JPH0471074B2 - - Google Patents

Info

Publication number
JPH0471074B2
JPH0471074B2 JP59127266A JP12726684A JPH0471074B2 JP H0471074 B2 JPH0471074 B2 JP H0471074B2 JP 59127266 A JP59127266 A JP 59127266A JP 12726684 A JP12726684 A JP 12726684A JP H0471074 B2 JPH0471074 B2 JP H0471074B2
Authority
JP
Japan
Prior art keywords
triazolo
compound according
phenyl
carbon atoms
amine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP59127266A
Other languages
English (en)
Japanese (ja)
Other versions
JPS6013792A (ja
Inventor
Wagunaa Hansu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
GD Searle LLC
Original Assignee
GD Searle LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by GD Searle LLC filed Critical GD Searle LLC
Publication of JPS6013792A publication Critical patent/JPS6013792A/ja
Publication of JPH0471074B2 publication Critical patent/JPH0471074B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10—Antioedematous agents; Diuretics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP59127266A 1983-06-20 1984-06-20 トリアゾロピリミジン化合物 Granted JPS6013792A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/506,157 US4483987A (en) 1983-06-20 1983-06-20 8-Substituted 7-phenyl-1,2,4-triazolo[2,3-c]pyrimidines-5-amines and amides
US506157 1983-06-20

Publications (2)

Publication Number Publication Date
JPS6013792A JPS6013792A (ja) 1985-01-24
JPH0471074B2 true JPH0471074B2 (enExample) 1992-11-12

Family

ID=24013440

Family Applications (1)

Application Number Title Priority Date Filing Date
JP59127266A Granted JPS6013792A (ja) 1983-06-20 1984-06-20 トリアゾロピリミジン化合物

Country Status (7)

Country Link
US (1) US4483987A (enExample)
EP (1) EP0129247A1 (enExample)
JP (1) JPS6013792A (enExample)
AU (1) AU566670B2 (enExample)
CA (1) CA1204741A (enExample)
ES (1) ES8506714A1 (enExample)
ZA (1) ZA844669B (enExample)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3130633A1 (de) * 1981-08-01 1983-02-17 Basf Ag, 6700 Ludwigshafen 7-amino-azolo(1,5-a)pyrimidine und diese enthaltende fungizide
US4562192A (en) * 1984-02-03 1985-12-31 G. D. Searle & Co. 6-Substituted-5-phenyltetrazolo[1,5-a][1,2,4]triazole[1,5-c]pyrimidines, and pharmaceutical compositions containing them
JPS62107954A (ja) * 1985-11-05 1987-05-19 Tomiji Saito 可塑性研磨材料
EP0244948A3 (en) * 1986-04-30 1989-03-15 Schering Agrochemicals Limited Triazolopyrimidine herbicides
JPH07115284B2 (ja) * 1986-07-18 1995-12-13 株式会社東芝 非球面部材のみがき装置
US5338743A (en) * 1988-06-06 1994-08-16 Fujisawa Pharmaceutical Co., Ltd. New use of the adenosine antagonist
US4866063A (en) * 1988-12-22 1989-09-12 G. D. Searle & Co. Diol metabolites of 7-phenyl-1,2,4-triazolo[2,3-c]pyrimidines-5-amines
FR2687676B1 (fr) * 1992-02-24 1994-07-08 Union Pharma Scient Appl Nouveaux derives de polyazaindenes antagonistes des recepteurs a l'angiotensine ii; leurs procedes de preparation, compositions pharmaceutiques les contenant.
CA2284737C (en) * 1997-03-24 2007-03-13 Kyowa Hakko Kogyo Co., Ltd. [1,2,4]triazolo[1,5-c]pyrimidine derivatives
WO2000017201A1 (en) 1998-09-22 2000-03-30 Kyowa Hakko Kogyo Co., Ltd. [1,2,4]TRIAZOLO[1,5-c]PYRIMIDINE DERIVATIVES
JP2001302667A (ja) * 2000-04-28 2001-10-31 Bayer Ag イミダゾピリミジン誘導体およびトリアゾロピリミジン誘導体
US6998148B1 (en) 2001-03-28 2006-02-14 Shipley Company, L.L.C. Porous materials
MXPA04004534A (es) * 2001-11-16 2004-08-11 Childrens Medical Center Aumento de la funcion de un organo.
AU2003272886A1 (en) * 2002-09-24 2004-04-19 Kyowa Hakko Kogyo Co., Ltd. (1,2,4)-TRIAZOLO(1,5-c)PYRIMIDINE DERIVATIVE
WO2020106560A1 (en) * 2018-11-20 2020-05-28 Merck Sharp & Dohme Corp. Substituted amino triazolopyrimidine and amino triazolopyrazine adenosine receptor antagonists, pharmaceutical compositions and their use

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3053844A (en) * 1959-04-13 1962-09-11 Ici Ltd Mono-acyl derivatives of s-triazolo [2, 3-c] pyrimidines
US3046276A (en) * 1959-06-15 1962-07-24 Ici Ltd S-triazolo-[2, 3-c] pyrimidine derivatives
US4205169A (en) * 1979-04-09 1980-05-27 G. D. Searle & Co. N-[4-Azido-5-(2-ethoxyethyl)-6-phenyl-2-pyrimidinyl]acetamide and congeners
US4405780A (en) * 1979-08-08 1983-09-20 G. D. Searle & Co. 8-Substituted 7-phenyl-1,2,4,-triazolo[4,3-c]/[2,3-c]pyrimidines-5-amines and amides
AU531507B2 (en) * 1979-08-08 1983-08-25 G.D. Searle & Co. 8-substituted 7-phenyl-1,2,4-triazolo(4,3-c) pyrimidines -5-amines and amides
US4269980A (en) * 1979-12-17 1981-05-26 American Cyanamid Company (Substituted-phenyl)-1,2,4-triazolo[4,3-c]pyrimidines and (substituted-phenyl)-1,2,4-triazolo[1,5-c]pyrimidines

Also Published As

Publication number Publication date
CA1204741A (en) 1986-05-20
ES533537A0 (es) 1985-08-01
ES8506714A1 (es) 1985-08-01
AU2949484A (en) 1985-01-03
AU566670B2 (en) 1987-10-29
ZA844669B (en) 1985-08-28
JPS6013792A (ja) 1985-01-24
EP0129247A1 (en) 1984-12-27
US4483987A (en) 1984-11-20

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