利福霉素s钠盐连续生产制备利福平的方法
CN111848639A (zh) * 2020-07-09 2020-10-30 华东理工大学 一种合成利福平的工艺方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1090115A (en) * 1964-04-02 1967-11-08 Lepetit Spa Mannich bases of rifamycin sv
FR208F (ja) * 1964-07-31
DE1795568C3 (de) * 1964-07-31 1974-07-18 Gruppo Lepetit S.P.A., Mailand (Italien) 3-Hydroxymethyl-rifamycin SV und Verfahren zu seiner Herstellung. Ausscheidung aus: 1595883
US3542762A (en) * 1967-06-07 1970-11-24 Lepetit Spa Process for rifamycins
AR207762A1 (es) * 1973-07-25 1976-10-29 Archifar Ind Chim Trentino Procedimiento para la preparacion de 3-((4-metil-1-piperazin-1-il)-imino)-metil-rifamicina sv o rifampicina

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5473798A (en) * 1977-11-15 1979-06-13 Kanebo Ltd Novel 1,3-oxazino (5,6-c) rifamycin derivative
JPS5473799A (en) * 1977-11-16 1979-06-13 Kanebo Ltd Preparation of 1,3-oxazino (5,6-c) rifamycin derivative
JPS5484600A (en) * 1977-12-15 1979-07-05 Kanebo Ltd Preparation of 1,3-oxazino 5,6-c rifamycin derivative
JPS5776597A (en) * 1980-10-30 1982-05-13 Kiyouritsu Kurieiteibu Asoshie Electric musical instrument

Also Published As

Publication number Publication date
NO741764L (ja) 1975-02-24
DD112267A5 (ja) 1975-04-05
FI153574A (ja) 1975-01-26
FI60397C (fi) 1982-01-11
BE817823A (fr) 1974-11-18
NO142305C (no) 1980-07-30
FR2245631B1 (ja) 1978-09-15
AT334530B (de) 1976-01-25
GB1454802A (en) 1976-11-03
ATA496174A (de) 1976-05-15
AU6990574A (en) 1975-12-11
DK135286B (da) 1977-03-28
CH611296A5 (ja) 1979-05-31
CA1024139A (en) 1978-01-10
USRE31587E (en) 1984-05-22
YU36719B (en) 1984-08-31
DK284774A (ja) 1975-01-26
US3925366A (en) 1975-12-09
IE39389B1 (en) 1978-09-27
FR2257297B1 (ja) 1978-07-21
SE7406073L (ja) 1975-01-27
SU576943A3 (ru) 1977-10-15
IN138735B (ja) 1976-03-27
SE7406074L (ja) 1975-01-27
YU132574A (en) 1981-11-13
SE393112B (sv) 1977-05-02
DE2433105A1 (de) 1975-02-06
SU613725A3 (ru) 1978-06-30
NL181992B (nl) 1987-07-16
AU6991074A (en) 1975-12-11
HU168723B (ja) 1976-07-28
AR207762A1 (es) 1976-10-29
DK284874A (da) 1975-01-26
DE2428387A1 (de) 1975-02-13
PL91647B1 (ja) 1977-03-31
HU167983B (ja) 1976-02-28
NO142305B (no) 1980-04-21
NL181992C (nl) 1987-12-16
YU132474A (en) 1981-11-13
NL7409955A (nl) 1975-01-28
JPS5314080B2 (ja) 1978-05-15
ES429059A1 (es) 1976-08-16
YU36720B (en) 1984-08-31
NL7409892A (nl) 1975-01-28
JPS5041897A (ja) 1975-04-16
RO63865A (fr) 1979-01-15
CH615683A5 (ja) 1980-02-15
AR207763A1 (es) 1976-10-29
CA1022548A (en) 1977-12-13
BE815122A (fr) 1974-09-16
JPS5339440B2 (ja) 1978-10-21
IE39388B1 (en) 1978-09-27
FI60397B (fi) 1981-09-30
IE39388L (en) 1975-01-25
SE407803B (sv) 1979-04-23
IN139074B (ja) 1976-05-01
FI157574A (ja) 1975-01-26
NO741763L (ja) 1975-02-24
FR2257297A1 (ja) 1975-08-08
US3963705A (en) 1976-06-15
PH13691A (en) 1980-09-01
GB1454801A (en) 1976-11-03
IE39389L (en) 1975-01-25
FR2245631A1 (ja) 1975-04-25
DD112133A5 (ja) 1975-03-20
DK135286C (ja) 1977-09-05
DE2433105C2 (ja) 1988-03-31
SU613725A1 (ja) 1978-06-30
ES429060A1 (es) 1976-08-16
AT334531B (de) 1976-01-25
ATA596774A (de) 1976-05-15

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