JPH06506443A - アザ二環式およびアザ三環式誘導体、その製法および中間体ならびに該化合物含有の医薬組成物 - Google Patents
アザ二環式およびアザ三環式誘導体、その製法および中間体ならびに該化合物含有の医薬組成物Info
- Publication number
- JPH06506443A JPH06506443A JP4502573A JP50257392A JPH06506443A JP H06506443 A JPH06506443 A JP H06506443A JP 4502573 A JP4502573 A JP 4502573A JP 50257392 A JP50257392 A JP 50257392A JP H06506443 A JPH06506443 A JP H06506443A
- Authority
- JP
- Japan
- Prior art keywords
- hydrogen
- alkyl
- formula
- compound
- tables
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB919100370A GB9100370D0 (en) | 1991-01-09 | 1991-01-09 | Pharmaceuticals |
GB9100370.7 | 1991-01-09 | ||
GB9100580.1 | 1991-01-10 | ||
GB919100580A GB9100580D0 (en) | 1991-01-10 | 1991-01-10 | Pharmaceuticals |
PCT/GB1992/000050 WO1992012149A1 (fr) | 1991-01-09 | 1992-01-09 | Derives azabicydiques et azatricydiques, leurs procedes et intermediaires de preparation et compositions pharmaceutiques les contenant |
Publications (1)
Publication Number | Publication Date |
---|---|
JPH06506443A true JPH06506443A (ja) | 1994-07-21 |
Family
ID=26298233
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP4502573A Pending JPH06506443A (ja) | 1991-01-09 | 1992-01-09 | アザ二環式およびアザ三環式誘導体、その製法および中間体ならびに該化合物含有の医薬組成物 |
Country Status (4)
Country | Link |
---|---|
EP (1) | EP0566609A1 (fr) |
JP (1) | JPH06506443A (fr) |
AU (1) | AU1161292A (fr) |
WO (1) | WO1992012149A1 (fr) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2008044701A1 (fr) | 2006-10-11 | 2008-04-17 | Nippon Soda Co., Ltd. | Procédé de production d'un dérivé de pipéridine-4-one |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9214184D0 (en) * | 1992-07-03 | 1992-08-12 | Smithkline Beecham Plc | Pharmaceuticals |
JP3235913B2 (ja) * | 1993-07-30 | 2001-12-04 | エーザイ株式会社 | アミノ安息香酸誘導体 |
GB9721139D0 (en) * | 1997-10-07 | 1997-12-03 | Glaxo Group Ltd | Medicaments |
IT1303123B1 (it) * | 1998-10-13 | 2000-10-30 | Rotta Research Lab | Derivati basici di benz(e)isoindol-1-oni e pirrolo(3,4-c)chinolin-1-oni ad attivita' 5ht3 antagonista, loro preparazione ed |
TW200306189A (en) | 2002-03-21 | 2003-11-16 | Merz Pharma Gmbh & Co Kgaa | Azabicyclic, azatricyclic and azaspirocyclic derivatives of aminocyclohexane NMDA, 5HT3, and neuronal nicotinic receptor antagonists |
EE05516B1 (et) | 2002-09-25 | 2012-02-15 | Memory@Pharmaceuticals@Corporation | Indasoolid bensotiasoolid ja bensoisotiasoolid nende valmistamine ning kasutamine |
US6984652B2 (en) | 2003-09-05 | 2006-01-10 | Warner-Lambert Company Llc | Gyrase inhibitors |
ES2295973T3 (es) | 2003-12-22 | 2008-04-16 | Memory Pharmaceuticals Corporation | Indoles, 1h-indazoles, 1,2-bencisoxazoles, y 1,2-bencisotiazoles, y preparacion y usos de los mismos. |
EP1735306A2 (fr) | 2004-03-25 | 2006-12-27 | Memory Pharmaceuticals Corporation | Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, et leur preparation et leurs utilisations |
DE602005024677D1 (de) | 2004-04-22 | 2010-12-23 | Memory Pharm Corp | Indole, 1h-indazole, 1,2-benzisoxazole, 1,2-benzoisothiazole, deren herstellung und verwendungen |
BRPI0510212A (pt) | 2004-05-07 | 2007-10-16 | Memory Pharm Corp | 1h-indazóis, benzotiazóis, 1,2 - benzoisoxazóis, 1,2-benzoisotiazóis, e cromonas e a preparação e usos dos mesmos |
US7737163B2 (en) | 2004-06-15 | 2010-06-15 | Pfizer Inc. | Benzimidazolone carboxylic acid derivatives |
EP1758891A2 (fr) | 2004-06-15 | 2007-03-07 | Pfizer Japan Inc. | Derives de benzimidazolone d'acide carboxylique |
RU2418797C2 (ru) | 2004-12-22 | 2011-05-20 | Мемори Фармасьютиклз Корпорейшн | Лиганды никотинового рецептора альфа-7, их получение и применение |
JP4130220B1 (ja) | 2005-02-22 | 2008-08-06 | ファイザー株式会社 | 5ht4受容体アゴニストとしてのオキシインドール誘導体 |
US8106066B2 (en) | 2005-09-23 | 2012-01-31 | Memory Pharmaceuticals Corporation | Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof |
WO2022175402A1 (fr) | 2021-02-18 | 2022-08-25 | Aprea Therapeutics Ab | Dérivés de quinuclidine-3-one |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL59004A0 (en) * | 1978-12-30 | 1980-03-31 | Beecham Group Ltd | Substituted benzamides their preparation and pharmaceutical compositions containing them |
-
1992
- 1992-01-09 JP JP4502573A patent/JPH06506443A/ja active Pending
- 1992-01-09 WO PCT/GB1992/000050 patent/WO1992012149A1/fr not_active Application Discontinuation
- 1992-01-09 AU AU11612/92A patent/AU1161292A/en not_active Abandoned
- 1992-01-09 EP EP19920902098 patent/EP0566609A1/fr not_active Withdrawn
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2008044701A1 (fr) | 2006-10-11 | 2008-04-17 | Nippon Soda Co., Ltd. | Procédé de production d'un dérivé de pipéridine-4-one |
Also Published As
Publication number | Publication date |
---|---|
WO1992012149A1 (fr) | 1992-07-23 |
AU1161292A (en) | 1992-08-17 |
EP0566609A1 (fr) | 1993-10-27 |
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