JPH0770082A - ２−ヒドロキシ−３−〔１−（１ｈ−イミダゾール−４−イル）アルキル〕−ベンゼンカルボキシミダミド - Google Patents

２−ヒドロキシ−３−〔１−（１ｈ−イミダゾール−４−イル）アルキル〕−ベンゼンカルボキシミダミド

Info

Publication number
JPH0770082A
JPH0770082A JP6112960A JP11296094A JPH0770082A JP H0770082 A JPH0770082 A JP H0770082A JP 6112960 A JP6112960 A JP 6112960A JP 11296094 A JP11296094 A JP 11296094A JP H0770082 A JPH0770082 A JP H0770082A
Authority
JP
Japan
Prior art keywords
hydroxy
imidazol
alkyl
benzenecarboximidamide
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP6112960A
Other languages
English (en)
Japanese (ja)
Inventor
Michel Philippe
ミシェル フィリップ
Eric Cossement
コスマン エリック
Jean Gobert
ゴベール ジャン
Ernst Wuelfert
ヴルフェルト エルンスト
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
UCB SA
Original Assignee
UCB SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by UCB SA filed Critical UCB SA
Publication of JPH0770082A publication Critical patent/JPH0770082A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Treatments For Attaching Organic Compounds To Fibrous Goods (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
JP6112960A 1993-05-27 1994-05-26 ２−ヒドロキシ−３−〔１−（１ｈ−イミダゾール−４−イル）アルキル〕−ベンゼンカルボキシミダミド Pending JPH0770082A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB93109650 1993-05-27
GB939310965A GB9310965D0 (en) 1993-05-27 1993-05-27 2-hydroxy-3-(1h-imidazol-4-yl)alkyl)benzenecarboximidamides

Publications (1)

Publication Number Publication Date
JPH0770082A true JPH0770082A (ja) 1995-03-14

Family

ID=10736226

Family Applications (1)

Application Number Title Priority Date Filing Date
JP6112960A Pending JPH0770082A (ja) 1993-05-27 1994-05-26 ２−ヒドロキシ−３−〔１−（１ｈ−イミダゾール−４−イル）アルキル〕−ベンゼンカルボキシミダミド

Country Status (21)

Country Link
US (1) US5385927A (https=)
EP (1) EP0626372B1 (https=)
JP (1) JPH0770082A (https=)
AT (1) ATE198196T1 (https=)
AU (1) AU673422B2 (https=)
CA (1) CA2124289A1 (https=)
CZ (1) CZ287136B6 (https=)
DE (1) DE69426433D1 (https=)
FI (1) FI942390L (https=)
GB (1) GB9310965D0 (https=)
HU (1) HUT67813A (https=)
IL (1) IL109750A (https=)
MY (1) MY111216A (https=)
NO (1) NO303824B1 (https=)
NZ (1) NZ260588A (https=)
PL (1) PL175970B1 (https=)
RU (1) RU2125557C1 (https=)
SG (1) SG42791A1 (https=)
SK (1) SK60394A3 (https=)
TW (1) TW263500B (https=)
ZA (1) ZA943651B (https=)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2011509297A (ja) * 2008-01-09 2011-03-24 アラーガン、インコーポレイテッド α２Ｂおよび／またはα２Ｃアドレナリン受容体のサブタイプ選択的モジュレーターとしての置換アリール−２−フェニルエチル−１Ｈ−イミダゾール化合物

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9521680D0 (en) * 1995-10-23 1996-01-03 Orion Yhtymo Oy New use of imidazole derivatives
US6200967B1 (en) 1996-06-25 2001-03-13 Eli Lilly And Company Anticoagulant agents
CA2258915A1 (en) * 1996-06-25 1997-12-31 Michael Robert Wiley Anticoagulant agents
PL360707A1 (en) * 2000-07-14 2004-09-20 Allergan Inc. Compositions containing alpha-2-adrenergic agonist components
EP2196461A1 (de) 2008-12-15 2010-06-16 Bayer CropScience AG 4-Amino-1,2,3-benzoxathiazin-Derivate als Pestizide

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8626287D0 (en) * 1986-11-04 1986-12-03 Ucb Sa Substituted 1h-imidazoles
GB8810067D0 (en) * 1988-04-28 1988-06-02 Ucb Sa Substituted 1-(1h-imidazol-4-yl)alkyl-benzamides
FI98815C (fi) * 1990-11-30 1997-08-25 Santen Oy Menetelmä uusien, farmakologisesti käyttökelpoisten bispilokarpiinihapon esterijohdannaisten valmistamiseksi

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2011509297A (ja) * 2008-01-09 2011-03-24 アラーガン、インコーポレイテッド α２Ｂおよび／またはα２Ｃアドレナリン受容体のサブタイプ選択的モジュレーターとしての置換アリール−２−フェニルエチル−１Ｈ−イミダゾール化合物

Also Published As

Publication number Publication date
HUT67813A (en) 1995-05-29
TW263500B (https=) 1995-11-21
PL175970B1 (pl) 1999-03-31
ZA943651B (en) 1995-01-26
US5385927A (en) 1995-01-31
RU2125557C1 (ru) 1999-01-27
EP0626372B1 (fr) 2000-12-20
MY111216A (en) 1999-09-30
NO941932D0 (no) 1994-05-25
CZ287136B6 (en) 2000-09-13
IL109750A0 (en) 1994-08-26
NO941932L (no) 1994-11-28
DE69426433D1 (de) 2001-01-25
CA2124289A1 (en) 1994-11-28
NO303824B1 (no) 1998-09-07
AU6330394A (en) 1994-12-01
FI942390A7 (fi) 1994-11-28
EP0626372A1 (fr) 1994-11-30
IL109750A (en) 1998-06-15
FI942390L (fi) 1994-11-28
NZ260588A (en) 1995-09-26
SG42791A1 (en) 1997-10-17
AU673422B2 (en) 1996-11-07
CZ124794A3 (en) 1994-12-15
FI942390A0 (fi) 1994-05-24
SK60394A3 (en) 1995-07-11
ATE198196T1 (de) 2001-01-15
HU9401574D0 (en) 1994-08-29
GB9310965D0 (en) 1993-07-14

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