MX2020009937A - Uso de una composición no hormonal para sujetos masculinos, que comprende el antagonista del adrenorreceptor alfa-1: (r)- silodosina para inducir aspermia y azoospermia u oligozoospermia suficiente para lograr un efecto anticonceptivo. - Google Patents
Uso de una composición no hormonal para sujetos masculinos, que comprende el antagonista del adrenorreceptor alfa-1: (r)- silodosina para inducir aspermia y azoospermia u oligozoospermia suficiente para lograr un efecto anticonceptivo.Info
- Publication number
- MX2020009937A MX2020009937A MX2020009937A MX2020009937A MX2020009937A MX 2020009937 A MX2020009937 A MX 2020009937A MX 2020009937 A MX2020009937 A MX 2020009937A MX 2020009937 A MX2020009937 A MX 2020009937A MX 2020009937 A MX2020009937 A MX 2020009937A
- Authority
- MX
- Mexico
- Prior art keywords
- composition
- contraception
- methods
- once daily
- male contraception
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 4
- 238000000034 method Methods 0.000 title abstract 3
- 206010003883 azoospermia Diseases 0.000 abstract 2
- 229940122878 Alpha 1 adrenoreceptor antagonist Drugs 0.000 abstract 1
- 206010003495 Aspermia Diseases 0.000 abstract 1
- 230000003054 hormonal effect Effects 0.000 abstract 1
- 230000001771 impaired effect Effects 0.000 abstract 1
- 208000008634 oligospermia Diseases 0.000 abstract 1
- 238000004806 packaging method and process Methods 0.000 abstract 1
- 230000002441 reversible effect Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/4045—Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/16—Masculine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Physiology (AREA)
- Nutrition Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862763129P | 2018-03-23 | 2018-03-23 | |
| EP18305328 | 2018-03-23 | ||
| PCT/EP2019/057267 WO2019180217A1 (en) | 2018-03-23 | 2019-03-22 | Non-hormonal compositions and methods for male contraception |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2020009937A true MX2020009937A (es) | 2022-09-30 |
Family
ID=65955198
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2020009937A MX2020009937A (es) | 2018-03-23 | 2019-03-22 | Uso de una composición no hormonal para sujetos masculinos, que comprende el antagonista del adrenorreceptor alfa-1: (r)- silodosina para inducir aspermia y azoospermia u oligozoospermia suficiente para lograr un efecto anticonceptivo. |
Country Status (19)
| Country | Link |
|---|---|
| US (3) | US10912762B2 (https=) |
| EP (2) | EP3750538B1 (https=) |
| JP (1) | JP7270901B2 (https=) |
| KR (1) | KR102496504B1 (https=) |
| CN (1) | CN112074269A (https=) |
| AU (1) | AU2019237228B2 (https=) |
| BR (1) | BR112020018925A2 (https=) |
| CA (1) | CA3094016C (https=) |
| DK (2) | DK3562485T3 (https=) |
| ES (2) | ES2989170T3 (https=) |
| FI (1) | FI3750538T3 (https=) |
| IL (1) | IL277372B2 (https=) |
| MA (1) | MA53626B1 (https=) |
| MX (1) | MX2020009937A (https=) |
| PL (2) | PL3562485T3 (https=) |
| PT (1) | PT3562485T (https=) |
| SG (1) | SG11202008794TA (https=) |
| UA (1) | UA128502C2 (https=) |
| WO (1) | WO2019180217A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3750538B1 (en) * | 2018-03-23 | 2024-08-14 | Pharmajor International | Non-hormonal methods for male contraception comprising (r)-silodosin |
| IL319287A (en) | 2022-11-23 | 2025-04-01 | Pharmajor Incorporated | Silodosin formulations with different release and their use in male contraceptive methods |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US1091276A (en) | 1911-12-09 | 1914-03-24 | Basf Ag | Producing unsaturated terpene hydrocarbons. |
