JP7619730B2 - アルキルシリルオキシ置換ベンジルアミン化合物の製造方法 - Google Patents
アルキルシリルオキシ置換ベンジルアミン化合物の製造方法 Download PDFInfo
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- JP7619730B2 JP7619730B2 JP2024508080A JP2024508080A JP7619730B2 JP 7619730 B2 JP7619730 B2 JP 7619730B2 JP 2024508080 A JP2024508080 A JP 2024508080A JP 2024508080 A JP2024508080 A JP 2024508080A JP 7619730 B2 JP7619730 B2 JP 7619730B2
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- carbon atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B61/00—Other general methods
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C249/00—Preparation of compounds containing nitrogen atoms doubly-bound to a carbon skeleton
- C07C249/02—Preparation of compounds containing nitrogen atoms doubly-bound to a carbon skeleton of compounds containing imino groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
- C07C251/02—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton containing imino groups
- C07C251/04—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton containing imino groups having carbon atoms of imino groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C251/10—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton containing imino groups having carbon atoms of imino groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton
- C07C251/16—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton containing imino groups having carbon atoms of imino groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton containing six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C269/04—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups from amines with formation of carbamate groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C271/06—Esters of carbamic acids
- C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
- C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C271/12—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2022155408 | 2022-09-28 | ||
| JP2022155408 | 2022-09-28 | ||
| PCT/JP2023/035097 WO2024071178A1 (ja) | 2022-09-28 | 2023-09-27 | アルキルシリルオキシ置換ベンジルアミン化合物の製造方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JPWO2024071178A1 JPWO2024071178A1 (https=) | 2024-04-04 |
| JPWO2024071178A5 JPWO2024071178A5 (https=) | 2024-09-05 |
| JP7619730B2 true JP7619730B2 (ja) | 2025-01-22 |
Family
ID=90477826
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024508080A Active JP7619730B2 (ja) | 2022-09-28 | 2023-09-27 | アルキルシリルオキシ置換ベンジルアミン化合物の製造方法 |
Country Status (4)
| Country | Link |
|---|---|
| JP (1) | JP7619730B2 (https=) |
| CN (1) | CN119948011A (https=) |
| TW (1) | TW202419441A (https=) |
| WO (1) | WO2024071178A1 (https=) |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20150010469A1 (en) | 2013-07-03 | 2015-01-08 | British Columbia Cancer Agency Branch | Bisphenol ether compounds with novel bridging groups and methods for their use |
| WO2019208043A1 (ja) | 2018-04-24 | 2019-10-31 | 国立大学法人九州大学 | 窒素上無保護イミン化合物の製造方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2998885C (en) * | 2015-09-24 | 2020-09-01 | Cyclenium Pharma Inc. | Libraries of heteroaryl-containing macrocyclic compounds and methods of making and using the same |
| JP7063408B1 (ja) * | 2021-07-02 | 2022-05-09 | ペプチスター株式会社 | 液相ペプチド製造方法 |
| JP2025001050A (ja) * | 2021-09-01 | 2025-01-08 | 積水メディカル株式会社 | ガニレリクス又はその塩の製造法 |
| JP2025001049A (ja) * | 2021-09-01 | 2025-01-08 | 積水メディカル株式会社 | アルギニン誘導体 |
-
2023
- 2023-09-27 CN CN202380069012.7A patent/CN119948011A/zh active Pending
- 2023-09-27 WO PCT/JP2023/035097 patent/WO2024071178A1/ja not_active Ceased
- 2023-09-27 JP JP2024508080A patent/JP7619730B2/ja active Active
- 2023-09-28 TW TW112137270A patent/TW202419441A/zh unknown
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20150010469A1 (en) | 2013-07-03 | 2015-01-08 | British Columbia Cancer Agency Branch | Bisphenol ether compounds with novel bridging groups and methods for their use |
| WO2019208043A1 (ja) | 2018-04-24 | 2019-10-31 | 国立大学法人九州大学 | 窒素上無保護イミン化合物の製造方法 |
Non-Patent Citations (3)
| Title |
|---|
| CAS REGISTRY No. 1420067-97-5, 807308-57-2, 790602-34-5, 754129-25-4, 729550-05-4，DATABASE REGISTRY, [online]，2013年，[検索日: 2023.11.14], retrieved from: STN |
| CAS REGISTRY No. 2770500-65-5, 2764021-24-9, 2764016-02-4, 2764005-95-8，DATABASE REGISTRY, [online]，2022年06月05日，[検索日: 2023.11.14], retrieved from: STN |
| KONDO, Y. et al.，A Convenient Preparation Method for Benzophenone Imine Catalyzed by Tetrabutylammonium Fluoride，Organic Process Research & Development，2019年，Vol. 23, No. 8，pp. 1718-1724，DOI: 10.1021/acs.oprd.9b00226 |
Also Published As
| Publication number | Publication date |
|---|---|
| CN119948011A (zh) | 2025-05-06 |
| TW202419441A (zh) | 2024-05-16 |
| WO2024071178A1 (ja) | 2024-04-04 |
| JPWO2024071178A1 (https=) | 2024-04-04 |
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