JPH0517920B2 - - Google Patents

Info

Publication number
JPH0517920B2
JPH0517920B2 JP59273919A JP27391984A JPH0517920B2 JP H0517920 B2 JPH0517920 B2 JP H0517920B2 JP 59273919 A JP59273919 A JP 59273919A JP 27391984 A JP27391984 A JP 27391984A JP H0517920 B2 JPH0517920 B2 JP H0517920B2
Authority
JP
Japan
Prior art keywords
phosphate
fluoro
stirring
dissolved
room temperature
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP59273919A
Other languages
English (en)
Japanese (ja)
Other versions
JPS61152694A (ja
Inventor
Takako Hori
Isao Myokan
Maki Myahara
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Toyama Chemical Co Ltd
Original Assignee
Toyama Chemical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Toyama Chemical Co Ltd filed Critical Toyama Chemical Co Ltd
Priority to JP59273919A priority Critical patent/JPS61152694A/ja
Publication of JPS61152694A publication Critical patent/JPS61152694A/ja
Publication of JPH0517920B2 publication Critical patent/JPH0517920B2/ja
Granted legal-status Critical Current

Links

Classifications

    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
JP59273919A 1984-12-27 1984-12-27 新規な５−フルオロ−２′−デオキシウリジン−５′−ホスフエ−ト誘導体およびその塩 Granted JPS61152694A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP59273919A JPS61152694A (ja) 1984-12-27 1984-12-27 新規な５−フルオロ−２′−デオキシウリジン−５′−ホスフエ−ト誘導体およびその塩

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP59273919A JPS61152694A (ja) 1984-12-27 1984-12-27 新規な５−フルオロ−２′−デオキシウリジン−５′−ホスフエ−ト誘導体およびその塩

Publications (2)

Publication Number Publication Date
JPS61152694A JPS61152694A (ja) 1986-07-11
JPH0517920B2 true JPH0517920B2 (en:Method) 1993-03-10

Family

ID=17534395

Family Applications (1)

Application Number Title Priority Date Filing Date
JP59273919A Granted JPS61152694A (ja) 1984-12-27 1984-12-27 新規な５−フルオロ−２′−デオキシウリジン−５′−ホスフエ−ト誘導体およびその塩

Country Status (1)

Country Link
JP (1) JPS61152694A (en:Method)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0262876B1 (en) * 1986-09-27 1992-04-29 Toyo Jozo Kabushiki Kaisha Nucleoside-phospholipid conjugate
AU610344B2 (en) * 1988-02-29 1991-05-16 Taiho Pharmaceutical Co., Ltd. 2'-deoxy-5-fluorouridine derivatives
US7517858B1 (en) * 1995-06-07 2009-04-14 The Regents Of The University Of California Prodrugs of pharmaceuticals with improved bioavailability
IL131887A0 (en) * 1999-09-14 2001-03-19 Dpharm Ltd Phospholipid prodrugs of anti-proliferative drugs
NZ533094A (en) * 2001-11-21 2006-01-27 Heidelberg Pharma Gmbh Phospholipid derivatives of nucleosides as antitumoral medicaments
WO2007130783A2 (en) 2006-05-03 2007-11-15 Chimerix, Inc. Metabolically stable alkoxyalkyl esters of antiviral or antiproliferative phosphonates, nucleoside phosphonates and nucleoside phosphates
US8993542B2 (en) 2008-01-25 2015-03-31 Chimerix Inc. Methods of treating viral infections
AU2011216243B2 (en) 2010-02-12 2015-07-09 Chimerix, Inc. Nucleoside phosphonate salts
EP2563367A4 (en) 2010-04-26 2013-12-04 Chimerix Inc Methods of treating retroviral infections and related dosage regimes

Also Published As

Publication number Publication date
JPS61152694A (ja) 1986-07-11

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