| US4210644A (en) | 1978-02-23 | 1980-07-01 | The Johns Hopkins University | Male contraception |
| DE4308406C1 (de) | 1993-03-12 | 1994-06-16 | Jenapharm Gmbh | Kombinationspräparat zur Kontrazeption |
| ATE474580T1 (de) | 2000-02-15 | 2010-08-15 | Bayer Schering Pharma Ag | Zusammensetzung zur männlichen kontrazeption, norethisteron enthaltend |
| FR2861990B1 (fr) * | 2003-11-10 | 2006-02-10 | Nouveaux Produits Pharma | Comprimes faiblement doses a reseau de polymeres |
| UA95085C2 (ru) * | 2005-09-29 | 2011-07-11 | Баер Шеринг Фарма Акциенгезельшафт | Применение варденафила для лечения урологических расстройств |
| JP2009509984A (ja) * | 2005-09-29 | 2009-03-12 | バイエル・ヘルスケア・アクチェンゲゼルシャフト | 泌尿器系障害の処置用のｐｄｅ阻害剤およびそれらの組合せ |
| US20100098735A1 (en) * | 2006-10-05 | 2010-04-22 | Rajesh Jain | Injectable depot compositions and its process of preparation |
| GB0700893D0 (en) | 2007-01-17 | 2007-02-21 | King S College London | Male contraceptive |
| MX2009009230A (es) | 2007-02-28 | 2009-11-26 | Kissei Pharmaceutical | Uso de silodosina en una administracion diaria para tratar hiperplasia prostatica benigna. |
| US20120184591A1 (en) * | 2011-01-13 | 2012-07-19 | Watson Pharmaceuticals, Inc. | Methods for treating prostatitis |
| CN102283816B (zh) * | 2011-08-05 | 2013-09-11 | 北京海步国际医药科技发展有限公司 | 西洛多辛缓释片剂及其制备方法 |
| WO2014118606A2 (en) * | 2013-01-29 | 2014-08-07 | Alembic Pharmaceuticals Limited | A novel process for the preparation of silodosin |
| WO2016051782A1 (ja) | 2014-09-30 | 2016-04-07 | キッセイ薬品工業株式会社 | 苦味を有する薬剤の苦味をマスキングした経口投与製剤 |
| US20170049834A1 (en) * | 2015-08-18 | 2017-02-23 | Golden Biotechnology Corporation | Benign prostatic hyperplasia add-on therapy |
| EP3750538B1 (en) * | 2018-03-23 | 2024-08-14 | Pharmajor International | Non-hormonal methods for male contraception comprising (r)-silodosin |
-
2019
- 2019-03-22 EP EP20182691.4A patent/EP3750538B1/en active Active
- 2019-03-22 US US16/362,081 patent/US10912762B2/en active Active
- 2019-03-22 FI FIEP20182691.4T patent/FI3750538T3/fi active
- 2019-03-22 WO PCT/EP2019/057267 patent/WO2019180217A1/en not_active Ceased
- 2019-03-22 KR KR1020207029031A patent/KR102496504B1/ko active Active
- 2019-03-22 AU AU2019237228A patent/AU2019237228B2/en active Active
- 2019-03-22 IL IL277372A patent/IL277372B2/en unknown
- 2019-03-22 PT PT197141500T patent/PT3562485T/pt unknown
- 2019-03-22 MA MA53626A patent/MA53626B1/fr unknown
- 2019-03-22 SG SG11202008794TA patent/SG11202008794TA/en unknown
- 2019-03-22 CA CA3094016A patent/CA3094016C/en active Active
- 2019-03-22 PL PL19714150T patent/PL3562485T3/pl unknown
- 2019-03-22 CN CN201980030077.4A patent/CN112074269A/zh active Pending
- 2019-03-22 ES ES20182691T patent/ES2989170T3/es active Active
- 2019-03-22 MX MX2020009937A patent/MX2020009937A/es unknown
- 2019-03-22 ES ES19714150T patent/ES2813084T3/es active Active
- 2019-03-22 JP JP2021500350A patent/JP7270901B2/ja active Active
- 2019-03-22 EP EP19714150.0A patent/EP3562485B8/en active Active
- 2019-03-22 DK DK19714150.0T patent/DK3562485T3/da active
- 2019-03-22 PL PL20182691.4T patent/PL3750538T3/pl unknown
- 2019-03-22 DK DK20182691.4T patent/DK3750538T3/da active
- 2019-03-22 BR BR112020018925-1A patent/BR112020018925A2/pt unknown
- 2019-03-22 UA UAA202006637A patent/UA128502C2/uk unknown
-
2020
- 2020-12-30 US US17/137,747 patent/US11583518B2/en active Active
-
2023
- 2023-01-06 US US18/093,940 patent/US11951095B2/en active Active
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