AU1161292A - Azabicydic and azatricydic derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them - Google Patents

Azabicydic and azatricydic derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them

Info

Publication number
AU1161292A
AU1161292A AU11612/92A AU1161292A AU1161292A AU 1161292 A AU1161292 A AU 1161292A AU 11612/92 A AU11612/92 A AU 11612/92A AU 1161292 A AU1161292 A AU 1161292A AU 1161292 A AU1161292 A AU 1161292A
Authority
AU
Australia
Prior art keywords
azatricydic
azabicydic
intermediates
derivatives
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU11612/92A
Other languages
English (en)
Inventor
Francis David King
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Ltd
Original Assignee
SmithKline Beecham Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB919100370A external-priority patent/GB9100370D0/en
Priority claimed from GB919100580A external-priority patent/GB9100580D0/en
Application filed by SmithKline Beecham Ltd filed Critical SmithKline Beecham Ltd
Publication of AU1161292A publication Critical patent/AU1161292A/en
Abandoned legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU11612/92A 1991-01-09 1992-01-09 Azabicydic and azatricydic derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them Abandoned AU1161292A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB919100370A GB9100370D0 (en) 1991-01-09 1991-01-09 Pharmaceuticals
GB9100370 1991-01-09
GB919100580A GB9100580D0 (en) 1991-01-10 1991-01-10 Pharmaceuticals
GB9100580 1991-01-10

Publications (1)

Publication Number Publication Date
AU1161292A true AU1161292A (en) 1992-08-17

Family

ID=26298233

Family Applications (1)

Application Number Title Priority Date Filing Date
AU11612/92A Abandoned AU1161292A (en) 1991-01-09 1992-01-09 Azabicydic and azatricydic derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them

Country Status (4)

Country Link
EP (1) EP0566609A1 (fr)
JP (1) JPH06506443A (fr)
AU (1) AU1161292A (fr)
WO (1) WO1992012149A1 (fr)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9214184D0 (en) * 1992-07-03 1992-08-12 Smithkline Beecham Plc Pharmaceuticals
JP3235913B2 (ja) * 1993-07-30 2001-12-04 エーザイ株式会社 アミノ安息香酸誘導体
GB9721139D0 (en) 1997-10-07 1997-12-03 Glaxo Group Ltd Medicaments
IT1303123B1 (it) 1998-10-13 2000-10-30 Rotta Research Lab Derivati basici di benz(e)isoindol-1-oni e pirrolo(3,4-c)chinolin-1-oni ad attivita' 5ht3 antagonista, loro preparazione ed
TW200306189A (en) 2002-03-21 2003-11-16 Merz Pharma Gmbh & Co Kgaa Azabicyclic, azatricyclic and azaspirocyclic derivatives of aminocyclohexane NMDA, 5HT3, and neuronal nicotinic receptor antagonists
ES2405594T3 (es) 2002-09-25 2013-05-31 Memory Pharmaceuticals Corporation Idazoles, benzotiazoles y benzisotiazoles, y preparación y usos de los mismos
US6984652B2 (en) 2003-09-05 2006-01-10 Warner-Lambert Company Llc Gyrase inhibitors
JP4824578B2 (ja) 2003-12-22 2011-11-30 メモリー・ファーマシューティカルズ・コーポレイション インドール類、1,2−ベンズイソオキサゾール類、および1,2−ベンゾイソチアゾール類、ならびにそれらの製造と使用
BRPI0508771A (pt) 2004-03-25 2007-08-14 Memory Pharm Corp indazóis, benzotiazóis, benzoisotiazóis, benzisoxazóis, e a preparação e usos dos mesmos
ATE487716T1 (de) 2004-04-22 2010-11-15 Memory Pharm Corp Indole, 1h-indazole, 1,2-benzisoxazole, 1,2- benzoisothiazole, deren herstellung und verwendungen
US7632831B2 (en) 2004-05-07 2009-12-15 Memory Pharmaceuticals Corporation 1H-indazoles, benzothiazoles, 1,2-benzoisoxazoles, 1,2-benzoisothiazoles, and chromones and preparation and uses thereof
US7737163B2 (en) 2004-06-15 2010-06-15 Pfizer Inc. Benzimidazolone carboxylic acid derivatives
EA200801608A1 (ru) 2004-06-15 2008-10-30 Пфайзер Инк. Производные бензимидазолонкарбоновой кислоты
AU2005319248A1 (en) 2004-12-22 2006-06-29 Memory Pharmaceuticals Corporation Nicotinic alpha-7 receptor ligands and preparation and uses thereof
NZ556627A (en) 2005-02-22 2010-09-30 Pfizer Oxyindole derivatives as 5HT4 receptor agonists
US8106066B2 (en) 2005-09-23 2012-01-31 Memory Pharmaceuticals Corporation Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof
DE602007008579D1 (de) 2006-10-11 2010-09-30 Nippon Soda Co Verfahren zur herstellung eines piperidin-4-on-derivats
WO2022175402A1 (fr) 2021-02-18 2022-08-25 Aprea Therapeutics Ab Dérivés de quinuclidine-3-one

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL59004A0 (en) * 1978-12-30 1980-03-31 Beecham Group Ltd Substituted benzamides their preparation and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
WO1992012149A1 (fr) 1992-07-23
JPH06506443A (ja) 1994-07-21
EP0566609A1 (fr) 1993-10-27

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