JPH08506123A - 側鎖フルオロ置換３−カルボキシステロイド - Google Patents

側鎖フルオロ置換３−カルボキシステロイド

Info

Publication number
JPH08506123A
JPH08506123A JP7514811A JP51481194A JPH08506123A JP H08506123 A JPH08506123 A JP H08506123A JP 7514811 A JP7514811 A JP 7514811A JP 51481194 A JP51481194 A JP 51481194A JP H08506123 A JPH08506123 A JP H08506123A
Authority
JP
Japan
Prior art keywords
methyl
androsta
carbamoyl
diene
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP7514811A
Other languages
English (en)
Japanese (ja)
Inventor
パンツエーリ，アキーレ
ネジ，マルチエラ
デイ・サーレ，エンリコ
Original Assignee
フアルマシア・エツセ・ピー・アー
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by フアルマシア・エツセ・ピー・アー filed Critical フアルマシア・エツセ・ピー・アー
Publication of JPH08506123A publication Critical patent/JPH08506123A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0066—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by a carbon atom forming part of an amide group
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP7514811A 1993-11-26 1994-11-17 側鎖フルオロ置換３−カルボキシステロイド Pending JPH08506123A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB939324371A GB9324371D0 (en) 1993-11-26 1993-11-26 Side chain fluoro substituted 3-carboxysteroids
GB9324371.5 1993-11-26
PCT/EP1994/003809 WO1995014709A1 (en) 1993-11-26 1994-11-17 Side chain fluoro substituted 3-carboxysteroids

Publications (1)

Publication Number Publication Date
JPH08506123A true JPH08506123A (ja) 1996-07-02

Family

ID=10745772

Family Applications (1)

Application Number Title Priority Date Filing Date
JP7514811A Pending JPH08506123A (ja) 1993-11-26 1994-11-17 側鎖フルオロ置換３−カルボキシステロイド

Country Status (4)

Country Link
EP (1) EP0681587A1 (de)
JP (1) JPH08506123A (de)
GB (1) GB9324371D0 (de)
WO (1) WO1995014709A1 (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9415183D0 (en) * 1994-07-28 1994-09-21 Erba Carlo Spa 3-carboxysteroids with a fluorinated side-chain

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1259419B (it) * 1991-05-24 1996-03-18 Erba Carlo Spa Steroidi 3-carbossi 17b - sostituiti insaturi utili come inibitori della testosterone 5 a reduttasi
EP0725074A3 (de) * 1992-04-20 1996-11-20 Sankyo Co Verbindungen zur Verwendung also Zwischenprodukte zur Herstellung von Androst-3,5-dien-3-carboxy-Derivaten

Also Published As

Publication number Publication date
EP0681587A1 (de) 1995-11-15
GB9324371D0 (en) 1994-01-12
WO1995014709A1 (en) 1995-06-01

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