JPH0447672B2 - - Google Patents
Info
- Publication number
- JPH0447672B2 JPH0447672B2 JP58163392A JP16339283A JPH0447672B2 JP H0447672 B2 JPH0447672 B2 JP H0447672B2 JP 58163392 A JP58163392 A JP 58163392A JP 16339283 A JP16339283 A JP 16339283A JP H0447672 B2 JPH0447672 B2 JP H0447672B2
- Authority
- JP
- Japan
- Prior art keywords
- formula
- alkoxy
- carboxy
- dihydro
- pyrrolo
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB8225582 | 1982-09-08 | ||
| GB8225582 | 1982-09-08 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS5965093A JPS5965093A (ja) | 1984-04-13 |
| JPH0447672B2 true JPH0447672B2 (enExample) | 1992-08-04 |
Family
ID=10532762
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP58163392A Granted JPS5965093A (ja) | 1982-09-08 | 1983-09-07 | ピロロジアゼピン誘導体 |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US4508730A (enExample) |
| EP (1) | EP0102602B1 (enExample) |
| JP (1) | JPS5965093A (enExample) |
| KR (1) | KR910000417B1 (enExample) |
| AT (1) | ATE51230T1 (enExample) |
| AU (1) | AU566404B2 (enExample) |
| CA (1) | CA1199633A (enExample) |
| DE (1) | DE3381355D1 (enExample) |
| DK (1) | DK161077C (enExample) |
| ES (2) | ES8503000A1 (enExample) |
| GR (1) | GR79626B (enExample) |
| IE (1) | IE56043B1 (enExample) |
| IL (1) | IL69473A (enExample) |
| ZA (1) | ZA835899B (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS60208488A (ja) * | 1984-04-03 | 1985-10-21 | Nippon Mining Co Ltd | スラグからの有価金属の回収法 |
| JP2016513117A (ja) | 2013-02-22 | 2016-05-12 | バイエル ファーマ アクチエンゲゼルシャフト | 過剰増殖性疾患を治療するためのbetタンパク質阻害剤としてのピロロ−およびピラゾロ−トリアゾロジアゼピン類 |
| HK1212345A1 (en) | 2013-02-22 | 2016-06-10 | Bayer Pharma Aktiengesellschaft | 4-substituted pyrrolo- and pyrazolo-diazepines |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3553207A (en) * | 1968-12-16 | 1971-01-05 | Parke Davis & Co | Phenylpyrazolodiazepinone compounds |
| US3553210A (en) * | 1968-12-16 | 1971-01-05 | Parke Davis & Co | 3-methyl-8-phenylpyrazolo(4,3-e)(1,4)diazepin-5(1h)-one, 7-oxide compounds |
| GB1433103A (en) * | 1974-03-20 | 1976-04-22 | Lepetit Spa | Pharmacologically active pyrrolodiazepines |
| GR76455B (enExample) * | 1981-06-04 | 1984-08-10 | Lepetit Spa | |
| IT1167788B (it) * | 1981-06-08 | 1987-05-13 | Lepetit Spa | Derivati pirrolo-diazepinici |
-
1983
- 1983-08-09 US US06/521,774 patent/US4508730A/en not_active Expired - Fee Related
- 1983-08-11 AU AU17900/83A patent/AU566404B2/en not_active Ceased
- 1983-08-11 ZA ZA835899A patent/ZA835899B/xx unknown
- 1983-08-12 IL IL69473A patent/IL69473A/xx unknown
- 1983-08-27 AT AT83108446T patent/ATE51230T1/de not_active IP Right Cessation
- 1983-08-27 EP EP83108446A patent/EP0102602B1/en not_active Expired - Lifetime
- 1983-08-27 DE DE8383108446T patent/DE3381355D1/de not_active Expired - Lifetime
- 1983-08-29 GR GR72324A patent/GR79626B/el unknown
- 1983-08-30 DK DK394483A patent/DK161077C/da active
- 1983-09-07 ES ES525442A patent/ES8503000A1/es not_active Expired
- 1983-09-07 IE IE2098/83A patent/IE56043B1/en not_active IP Right Cessation
- 1983-09-07 JP JP58163392A patent/JPS5965093A/ja active Granted
- 1983-09-07 CA CA000436167A patent/CA1199633A/en not_active Expired
- 1983-09-08 KR KR1019830004230A patent/KR910000417B1/ko not_active Expired
-
1984
- 1984-05-14 ES ES532487A patent/ES532487A0/es active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| AU566404B2 (en) | 1987-10-22 |
| US4508730A (en) | 1985-04-02 |
| IL69473A (en) | 1985-12-31 |
| ES525442A0 (es) | 1985-02-01 |
| EP0102602B1 (en) | 1990-03-21 |
| GR79626B (enExample) | 1984-10-31 |
| DK161077C (da) | 1991-11-18 |
| EP0102602A1 (en) | 1984-03-14 |
| JPS5965093A (ja) | 1984-04-13 |
| KR910000417B1 (ko) | 1991-01-25 |
| IE832098L (en) | 1984-03-08 |
| CA1199633A (en) | 1986-01-21 |
| ES8507551A1 (es) | 1985-09-01 |
| DK394483D0 (da) | 1983-08-30 |
| ATE51230T1 (de) | 1990-04-15 |
| KR840006248A (ko) | 1984-11-22 |
| DK394483A (da) | 1984-03-09 |
| ES8503000A1 (es) | 1985-02-01 |
| DE3381355D1 (de) | 1990-04-26 |
| IE56043B1 (en) | 1991-03-27 |
| ES532487A0 (es) | 1985-09-01 |
| IL69473A0 (en) | 1983-11-30 |
| ZA835899B (en) | 1984-07-25 |
| DK161077B (da) | 1991-05-27 |
| AU1790083A (en) | 1984-03-15 |
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