JP7270901B2 - 男性の避妊のための非ホルモン性組成物および方法 - Google Patents
男性の避妊のための非ホルモン性組成物および方法 Download PDFInfo
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- JP7270901B2 JP7270901B2 JP2021500350A JP2021500350A JP7270901B2 JP 7270901 B2 JP7270901 B2 JP 7270901B2 JP 2021500350 A JP2021500350 A JP 2021500350A JP 2021500350 A JP2021500350 A JP 2021500350A JP 7270901 B2 JP7270901 B2 JP 7270901B2
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
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- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
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| PCT/EP2019/057267 WO2019180217A1 (en) | 2018-03-23 | 2019-03-22 | Non-hormonal compositions and methods for male contraception |
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| JP2021518438A5 JP2021518438A5 (https=) | 2022-03-30 |
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| IL319287A (en) | 2022-11-23 | 2025-04-01 | Pharmajor Incorporated | Silodosin formulations with different release and their use in male contraceptive methods |
Citations (1)
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| US20080242717A1 (en) | 2007-02-28 | 2008-10-02 | Fumiyasu Sato | Methods for treating benign prostatic hyperplasia |
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| US1091276A (en) | 1911-12-09 | 1914-03-24 | Basf Ag | Producing unsaturated terpene hydrocarbons. |
| US4210644A (en) | 1978-02-23 | 1980-07-01 | The Johns Hopkins University | Male contraception |
| DE4308406C1 (de) | 1993-03-12 | 1994-06-16 | Jenapharm Gmbh | Kombinationspräparat zur Kontrazeption |
| ATE474580T1 (de) | 2000-02-15 | 2010-08-15 | Bayer Schering Pharma Ag | Zusammensetzung zur männlichen kontrazeption, norethisteron enthaltend |
| FR2861990B1 (fr) * | 2003-11-10 | 2006-02-10 | Nouveaux Produits Pharma | Comprimes faiblement doses a reseau de polymeres |
| UA95085C2 (ru) * | 2005-09-29 | 2011-07-11 | Баер Шеринг Фарма Акциенгезельшафт | Применение варденафила для лечения урологических расстройств |
| JP2009509984A (ja) * | 2005-09-29 | 2009-03-12 | バイエル・ヘルスケア・アクチェンゲゼルシャフト | 泌尿器系障害の処置用のｐｄｅ阻害剤およびそれらの組合せ |
| US20100098735A1 (en) * | 2006-10-05 | 2010-04-22 | Rajesh Jain | Injectable depot compositions and its process of preparation |
| GB0700893D0 (en) | 2007-01-17 | 2007-02-21 | King S College London | Male contraceptive |
| US20120184591A1 (en) * | 2011-01-13 | 2012-07-19 | Watson Pharmaceuticals, Inc. | Methods for treating prostatitis |
| CN102283816B (zh) * | 2011-08-05 | 2013-09-11 | 北京海步国际医药科技发展有限公司 | 西洛多辛缓释片剂及其制备方法 |
| WO2014118606A2 (en) * | 2013-01-29 | 2014-08-07 | Alembic Pharmaceuticals Limited | A novel process for the preparation of silodosin |
| WO2016051782A1 (ja) | 2014-09-30 | 2016-04-07 | キッセイ薬品工業株式会社 | 苦味を有する薬剤の苦味をマスキングした経口投与製剤 |
| US20170049834A1 (en) * | 2015-08-18 | 2017-02-23 | Golden Biotechnology Corporation | Benign prostatic hyperplasia add-on therapy |
| EP3750538B1 (en) * | 2018-03-23 | 2024-08-14 | Pharmajor International | Non-hormonal methods for male contraception comprising (r)-silodosin |
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Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20080242717A1 (en) | 2007-02-28 | 2008-10-02 | Fumiyasu Sato | Methods for treating benign prostatic hyperplasia |
Non-Patent Citations (6)
| Title |
|---|
| Andrology，2015年，Vol.3，pp.1076-1081 |
| Contraception，1988年，Vol.37, No.6，pp.621-629 |
| Indian Journal of Urology，2018年01月01日，Vol.34, Supplement 1，p.S7, Abstract No.BKP02 |
| International Journal of Impotence Research，2009年，Vol.21，pp.306-310 |
| Medical Hypotheses，2009年，Vol.73，pp.140-141 |
| Urology，2012年，Vol.80，pp.614-617 |
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